HK1042483B - 四氫噻唑的製造方法 - Google Patents

四氫噻唑的製造方法 Download PDF

Info

Publication number: HK1042483B
Authority: HK; Hong Kong
Prior art keywords: salts; thiazolidin; formula; production; reaction
Prior art date: 1999-06-10

Application number

HK02103306.1A

Other languages

German (de)

English (en)

French (fr)

Other versions

HK1042483A1 (zh

Inventor

Demuth Hans-Ulrich

Kruber Susanne

Original Assignee

Prosidion Limited

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-06-10

Filing date

2000-04-11

Publication date

2004-09-10

2000-04-11 Application filed by Prosidion Limited filed Critical Prosidion Limited

2002-08-16 Publication of HK1042483A1 publication Critical patent/HK1042483A1/zh

2004-09-10 Publication of HK1042483B publication Critical patent/HK1042483B/zh

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

HK02103306.1A 1999-06-10 2000-04-11 四氫噻唑的製造方法 HK1042483B (zh)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE19926233.0		1999-06-10
DE19926233A DE19926233C1 (de)	1999-06-10	1999-06-10	Verfahren zur Herstellung von Thiazolidin
PCT/EP2000/003213 WO2000076986A1 (de)	1999-06-10	2000-04-11	Verfahren zur herstellung von thiazolidin

Publications (2)

Publication Number	Publication Date
HK1042483A1 HK1042483A1 (zh)	2002-08-16
HK1042483B true HK1042483B (zh)	2004-09-10

Family

ID=7910641

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HK02103306.1A HK1042483B (zh)	1999-06-10	2000-04-11	四氫噻唑的製造方法

Country Status (18)

Country	Link
US (1)	US6559314B2 (zh)
EP (1)	EP1185520B1 (zh)
JP (1)	JP3803292B2 (zh)
KR (1)	KR100467898B1 (zh)
CN (1)	CN1169799C (zh)
AT (1)	ATE261946T1 (zh)
AU (1)	AU758605B2 (zh)
BR (1)	BR0011445A (zh)
CA (1)	CA2373834C (zh)
DE (2)	DE19926233C1 (zh)
DK (1)	DK1185520T3 (zh)
ES (1)	ES2215045T3 (zh)
HK (1)	HK1042483B (zh)
MX (1)	MXPA01012237A (zh)
NZ (1)	NZ515561A (zh)
PT (1)	PT1185520E (zh)
RU (1)	RU2218336C2 (zh)
WO (1)	WO2000076986A1 (zh)

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US7169926B1 (en)	2003-08-13	2007-01-30	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
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US7678909B1 (en)	2003-08-13	2010-03-16	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
EP1699777B1 (en)	2003-09-08	2012-12-12	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
US7732446B1 (en)	2004-03-11	2010-06-08	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
BRPI0418639B8 (pt)	2004-03-15	2021-05-25	Takeda Pharmaceutical	compostos inibidores de dipeptidil peptidase, assim como composição farmacêutica contendo os mesmos
US7687638B2 (en) *	2004-06-04	2010-03-30	Takeda San Diego, Inc.	Dipeptidyl peptidase inhibitors
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HRP20140091T4 (hr) *	2005-09-14	2021-12-24	Takeda Pharmaceutical Company Limited	Davanje inhibitora dipeptidil peptidaze
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TW200745079A (en) *	2005-09-16	2007-12-16	Takeda Pharmaceuticals Co	Polymorphs of benzoate salt of 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-benzonitrile and methods of use therefor
CN101360723A (zh)	2005-09-16	2009-02-04	武田药品工业株式会社	制备嘧啶二酮衍生物的方法
WO2007112347A1 (en)	2006-03-28	2007-10-04	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
US8460362B2 (en) *	2006-07-20	2013-06-11	Orbusneich Medical, Inc.	Bioabsorbable polymeric medical device
BRPI0716971A2 (pt) *	2006-09-13	2013-10-15	Takeda Pharmaceutical	Uso de 2-6(3-amino-piperini-l-il)-3-metil-2,4-dioxo-3,4-dihidro-2 h-pirimidin-1ilmetil-4-fluoro-benxonitrila
US8324383B2 (en)	2006-09-13	2012-12-04	Takeda Pharmaceutical Company Limited	Methods of making polymorphs of benzoate salt of 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-benzonitrile
TW200838536A (en)	2006-11-29	2008-10-01	Takeda Pharmaceutical	Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor
US8093236B2 (en)	2007-03-13	2012-01-10	Takeda Pharmaceuticals Company Limited	Weekly administration of dipeptidyl peptidase inhibitors
CN104910128A (zh) *	2015-06-02	2015-09-16	安徽兴东化工有限公司	一种2,2-二甲基四氢噻唑的制备方法

