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HN2008000646A - Antagonistas de los receptores 2 de dopamina de rapida disociacion - Google Patents

Antagonistas de los receptores 2 de dopamina de rapida disociacion

Info

Publication number
HN2008000646A
HN2008000646A HN2008000646A HN2008000646A HN2008000646A HN 2008000646 A HN2008000646 A HN 2008000646A HN 2008000646 A HN2008000646 A HN 2008000646A HN 2008000646 A HN2008000646 A HN 2008000646A HN 2008000646 A HN2008000646 A HN 2008000646A
Authority
HN
Honduras
Prior art keywords
rapida
antagonists
disociacion
dopamine
receptors
Prior art date
Application number
HN2008000646A
Other languages
English (en)
Inventor
Franz Leopold Marcel
James Macdonald Gregor
Edmond Josephine Kennis Ludo
Jean Michael Langlois Xavier
Alfons Maria Van Den Keybus Frans
Emiel Maria Van Roosbroeck Yves
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HN2008000646A publication Critical patent/HN2008000646A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A COMPUESTOS QUE SON ANTAGONISTAS DE LOS RECEPTORES 2 DE DOPAMIMNA DE RAPIDA DISOCIACION A PROCESOS PARA PREPARAR DICHOS COMPUESTOS Y A COMPOSICIONES FARMACEUTICA QUE COMPRENDEN DICHOS COMPUESTOS COMO INGREDIENTE ACTIVO.
HN2008000646A 2005-10-26 2008-04-23 Antagonistas de los receptores 2 de dopamina de rapida disociacion HN2008000646A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05110028 2005-10-26

Publications (1)

Publication Number Publication Date
HN2008000646A true HN2008000646A (es) 2011-02-16

Family

ID=35734993

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2008000646A HN2008000646A (es) 2005-10-26 2008-04-23 Antagonistas de los receptores 2 de dopamina de rapida disociacion

Country Status (34)

Country Link
US (3) US8940743B2 (es)
EP (1) EP1943242B1 (es)
JP (1) JP5140598B2 (es)
KR (1) KR101351910B1 (es)
CN (1) CN101291925B (es)
AP (1) AP2607A (es)
AR (1) AR058151A1 (es)
AT (1) ATE495167T1 (es)
AU (1) AU2006307930B2 (es)
BR (1) BRPI0617787A2 (es)
CA (1) CA2623160C (es)
CR (1) CR10020A (es)
CY (1) CY1111977T1 (es)
DE (1) DE602006019624D1 (es)
DK (1) DK1943242T3 (es)
EA (1) EA015681B1 (es)
EC (1) ECSP088396A (es)
ES (1) ES2359020T3 (es)
GT (1) GT200800033A (es)
HN (1) HN2008000646A (es)
HR (1) HRP20110226T1 (es)
IL (1) IL191016A (es)
JO (1) JO2769B1 (es)
MY (1) MY145609A (es)
NO (1) NO20082350L (es)
NZ (1) NZ566785A (es)
PL (1) PL1943242T3 (es)
PT (1) PT1943242E (es)
RS (1) RS51674B (es)
SI (1) SI1943242T1 (es)
TW (1) TWI399373B (es)
UA (1) UA94058C2 (es)
WO (1) WO2007048779A1 (es)
ZA (1) ZA200803668B (es)

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Also Published As

Publication number Publication date
ZA200803668B (en) 2009-09-30
DK1943242T3 (da) 2011-04-26
SI1943242T1 (sl) 2011-05-31
US20170022181A1 (en) 2017-01-26
PL1943242T3 (pl) 2011-06-30
EA200801184A1 (ru) 2008-08-29
HK1124317A1 (en) 2009-07-10
DE602006019624D1 (de) 2011-02-24
JP5140598B2 (ja) 2013-02-06
ATE495167T1 (de) 2011-01-15
US9751860B2 (en) 2017-09-05
ECSP088396A (es) 2008-05-30
CN101291925B (zh) 2013-04-10
TWI399373B (zh) 2013-06-21
AP2607A (en) 2013-03-05
JP2009514815A (ja) 2009-04-09
CA2623160A1 (en) 2007-05-03
AU2006307930B2 (en) 2011-10-06
BRPI0617787A2 (pt) 2009-12-01
HRP20110226T1 (hr) 2011-05-31
EA015681B1 (ru) 2011-10-31
IL191016A (en) 2013-10-31
WO2007048779A1 (en) 2007-05-03
US8940743B2 (en) 2015-01-27
AR058151A1 (es) 2008-01-23
UA94058C2 (ru) 2011-04-11
EP1943242B1 (en) 2011-01-12
ES2359020T3 (es) 2011-05-17
CA2623160C (en) 2013-10-15
TW200732321A (en) 2007-09-01
NZ566785A (en) 2010-03-26
CY1111977T1 (el) 2015-11-04
KR101351910B1 (ko) 2014-01-16
NO20082350L (no) 2008-07-01
RS51674B (sr) 2011-10-31
PT1943242E (pt) 2011-04-06
US20150141432A1 (en) 2015-05-21
US9468640B2 (en) 2016-10-18
AU2006307930A1 (en) 2007-05-03
KR20080067658A (ko) 2008-07-21
AP2008004441A0 (en) 2008-04-30
GT200800033A (es) 2009-08-20
CN101291925A (zh) 2008-10-22
US20080227791A1 (en) 2008-09-18
MY145609A (en) 2012-03-15
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EP1943242A1 (en) 2008-07-16
CR10020A (es) 2009-01-16

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