GT200400203A - DERIVATIVES OF TROPANO - Google Patents
DERIVATIVES OF TROPANOInfo
- Publication number
- GT200400203A GT200400203A GT200400203A GT200400203A GT200400203A GT 200400203 A GT200400203 A GT 200400203A GT 200400203 A GT200400203 A GT 200400203A GT 200400203 A GT200400203 A GT 200400203A GT 200400203 A GT200400203 A GT 200400203A
- Authority
- GT
- Guatemala
- Prior art keywords
- tropano
- derivatives
- compounds
- chemioquine
- ccr5
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102100035875 C-C chemokine receptor type 5 Human genes 0.000 abstract 1
- 101710149870 C-C chemokine receptor type 5 Proteins 0.000 abstract 1
- 230000008485 antagonism Effects 0.000 abstract 1
- 102000005962 receptors Human genes 0.000 abstract 1
- 108020003175 receptors Proteins 0.000 abstract 1
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A COMPUESTOS DE LA FORMULA GENERAL I EN LA QUE R1,R2,ME, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS ESTAN IMPLICADOS EN LA MODULACION, EN PARTICULAR EL ANTAGONISMO DE RECEPTORES CCR5 DE QUIMIOQUINA POR LO QUE SON DE UTILIDAD EN CUADROS DE VIH.THIS INVENTION CONCERNS COMPOUNDS OF GENERAL FORMULA I IN WHICH R1, R2, ME, ARE FUNCTIONAL GROUPS DESCRIBED IN THE RECORD. THESE COMPOUNDS ARE INVOLVED IN THE MODULATION, IN PARTICULAR THE ANTAGONISM OF CCR5 CHEMIOQUINE RECEPTORS, SO THEY ARE USEFUL IN HIV TABLES.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0323236.0A GB0323236D0 (en) | 2003-10-03 | 2003-10-03 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT200400203A true GT200400203A (en) | 2005-04-18 |
Family
ID=29415495
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT200400203A GT200400203A (en) | 2003-10-03 | 2004-10-01 | DERIVATIVES OF TROPANO |
Country Status (5)
| Country | Link |
|---|---|
| CN (2) | CN100526313C (en) |
| GB (1) | GB0323236D0 (en) |
| GT (1) | GT200400203A (en) |
| UA (1) | UA84714C2 (en) |
| ZA (1) | ZA200602096B (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5476307B2 (en) * | 2007-10-25 | 2014-04-23 | エグゼリクシス, インコーポレイテッド | Tropane compound |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20001420A1 (en) * | 1998-12-23 | 2000-12-18 | Pfizer | CCR5 MODULATORS |
| EP1492789B1 (en) * | 2002-04-08 | 2006-06-07 | Pfizer Limited | Tropane derivatives as ccr5 modulators |
-
2003
- 2003-10-03 GB GBGB0323236.0A patent/GB0323236D0/en not_active Ceased
-
2004
- 2004-09-28 CN CNB2004800286836A patent/CN100526313C/en not_active Expired - Fee Related
- 2004-09-28 CN CN200910146182A patent/CN101632664A/en active Pending
- 2004-09-28 UA UAA200603711A patent/UA84714C2/en unknown
- 2004-10-01 GT GT200400203A patent/GT200400203A/en unknown
-
2006
- 2006-03-10 ZA ZA200602096A patent/ZA200602096B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB0323236D0 (en) | 2003-11-05 |
| CN100526313C (en) | 2009-08-12 |
| UA84714C2 (en) | 2008-11-25 |
| CN1863801A (en) | 2006-11-15 |
| ZA200602096B (en) | 2007-05-30 |
| CN101632664A (en) | 2010-01-27 |
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