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HN2010001235A - Sales farmaceuticas aceptables de (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihodro-9h-purin-9-il)propil](3-morfolin-4-ilpropil)amino]metil]fenil)acetato de metilo y sus usos en terapia - Google Patents

Sales farmaceuticas aceptables de (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihodro-9h-purin-9-il)propil](3-morfolin-4-ilpropil)amino]metil]fenil)acetato de metilo y sus usos en terapia

Info

Publication number
HN2010001235A
HN2010001235A HN2010001235A HN2010001235A HN2010001235A HN 2010001235 A HN2010001235 A HN 2010001235A HN 2010001235 A HN2010001235 A HN 2010001235A HN 2010001235 A HN2010001235 A HN 2010001235A HN 2010001235 A HN2010001235 A HN 2010001235A
Authority
HN
Honduras
Prior art keywords
amino
methyl
purin
oxo
therapy
Prior art date
Application number
HN2010001235A
Other languages
English (en)
Inventor
Mcinally Thomas
Schulz Hakan
Original Assignee
Astrazeneca
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40795767&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HN2010001235(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca filed Critical Astrazeneca
Publication of HN2010001235A publication Critical patent/HN2010001235A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Abstract

LA PRESENTE INVENCION SE RELACIONA CON SALES DE CLORHIDRATO, BROMHIDRATO O MALETO ACIDO HIDROCLORICO, HIDROBROMICO Y MALEICO DE (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihidro-9h-purin-9-il)propil)](3-morfolin-4-ilpropil)amino]metil}fenil)acetato de metilo COMPOSICIONES FARMACEUTICAS QUE LAS CONTIENEN Y SU USO EN TERAPIA.
HN2010001235A 2007-12-17 2010-06-17 Sales farmaceuticas aceptables de (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihodro-9h-purin-9-il)propil](3-morfolin-4-ilpropil)amino]metil]fenil)acetato de metilo y sus usos en terapia HN2010001235A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1416407P 2007-12-17 2007-12-17

Publications (1)

Publication Number Publication Date
HN2010001235A true HN2010001235A (es) 2013-02-11

Family

ID=40795767

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2010001235A HN2010001235A (es) 2007-12-17 2010-06-17 Sales farmaceuticas aceptables de (3-{[[3-(6-amino-2-butoxi-8-oxo-7,8-dihodro-9h-purin-9-il)propil](3-morfolin-4-ilpropil)amino]metil]fenil)acetato de metilo y sus usos en terapia

Country Status (26)

Country Link
US (1) US8673907B2 (es)
EP (1) EP2235018A4 (es)
JP (1) JP5557748B2 (es)
KR (2) KR20100093566A (es)
CN (1) CN101903389B (es)
AR (1) AR069780A1 (es)
AU (1) AU2008339095B2 (es)
BR (1) BRPI0821020A2 (es)
CA (1) CA2709126C (es)
CL (1) CL2008003750A1 (es)
CO (1) CO6280403A2 (es)
CR (1) CR11507A (es)
CU (1) CU23932B1 (es)
EA (1) EA017532B1 (es)
EC (1) ECSP10010265A (es)
HN (1) HN2010001235A (es)
IL (1) IL206039A0 (es)
NI (1) NI201000104A (es)
NZ (1) NZ585961A (es)
PE (1) PE20091156A1 (es)
SV (1) SV2010003596A (es)
TW (1) TWI424848B (es)
UA (1) UA100996C2 (es)
UY (1) UY31531A1 (es)
WO (1) WO2009078798A1 (es)
ZA (1) ZA201003877B (es)

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* Cited by examiner, † Cited by third party
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MXPA06011080A (es) 2004-03-26 2007-04-16 Astrazeneca Ab Compuesto de 8-oxoadenina 9-sustituido.
TW200831105A (en) 2006-12-14 2008-08-01 Astrazeneca Ab Novel compounds
WO2008114006A1 (en) 2007-03-19 2008-09-25 Astrazeneca Ab 9-substituted-8-oxo-adenine compounds as toll-like receptor (tlr7) modulators
US8067413B2 (en) 2007-03-19 2011-11-29 Astrazeneca Ab 9-substituted-8-oxo-adenine compounds as toll-like receptor (TLR7 ) modulators
WO2008114819A1 (ja) 2007-03-20 2008-09-25 Dainippon Sumitomo Pharma Co., Ltd. 新規アデニン化合物
PE20091236A1 (es) 2007-11-22 2009-09-16 Astrazeneca Ab Derivados de pirimidina como immunomoduladores de tlr7
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