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GB1458029A - Sulphamylbenzoic acids and preparation thereof - Google Patents

Sulphamylbenzoic acids and preparation thereof

Info

Publication number
GB1458029A
GB1458029A GB5720773A GB5720773A GB1458029A GB 1458029 A GB1458029 A GB 1458029A GB 5720773 A GB5720773 A GB 5720773A GB 5720773 A GB5720773 A GB 5720773A GB 1458029 A GB1458029 A GB 1458029A
Authority
GB
United Kingdom
Prior art keywords
formula
compound
alkyl
prepared
hexamethyleneimino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB5720773A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Inc
Original Assignee
Pfizer Corp Belgium
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US00318213A external-priority patent/US3843662A/en
Application filed by Pfizer Corp Belgium, Pfizer Inc filed Critical Pfizer Corp Belgium
Publication of GB1458029A publication Critical patent/GB1458029A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/34Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/42Oxygen atoms attached in position 3 or 5
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/155Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fodder In General (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

1458029 Sulphamylbenzoic acids PFIZER Inc 10 Dec 1973 [26 Dec 1972] 57207/73 Addition to 1353357 Heading C2C Novel compounds of Formula I (in which Q is H, Cl, F, Br, 1-4C alkoxy, di- (1-4C alkyl)amino, OH, SCH 3 , piperidino or hexamethyleneimino; T is Cl, F, Br, CH 3 , OCH 3 or CF 3 ; R<SP>16</SP> is H or 2-4C alkyl; and R<SP>17</SP> is 2-4C alkyl or a group of Formula II in which n is 1-3; and R 10 and R 11 are H, Cl, Br, CH3 or phenyl; with the proviso that where R<SP>17</SP> is 2-4C alkyl, R<SP>16</SP> is not H; or -NR<SP>16</SP>R<SP>17</SP> is morpholino, piperidino, mono- or di-methylpiperidino or hexamethyleneimino) and amides, 1-4C alkyl esters and salts thereof are prepared by reacting an amine R<SP>16</SP>R<SP>17</SP>NH with a compound of Formula III (in which Hal is halo); or by hydrolysis of a compound of Formula IV or by reacting a compound of Formula V (a) with a 1-4C alkanol or CH 3 SH in the presence of a base to give a compound of Formula I in which O is 1-4C alkoxy or SCH 3 ; (b) with an amine R<SP>1</SP>R<SP>11</SP>NH to give a compound of Formula I in which Q is NR<SP>1</SP>R<SP>1</SP> and, R<SP>1</SP> and R<SP>11</SP> are 1-4C alkyl or NR<SP>1</SP>R<SP>11</SP> is piperidino or hexamethyleneimino; or (c) with a base to give a compound of Formula I in which Q is OH. 2,3 - Dichloro - 5 - chlorosulphonyl - benzoic acid is prepared by reaction of 2,6-dichlorobenzoic acid with chlorosulphonic acid. 2,6- Dichloro - 5 - chlorosulphonyl - benzoic acid is prepared in a similar manner. Methyl 3-amino- 2-chlorobenzoate HCl. is prepared by reduction of methyl 3-nitro-2-chlorobenzoate with SnCl 2 / HCl. Methyl 2 - chloro - 3 - chlorosulphonylbenzoate is prepared by reaction of the previous intermediate with NaNO 2 , then SO 2 and CuCl 2 . Pharmaceutical compositions used in treating atherosclerosis comprise a compound of Formula I together with a suitable carrier and are administered orally or parenterally.
GB5720773A 1972-12-26 1973-12-10 Sulphamylbenzoic acids and preparation thereof Expired GB1458029A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US00318213A US3843662A (en) 1971-12-09 1972-12-26 2-halo-5-(substituted piperidino sulfonyl)benzoic acids

Publications (1)

Publication Number Publication Date
GB1458029A true GB1458029A (en) 1976-12-08

Family

ID=23237158

Family Applications (1)

Application Number Title Priority Date Filing Date
GB5720773A Expired GB1458029A (en) 1972-12-26 1973-12-10 Sulphamylbenzoic acids and preparation thereof

Country Status (11)

Country Link
JP (2) JPS4986522A (en)
AR (1) AR214849A1 (en)
AU (1) AU6366973A (en)
BE (1) BE808939R (en)
CA (1) CA1012974A (en)
DE (1) DE2363786A1 (en)
ES (2) ES421767A2 (en)
FR (1) FR2211261B2 (en)
GB (1) GB1458029A (en)
NL (1) NL7317455A (en)
ZA (1) ZA739662B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0068407A1 (en) * 1981-06-22 1983-01-05 Hodogaya Chemical Co., Ltd. Aminosulfonylbenzoic acid derivatives
US4999134A (en) * 1987-09-25 1991-03-12 Basf Aktiengesellschaft Zinc salts, lead salts and/or calcium salts of carboxylic acids and their use as corrosion inhibitors

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0068408A1 (en) * 1980-11-10 1983-01-05 Mochida Pharmaceutical Co., Ltd. Antiviral compositions and a method for treating virus diseases
EP0132540A1 (en) * 1981-06-22 1985-02-13 Mochida Pharmaceutical Co., Ltd. Antiviral compositions
DE19941540C2 (en) * 1999-09-01 2002-08-29 Aventis Pharma Gmbh Sulfonylcarboxamides for the manufacture of medicaments for the prophylaxis or treatment of hyperlipidemia

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1122541B (en) * 1959-12-28 1962-01-25 Hoechst Ag Process for the production of sulfamyl-anthranilic acids
FR1472906A (en) * 1961-05-08 1967-03-17 Parke Davis & Co Esters of 4-halo-3-sulfamoylbenzoic acids and their production process
FR1450358A (en) * 1960-09-03 1966-06-24 Parke Davis & Co Production of new 4-halogeno-3-sulfamylbenzamides
FR1311859A (en) * 1961-09-18 1962-12-14 Soc Ind Fab Antibiotiques Sifa New sulfonamide derivatives, and method of preparation
US3565920A (en) * 1966-12-29 1971-02-23 Ciba Geigy Corp 5-sulfamyl-anthranilic acids
US3567746A (en) * 1968-07-10 1971-03-02 Pennwalt Corp N-aryl benzamides
US3700773A (en) * 1969-06-25 1972-10-24 Merck & Co Inc Substituted phenylsulfamyl salicyclic acids and derivatives thereof in the treatment of inflammation

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0068407A1 (en) * 1981-06-22 1983-01-05 Hodogaya Chemical Co., Ltd. Aminosulfonylbenzoic acid derivatives
US4999134A (en) * 1987-09-25 1991-03-12 Basf Aktiengesellschaft Zinc salts, lead salts and/or calcium salts of carboxylic acids and their use as corrosion inhibitors

Also Published As

Publication number Publication date
ES421767A2 (en) 1977-07-01
CA1012974A (en) 1977-06-28
FR2211261A2 (en) 1974-07-19
FR2211261B2 (en) 1977-04-15
BE808939R (en) 1974-06-21
AU6366973A (en) 1975-06-19
JPS4986522A (en) 1974-08-19
ES425208A1 (en) 1976-06-16
AR214849A1 (en) 1979-08-15
NL7317455A (en) 1974-06-28
JPS5924975B2 (en) 1984-06-13
JPS58170756A (en) 1983-10-07
DE2363786A1 (en) 1974-07-11
ZA739662B (en) 1975-01-29

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PCNP Patent ceased through non-payment of renewal fee