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1999
- 1999-06-10 DE DE19926233A patent/DE19926233C1/de not_active Expired - Lifetime
2000
- 2000-04-11 CA CA002373834A patent/CA2373834C/en not_active Expired - Fee Related
- 2000-04-11 DE DE50005699T patent/DE50005699D1/de not_active Expired - Lifetime
- 2000-04-11 MX MXPA01012237A patent/MXPA01012237A/es unknown
- 2000-04-11 EP EP00925194A patent/EP1185520B1/de not_active Expired - Lifetime
- 2000-04-11 RU RU2002100203/04A patent/RU2218336C2/ru not_active IP Right Cessation
- 2000-04-11 PT PT00925194T patent/PT1185520E/pt unknown
- 2000-04-11 JP JP2001503844A patent/JP3803292B2/ja not_active Expired - Fee Related
- 2000-04-11 NZ NZ515561A patent/NZ515561A/xx not_active IP Right Cessation
- 2000-04-11 CN CNB008087253A patent/CN1169799C/zh not_active Expired - Fee Related
- 2000-04-11 ES ES00925194T patent/ES2215045T3/es not_active Expired - Lifetime
- 2000-04-11 HK HK02103306.1A patent/HK1042483B/zh not_active IP Right Cessation
- 2000-04-11 WO PCT/EP2000/003213 patent/WO2000076986A1/de not_active Ceased
- 2000-04-11 KR KR10-2001-7015763A patent/KR100467898B1/ko not_active Expired - Fee Related
- 2000-04-11 DK DK00925194T patent/DK1185520T3/da active
- 2000-04-11 AU AU43996/00A patent/AU758605B2/en not_active Ceased
- 2000-04-11 BR BR0011445-6A patent/BR0011445A/pt not_active IP Right Cessation
- 2000-04-11 AT AT00925194T patent/ATE261946T1/de active
2001
- 2001-12-10 US US10/012,786 patent/US6559314B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
DE50005699D1 (de)	2004-04-22
DE19926233C1 (de)	2000-10-19
KR100467898B1 (ko)	2005-02-21
CN1169799C (zh)	2004-10-06
HK1042483A1 (zh)	2002-08-16
CA2373834A1 (en)	2000-12-21
BR0011445A (pt)	2002-03-19
RU2218336C2 (ru)	2003-12-10
PT1185520E (pt)	2004-08-31
AU758605B2 (en)	2003-03-27
CN1355795A (zh)	2002-06-26
ES2215045T3 (es)	2004-10-01
ATE261946T1 (de)	2004-04-15
JP3803292B2 (ja)	2006-08-02
EP1185520A1 (de)	2002-03-13
KR20020022688A (ko)	2002-03-27
DK1185520T3 (da)	2004-06-28
JP2003502319A (ja)	2003-01-21
US20020082427A1 (en)	2002-06-27
EP1185520B1 (de)	2004-03-17
US6559314B2 (en)	2003-05-06
AU4399600A (en)	2001-01-02
WO2000076986A1 (de)	2000-12-21
NZ515561A (en)	2003-06-30
CA2373834C (en)	2005-11-08
MXPA01012237A (es)	2002-08-12

Publication	Publication Date	Title
HK1042483B (zh)	2004-09-10	四氫噻唑的製造方法
MC1199A1 (fr)	1979-03-19	Composes tricycliques
IL29569A (en)	1971-12-29	1,4-dihydropyridine derivatives and their production
SK282736B6 (sk)	2002-11-06	Spôsob prípravy amlodipín benzénsulfonátu
US4127671A (en)	1978-11-28	P-acetamidophenyl diethylaminoacetate
JPS60126284A (ja)	1985-07-05	ピリドンカルボン酸誘導体およびその塩
JPH0587064B2 (zh)	1993-12-15
FI63568C (fi)	1983-07-11	Foerfarande foer framstaellning av nya terapeutiskt anvaendbara i 7-staellning substituerade 8-aminometylisoflavonderivat
JPH0215067A (ja)	1990-01-18	イソキノリンスルホンアミド誘導体
US4609659A (en)	1986-09-02	2,6-disubstituted derivatives of 3-nitropyrazines useful as adjuncts to radiation therapy
JPH0573754B2 (zh)	1993-10-15
US4317914A (en)	1982-03-02	Oxazolines
HU198473B (en)	1989-10-30	Process for producing 8-thiotetrahydro-quinoline derivatives and salts thereof, as well as pharmaceutical compositions comprising same as active ingredient
JPS6310955B2 (zh)	1988-03-10
PL144481B1 (en)	1988-05-31	Process for preparing derivatives of pyrimidinotrione
US3998820A (en)	1976-12-21	10'-[ω-N-/1,4-diazabicyclo(4,m,o)-alkanyl/-acyl]-phenothiazines, their acidic addition salts and quaternary salts, process for producing same and use
US3714166A (en)	1973-01-30	Cocarboxylase arginate and process for the production thereof
DK142172B (da)	1980-09-15	Analogifremgangsmaade til fremstilling af basisk substituerede2-alkylamino-4-phenylimidazoliner eller syreadditionssalte heraf
JPS59141565A (ja)	1984-08-14	向精神性活性を有するピリダジン誘導体，その製造方法および該誘導体を含有する薬剤
US4083976A (en)	1978-04-11	10'-( ω-N)-1,4-Diazabicyclo(4,3,0)-alkanyl-lacyl) -phenothiazine compositions
JPH0324077A (ja)	1991-02-01	イミダゾール誘導体の製法
KR850000431B1 (ko)	1985-04-03	피롤 유도체의 제조방법
JPS63165368A (ja)	1988-07-08	新規複素環化合物およびその製造法
JPH01216980A (ja)	1989-08-30	アルキル―ピペラジニル―５，６―アルキレンピリミジン類
KR840001286B1 (ko)	1984-09-07	2-이미다졸린 유도체류의 제조방법

Legal Events

Date	Code	Title	Description
2004-12-15	PF	Patent in force
2005-04-15	CHRG	Changes in the register	Free format text: FROM PROBIODRUG AG TO PROSIDION LIMITED; JOURNAL NO.: 106; PUBLICATION DATE: 15-04-2005; SECTION NAME: CHANGES IN THE REGISTER 266/280
2013-11-08	PC	Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)	Effective date: 20130411