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GB902369A - Improvements in or relating to tablets or granules - Google Patents

Improvements in or relating to tablets or granules

Info

Publication number
GB902369A
GB902369A GB3708759A GB3708759A GB902369A GB 902369 A GB902369 A GB 902369A GB 3708759 A GB3708759 A GB 3708759A GB 3708759 A GB3708759 A GB 3708759A GB 902369 A GB902369 A GB 902369A
Authority
GB
United Kingdom
Prior art keywords
acid
granules
tablets
medicament
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB3708759A
Inventor
Joseph Stanley Dwight
Horst Rothing
Leslie John Gower
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER Ltd
Pfizer Ltd Great Britain
Original Assignee
PFIZER Ltd
Pfizer Ltd Great Britain
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER Ltd, Pfizer Ltd Great Britain filed Critical PFIZER Ltd
Priority to GB3708759A priority Critical patent/GB902369A/en
Publication of GB902369A publication Critical patent/GB902369A/en
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)

Abstract

Tablets or granules of medicament having a room temperature water-solubility of about 1% or less are prepared by applying to the surface of particles of the medicament a partial or complete envelope of a non-toxic film-forming substance, admixing the particles with a water-soluble ingestible ingredient selected from one or more of the following: glucose, dextrose, mannitol, sorbitol, lactose, glycine, leucine and delta glucono-lactone and with a pharmaceutically acceptable water-soluble solid acid or acid salt and then compressing the mixture so formed into tablets and granules. Specified film-forming substances are dimethyl phenyl silanes, ethyl cellulose, cellulose acetate phthalate, polyacrylic acid, polyacrylamide, polyvinylacetate, polyvinyl alcohol acetate, polyvinyl acetate stearate, polyvinyl methyl ether and ethylene glycol distearate, preferably on a dry basis used in an amount which is 1-10% by weight of the medicament. Specified acids and acid salts are tartaric acid, potassium acid tartrate, citric acid, mono- and di-sodium citrates, fumaric acid, adipic acid, malic acid and monosodium phosphate, preferably in an amount ranging from 1-6% by weight of the finished tablets or granules. Specified medicaments are 2-(b -chloroethyl)-2,3-dihydro-4-oxo-(benzo-1,3-oxazine), dihydroxy aluminium carbonate, phenacetin, acetyl salicylic acid, salicylamide, codeine, antibiotics, e.g. oxytetracycline, vitamins, e.g. Vitamin A, sulphathiazole and steroid hormones, e.g. hydrocortisone. The tablets or granules may also contain water-soluble drugs such as water-soluble vitamins, e.g. nicotinamide and stimulants, e.g. caffeine. Specified tableting and granulating additives are lubricants, e.g. stearic acid talc and magnesium stearate, sweetening agents, e.g. saccharin and sodium saccharin, lemon flavour, spearmint oil and sodium chloride. The coated medicament particles should have a size in the range 16-100 mesh B.S.S.
GB3708759A 1959-11-02 1959-11-02 Improvements in or relating to tablets or granules Expired GB902369A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
GB3708759A GB902369A (en) 1959-11-02 1959-11-02 Improvements in or relating to tablets or granules

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3708759A GB902369A (en) 1959-11-02 1959-11-02 Improvements in or relating to tablets or granules

Publications (1)

Publication Number Publication Date
GB902369A true GB902369A (en) 1962-08-01

Family

ID=10393618

Family Applications (1)

Application Number Title Priority Date Filing Date
GB3708759A Expired GB902369A (en) 1959-11-02 1959-11-02 Improvements in or relating to tablets or granules

Country Status (1)

Country Link
GB (1) GB902369A (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4451452A (en) * 1980-11-29 1984-05-29 Sandoz Ltd. Pharmaceutical compositions containing biodegradable polymers
US6541034B1 (en) * 1998-12-22 2003-04-01 Gerhard Gergely Matrix material containing sugars and/or sugar alcohols and process for its preparation
WO2010133267A1 (en) * 2009-05-18 2010-11-25 Krüger Gmbh & Co.Kg Sucralose-containing artificial sweetener compositions
US11291701B1 (en) * 2021-02-04 2022-04-05 Seed Edibles Orally disintegrating, sublingual and buccal formulations

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4451452A (en) * 1980-11-29 1984-05-29 Sandoz Ltd. Pharmaceutical compositions containing biodegradable polymers
US4615881A (en) * 1980-11-29 1986-10-07 Sandoz Ltd. Pharmaceutical compositions
US6541034B1 (en) * 1998-12-22 2003-04-01 Gerhard Gergely Matrix material containing sugars and/or sugar alcohols and process for its preparation
WO2010133267A1 (en) * 2009-05-18 2010-11-25 Krüger Gmbh & Co.Kg Sucralose-containing artificial sweetener compositions
EP2628397A1 (en) * 2009-05-18 2013-08-21 Krüger GmbH & Co. KG Sucralose-containing sweetener compositions
US11291701B1 (en) * 2021-02-04 2022-04-05 Seed Edibles Orally disintegrating, sublingual and buccal formulations

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