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HK1181775B - 含磷活性物质的立体有择合成 - Google Patents

含磷活性物质的立体有择合成 Download PDF

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Publication number
HK1181775B
HK1181775B HK13109048.8A HK13109048A HK1181775B HK 1181775 B HK1181775 B HK 1181775B HK 13109048 A HK13109048 A HK 13109048A HK 1181775 B HK1181775 B HK 1181775B
Authority
HK
Hong Kong
Prior art keywords
compound
mixture
group
mmol
alkyl
Prior art date
Application number
HK13109048.8A
Other languages
German (de)
English (en)
French (fr)
Other versions
HK1181775A1 (zh
Inventor
Bruce S. Ross
Michael Joseph Sofia
Ganapati Reddy Pamulapati
Suguna Rachakonda
Hai-Ren Zhang
Original Assignee
Gilead Pharmasset Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Pharmasset Llc filed Critical Gilead Pharmasset Llc
Priority claimed from PCT/US2011/030762 external-priority patent/WO2011123668A2/en
Publication of HK1181775A1 publication Critical patent/HK1181775A1/zh
Publication of HK1181775B publication Critical patent/HK1181775B/zh

Links

HK13109048.8A 2010-03-31 2011-03-31 含磷活性物质的立体有择合成 HK1181775B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US31951310P 2010-03-31 2010-03-31
US31954810P 2010-03-31 2010-03-31
US319513P 2010-03-31
US319548P 2010-03-31
PCT/US2011/030762 WO2011123668A2 (en) 2010-03-31 2011-03-31 Stereoselective synthesis of phosphorus containing actives

Publications (2)

Publication Number Publication Date
HK1181775A1 HK1181775A1 (zh) 2013-11-15
HK1181775B true HK1181775B (zh) 2015-06-19

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