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GT201200289A - 3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas - Google Patents

3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas

Info

Publication number
GT201200289A
GT201200289A GT201200289A GT201200289A GT201200289A GT 201200289 A GT201200289 A GT 201200289A GT 201200289 A GT201200289 A GT 201200289A GT 201200289 A GT201200289 A GT 201200289A GT 201200289 A GT201200289 A GT 201200289A
Authority
GT
Guatemala
Prior art keywords
fungicides
substituted
dihydropirimidine
onas
imino
Prior art date
Application number
GT201200289A
Other languages
English (en)
Inventor
Boebel Timothy
Lorsbach Beth
Martin Timothy
Owen W John
Sullenberger Michael
Webster Jeffery
Yao Chenglin
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT201200289A publication Critical patent/GT201200289A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

LA PRESENTE INVENCIÓN ESTÁ RELACIONADA CON EL CAMPO DE N3-SUSTITUIDO-N1-SULFONIL-5-FLÚORPIRIMIDINONA Y SUS DERIVADOS Y EL USO DE ESTOS COMPUESTOS COMO FUNGICIDAS.
GT201200289A 2010-04-26 2012-10-25 3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas GT201200289A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26

Publications (1)

Publication Number Publication Date
GT201200289A true GT201200289A (es) 2014-04-08

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201200289A GT201200289A (es) 2010-04-26 2012-10-25 3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas

Country Status (33)

Country Link
US (1) US8263603B2 (es)
EP (1) EP2563129B1 (es)
JP (1) JP5784705B2 (es)
KR (1) KR101793766B1 (es)
CN (1) CN102946730B (es)
AU (1) AU2011245544B2 (es)
BR (1) BR112012027439B1 (es)
CA (1) CA2797226C (es)
CL (1) CL2012002979A1 (es)
CO (1) CO6592042A2 (es)
CR (1) CR20120584A (es)
CY (1) CY1117956T1 (es)
DK (1) DK2563129T3 (es)
EC (1) ECSP12012302A (es)
ES (1) ES2588742T3 (es)
GT (1) GT201200289A (es)
HN (1) HN2012002272A (es)
HR (1) HRP20161107T1 (es)
HU (1) HUE029489T2 (es)
IL (1) IL222646A (es)
LT (1) LT2563129T (es)
ME (1) ME02530B (es)
MX (1) MX2012012530A (es)
NZ (1) NZ603151A (es)
PH (1) PH12012502138B1 (es)
PL (1) PL2563129T3 (es)
PT (1) PT2563129T (es)
RS (1) RS55239B1 (es)
RU (1) RU2562840C2 (es)
SI (1) SI2563129T1 (es)
SM (1) SMT201600298B (es)
UA (1) UA108101C2 (es)
WO (1) WO2011137002A1 (es)

