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ECSP12011652A - Derivados de 5-fluoro-2-oxopirimidinona-1 (2h)-carboxamida substituida-n1 - Google Patents

Derivados de 5-fluoro-2-oxopirimidinona-1 (2h)-carboxamida substituida-n1

Info

Publication number
ECSP12011652A
ECSP12011652A ECSP12011652A ECSP12011652A EC SP12011652 A ECSP12011652 A EC SP12011652A EC SP12011652 A ECSP12011652 A EC SP12011652A EC SP12011652 A ECSP12011652 A EC SP12011652A
Authority
EC
Ecuador
Prior art keywords
fluoro
derivatives
substituida
oxopirimidinona
carboxamida
Prior art date
Application number
Other languages
English (en)
Inventor
Timothy Martin
Mark Andrew Pobanz
Timothy Boebel
Kristy Bryan
Beth Lorsbach
W Owen
Jeffery Webster
Chenglin Yao
Scott Thornburgh
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP12011652(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP12011652A publication Critical patent/ECSP12011652A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente descripción se relaciona con el campo de las 5-fluoro-2-oxopirimidinona-1-(2H)-carboxamidas substituidas-N1 y sus derivados y el uso de estos compuestos como fungicidas.
ECSP12011652 2009-08-07 2012-02-07 Derivados de 5-fluoro-2-oxopirimidinona-1 (2h)-carboxamida substituida-n1 ECSP12011652A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
ECSP12011652A true ECSP12011652A (es) 2012-03-30

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP12011652 ECSP12011652A (es) 2009-08-07 2012-02-07 Derivados de 5-fluoro-2-oxopirimidinona-1 (2h)-carboxamida substituida-n1

Country Status (26)

Country Link
US (2) US8552020B2 (es)
EP (1) EP2461686B1 (es)
JP (1) JP5735510B2 (es)
KR (1) KR101792284B1 (es)
CN (1) CN102497781B (es)
BR (1) BR112012002757B1 (es)
CA (1) CA2769656C (es)
CL (1) CL2012000312A1 (es)
CO (1) CO6491115A2 (es)
CR (1) CR20120032A (es)
DK (1) DK2461686T3 (es)
EA (1) EA020910B1 (es)
EC (1) ECSP12011652A (es)
ES (1) ES2552097T3 (es)
HU (1) HUE027390T2 (es)
IL (1) IL217950A (es)
IN (1) IN2012DN00369A (es)
MX (1) MX2012001617A (es)
NI (1) NI201200021A (es)
NZ (1) NZ597483A (es)
PE (1) PE20120692A1 (es)
PL (1) PL2461686T3 (es)
PT (1) PT2461686E (es)
UA (1) UA107671C2 (es)
WO (1) WO2011017545A1 (es)
ZA (1) ZA201200813B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
NZ597597A (en) 2009-08-07 2014-01-31 Dow Agrosciences Llc Pesticidal compositions containing heteroaryl-n-aryl carbamate compounds
JP6258969B2 (ja) 2012-12-28 2018-01-10 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体
EP3689142A1 (en) * 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
DK2938194T3 (da) * 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
WO2015103144A1 (en) 2013-12-31 2015-07-09 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
CN118515619A (zh) 2017-07-17 2024-08-20 阿达玛克西姆股份有限公司 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物
KR20210136961A (ko) 2018-11-05 2021-11-17 아다마 마켓심 리미티드 5-플루오로-4-이미노-3-메틸-1-토실-3,4-디하이드로피리미딘-2-온을 포함하는 혼합물들과 조성물들 및 이들을 사용하는 방법들
CN114599639A (zh) 2019-09-23 2022-06-07 阿达玛马克西姆有限公司 用于制备5-(氟-4-亚氨基-3-甲基)-1-甲苯磺酰基-3,4-二氢嘧啶-(1h)-酮的方法
MX2022007134A (es) * 2019-12-10 2022-09-12 Syngenta Crop Protection Ag Metodos para controlar o prevenir la infestacion de plantas de cacahuate por microorganismos fitopatogenos.

Family Cites Families (24)

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US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (es) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
JPS60123486A (ja) * 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンｓおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
US6066638A (en) * 1995-07-05 2000-05-23 E. I. Du Pont De Nemours And Company Fungicidal pyrimidinones
NZ331175A (en) 1996-03-11 2000-02-28 Novartis Ag Pyrimidin-4-one derivatives useful as pesticides
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
EP1731523A4 (en) * 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
EP2044086A2 (en) * 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
JP5749017B2 (ja) 2008-01-22 2015-07-15 ダウ アグロサイエンシィズ エルエルシー ５−フルオロピリミジン誘導体
US20100029482A1 (en) 2008-08-01 2010-02-04 Benko Zoltan L Use of 5-fluorocytosine as a fungicide
DK2389375T3 (en) * 2009-01-23 2015-08-24 Euro Celtique Sa Hydroxamsyrederivater
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona

Also Published As

Publication number Publication date
KR20120052281A (ko) 2012-05-23
EP2461686B1 (en) 2015-10-07
PE20120692A1 (es) 2012-06-08
KR101792284B1 (ko) 2017-10-31
BR112012002757B1 (pt) 2020-10-06
HUE027390T2 (en) 2016-10-28
EP2461686A1 (en) 2012-06-13
CN102497781B (zh) 2014-12-10
CL2012000312A1 (es) 2012-10-05
EA020910B1 (ru) 2015-02-27
CR20120032A (es) 2012-03-22
US8552020B2 (en) 2013-10-08
CA2769656C (en) 2018-05-15
US20110034492A1 (en) 2011-02-10
JP5735510B2 (ja) 2015-06-17
WO2011017545A1 (en) 2011-02-10
UA107671C2 (en) 2015-02-10
IL217950A (en) 2015-04-30
IL217950A0 (en) 2012-03-29
HK1171915A1 (en) 2013-04-12
IN2012DN00369A (es) 2015-08-21
CO6491115A2 (es) 2012-07-31
NZ597483A (en) 2014-02-28
US9000002B2 (en) 2015-04-07
DK2461686T3 (en) 2016-01-18
ZA201200813B (en) 2013-05-29
CN102497781A (zh) 2012-06-13
US20140011824A1 (en) 2014-01-09
EP2461686A4 (en) 2013-02-13
AU2010279409A1 (en) 2012-02-02
NI201200021A (es) 2012-05-22
JP2013501727A (ja) 2013-01-17
PT2461686E (pt) 2015-11-18
MX2012001617A (es) 2012-04-11
ES2552097T3 (es) 2015-11-25
BR112012002757A2 (pt) 2019-12-17
PL2461686T3 (pl) 2016-04-29
CA2769656A1 (en) 2011-02-10
EA201270256A1 (ru) 2012-07-30

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