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HK1178882A1 - 作为btk激酶抑制剂的羟基嘌呤衍生物 - Google Patents

作为btk激酶抑制剂的羟基嘌呤衍生物 Download PDF

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Publication number
HK1178882A1
HK1178882A1 HK13105581.9A HK13105581A HK1178882A1 HK 1178882 A1 HK1178882 A1 HK 1178882A1 HK 13105581 A HK13105581 A HK 13105581A HK 1178882 A1 HK1178882 A1 HK 1178882A1
Authority
HK
Hong Kong
Prior art keywords
group
amino
dihydro
purin
phenoxyphenyl
Prior art date
Application number
HK13105581.9A
Other languages
English (en)
Other versions
HK1178882B (zh
Inventor
Yamamoto Shingo
Yoshizawa Toshio
Original Assignee
Ono Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ono Pharmaceutical Co., Ltd. filed Critical Ono Pharmaceutical Co., Ltd.
Publication of HK1178882A1 publication Critical patent/HK1178882A1/zh
Publication of HK1178882B publication Critical patent/HK1178882B/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • A61K31/522Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK13105581.9A 2010-05-31 2011-05-30 作为btk激酶抑制剂的羟基嘌呤衍生物 HK1178882B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010-123727 2010-05-31
JP2010123727 2010-05-31
PCT/JP2011/062377 WO2011152351A1 (ja) 2010-05-31 2011-05-30 プリノン誘導体

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
HK17105517.4A Division HK1231869B (zh) 2010-05-31 2013-05-09 嘌呤衍生物作为btk激酶抑制剂

Related Child Applications (1)

Application Number Title Priority Date Filing Date
HK17105517.4A Addition HK1231869B (zh) 2010-05-31 2013-05-09 嘌呤衍生物作为btk激酶抑制剂

Publications (2)

Publication Number Publication Date
HK1178882A1 true HK1178882A1 (zh) 2013-09-19
HK1178882B HK1178882B (zh) 2017-08-18

Family

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Also Published As

Publication number Publication date
KR20130109941A (ko) 2013-10-08
HRP20161027T1 (hr) 2016-11-04
CN102918040A (zh) 2013-02-06
TW201209057A (en) 2012-03-01
JP5648686B2 (ja) 2015-01-07
EP2578585A4 (en) 2013-10-23
PH12012502369A1 (en) 2013-02-11
US20200048256A1 (en) 2020-02-13
US20130079327A1 (en) 2013-03-28
MY189483A (en) 2022-02-16
EP3590938A1 (en) 2020-01-08
JP2016185954A (ja) 2016-10-27
TW201533046A (zh) 2015-09-01
US20240083899A1 (en) 2024-03-14
CN102918040B (zh) 2015-03-18
KR101537148B1 (ko) 2015-07-15
EP3112368A1 (en) 2017-01-04
AU2011260961B9 (en) 2015-02-26
TWI500617B (zh) 2015-09-21
NZ603643A (en) 2014-07-25
SMT201600360B (it) 2016-11-10
US9879013B2 (en) 2018-01-30
ZA201208900B (en) 2013-09-25
MY169745A (en) 2019-05-14
US10233185B2 (en) 2019-03-19
BR112012030711B1 (pt) 2020-10-13
WO2011152351A1 (ja) 2011-12-08
PT2578585T (pt) 2016-09-23
ES2782873T3 (es) 2020-09-16
US20250197401A1 (en) 2025-06-19
AU2011260961B2 (en) 2015-02-05
SI2578585T1 (sl) 2016-10-28
EP2578585B1 (en) 2016-07-20
US20130217880A1 (en) 2013-08-22
JP2015052000A (ja) 2015-03-19
LT2578585T (lt) 2016-10-10
EP3590938B1 (en) 2023-05-24
US9926322B2 (en) 2018-03-27
SG185617A1 (en) 2012-12-28
ES2592152T3 (es) 2016-11-28
EP3112368B1 (en) 2020-02-12
US20180170933A1 (en) 2018-06-21
SG10201503991SA (en) 2015-07-30
JP6176353B2 (ja) 2017-08-09
CY1118088T1 (el) 2017-06-28
CA2800523A1 (en) 2011-12-08
US20190169192A1 (en) 2019-06-06
JPWO2011152351A1 (ja) 2013-08-01
US20170313705A1 (en) 2017-11-02
MX2012013622A (es) 2013-02-01
BR112012030711A2 (pt) 2016-11-01
US8940725B2 (en) 2015-01-27
BR122018011748B1 (pt) 2021-12-07
RU2012157072A (ru) 2014-07-20
US20220363684A1 (en) 2022-11-17
IL223361A (en) 2015-11-30
DK2578585T3 (en) 2016-11-14
ES2948312T3 (es) 2023-09-08
TWI535716B (zh) 2016-06-01
RS55184B1 (sr) 2017-01-31
AU2011260961A1 (en) 2013-01-10
HUE030720T2 (en) 2017-06-28
CA2800523C (en) 2018-09-18
US8557803B2 (en) 2013-10-15
US10487085B2 (en) 2019-11-26
JP5924393B2 (ja) 2016-05-25
US20150094299A1 (en) 2015-04-02
PL2578585T3 (pl) 2017-01-31
EP2578585A1 (en) 2013-04-10

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