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EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона
CN104884062B (zh) 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
AU2013370493B2 (en) * 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
KR20150103095A (ko) * 2012-12-28 2015-09-09 다우 아그로사이언시즈 엘엘씨 1-(치환된-벤조일)-5-플루오로-4-이미노-3-메틸-3,4-디히드로피리미딘-2(1h)-온 유도체
US9642368B2 (en) * 2012-12-31 2017-05-09 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
CR20210172A (es) 2013-12-31 2021-05-11 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2 (1h)-ona y los procesos para su preparación
BR112016015158A2 (pt) * 2013-12-31 2017-08-08 Adama Makhteshim Ltd Misturas fungicidas sinergísticas para controle de fungos em cereais
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
WO2018139560A1 (ja) 2017-01-26 2018-08-02 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2018190350A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CA3059702A1 (en) 2017-04-10 2018-10-18 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
MY190386A (en) 2017-04-11 2022-04-20 Mitsui Chemicals Agro Inc Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
JP7157738B2 (ja) 2017-06-08 2022-10-20 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
US11632954B2 (en) 2017-07-17 2023-04-25 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1 -tosyl-3,4-dihydropyrimidin-2-one
US12114658B2 (en) 2018-07-25 2024-10-15 Mitsui Chemicals Crop & Life Solutions, Inc. Compounds having a nitrogen-containing unsaturated six-membered ring and agricultural and horticultural fungicides containing the same as active ingredients
IL282939B2 (en) 2018-11-05 2024-10-01 Adama Makhteshim Ltd Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and methods of use thereof
US20220248673A1 (en) 2019-07-22 2022-08-11 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
UY38890A (es) 2019-09-23 2021-04-30 Adama Makhteshim Ltd Procedimiento para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
US20230104954A1 (en) * 2020-03-09 2023-04-06 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
MX2022013874A (es) 2020-05-04 2022-11-30 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y metodos de uso de las mismas.
WO2022009154A1 (en) 2020-07-08 2022-01-13 Adama Makhteshim Ltd. Fungicidal mixtures
US20240172750A1 (en) 2021-01-27 2024-05-30 Adama Makhteshim Ltd. 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Controlling Plant Diseases
MX2023012897A (es) 2021-05-04 2023-12-06 Adama Makhteshim Ltd Formas cristalinas de 5-fluoro-4-imino-3-metil-1-tosil-3,4- dihidropirimidin-2-ona, y mezclas, composiciones y metodos de uso de las mismas.
US20240351990A1 (en) * 2021-09-15 2024-10-24 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4- sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
CA3248206A1 (en) * 2022-01-12 2023-07-20 Adama Makhteshim Ltd. FUNGICIDE MIXTURES COMPRISING A COMBINATION CONTAINING PHTALIMIDE FUNGICIDES
UY40172A (es) 2022-03-03 2023-10-13 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
EP4609713A3 (en) 2022-05-26 2025-10-29 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AR132077A1 (es) 2023-03-09 2025-05-21 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
WO2024189563A1 (en) 2023-03-14 2024-09-19 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
IL308593A (en) 2023-11-15 2025-06-01 Adama Makhteshim Ltd Reducing environmental impact of fungicidal enhancement
AR134494A1 (es) 2023-11-28 2026-01-21 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas

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HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
CA2629295A1 (en) * 2005-11-22 2007-05-31 Ishihara Sangyo Kaisha, Ltd. Germicide composition for agricultural and gardening applications and method for controlling plant disease
HUE026195T2 (en) * 2008-01-22 2016-05-30 Dow Agrosciences Llc 4-Amino-5-fluoropyrimidine derivatives as fungicides
EP2647287A1 (en) * 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides
EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону

Also Published As

Publication number Publication date
US8263603B2 (en) 2012-09-11
ES2588742T3 (es) 2016-11-04
CL2012002979A1 (es) 2013-01-25
PH12012502138A1 (en) 2013-02-04
BR112012027439A8 (pt) 2017-07-11
CN102946730B (zh) 2015-02-04
SI2563129T1 (sl) 2016-12-30
PT2563129T (pt) 2016-09-05
NZ603151A (en) 2013-10-25
KR20130093000A (ko) 2013-08-21
JP2013525434A (ja) 2013-06-20
BR112012027439A2 (pt) 2015-09-15
CN102946730A (zh) 2013-02-27
CR20120584A (es) 2013-01-03
AU2011245544A1 (en) 2012-11-15
AU2011245544B2 (en) 2015-04-16
CA2797226C (en) 2019-02-26
PL2563129T3 (pl) 2017-08-31
US20110263627A1 (en) 2011-10-27
IL222646A (en) 2017-01-31
IL222646A0 (en) 2012-12-31
EP2563129A1 (en) 2013-03-06
HK1182594A1 (en) 2013-12-06
EP2563129A4 (en) 2013-08-07
PH12012502138B1 (en) 2019-09-25
HN2012002272A (es) 2015-04-27
WO2011137002A1 (en) 2011-11-03
CY1117956T1 (el) 2017-05-17
RS55239B1 (sr) 2017-02-28
KR101793766B1 (ko) 2017-11-03
RU2012150293A (ru) 2014-06-10
ECSP12012302A (es) 2012-12-28
JP5784705B2 (ja) 2015-09-24
DK2563129T3 (en) 2016-09-12
MX2012012530A (es) 2012-12-17
CA2797226A1 (en) 2011-11-03
UA108101C2 (xx) 2015-03-25
SMT201600298B (it) 2016-11-10
RU2562840C2 (ru) 2015-09-10
CO6592042A2 (es) 2013-01-02
BR112012027439B1 (pt) 2018-01-16
HRP20161107T1 (hr) 2016-12-30
HUE029489T2 (en) 2017-02-28
EP2563129B1 (en) 2016-06-01
ME02530B (me) 2017-02-20
LT2563129T (lt) 2016-10-25

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