[go: up one dir, main page]

ES8307233A1 - Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same - Google Patents

Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same

Info

Publication number
ES8307233A1
ES8307233A1 ES82511759A ES511759A ES8307233A1 ES 8307233 A1 ES8307233 A1 ES 8307233A1 ES 82511759 A ES82511759 A ES 82511759A ES 511759 A ES511759 A ES 511759A ES 8307233 A1 ES8307233 A1 ES 8307233A1
Authority
ES
Spain
Prior art keywords
hydrogen
alkyl
thiazane
derivatives
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES82511759A
Other languages
Spanish (es)
Other versions
ES511759A0 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
MIDIT
Original Assignee
MIDIT
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by MIDIT filed Critical MIDIT
Publication of ES8307233A1 publication Critical patent/ES8307233A1/en
Publication of ES511759A0 publication Critical patent/ES511759A0/en
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Facsimiles In General (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Derivatives of 1,4-thiazane-3-carboxylic acid represented by the formula I, wherein R1 and R2 are hydrogen, an alkyl radical or a phenyl nucleus substituted or not or form a cycloalkyl radical R3 is a hydroxyl group, OR9 group, wherein R9 may have different significations R4 is hydrogen, alkyl or CONH2, R3 and R4 forming a hydantoin cycle, R5 and R6 representing hydrogen, alkyl, phenyl substituted or not R7 is hydrogen, alkyl, particularly dimethyl, phenyl substituted or not, and the salts of those compounds. < IMAGE > as well as the pharmaceutical compositions containing them and the intermediaries for their preparation, having the formulas II, III, IV: < IMAGE >.
ES82511759A 1981-04-29 1982-04-28 PROCEDURE FOR PREPARING DERIVATIVES OF ACID 1,4-TIAZAN-3-CARBOXILICO. Granted ES511759A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LU83327A LU83327A1 (en) 1981-04-29 1981-04-29 PROCESS FOR THE PREPARATION OF 1,4-THIAZINE DERIVATIVES, THEIR USE AND COMPOSITIONS CONTAINING SUCH DERIVATIVES

Publications (2)

Publication Number Publication Date
ES8307233A1 true ES8307233A1 (en) 1983-07-01
ES511759A0 ES511759A0 (en) 1983-07-01

Family

ID=19729637

Family Applications (1)

Application Number Title Priority Date Filing Date
ES82511759A Granted ES511759A0 (en) 1981-04-29 1982-04-28 PROCEDURE FOR PREPARING DERIVATIVES OF ACID 1,4-TIAZAN-3-CARBOXILICO.

Country Status (16)

Country Link
JP (1) JPS58500713A (en)
KR (1) KR830010089A (en)
BE (1) BE893025A (en)
ES (1) ES511759A0 (en)
FI (1) FI66366C (en)
FR (1) FR2509303A1 (en)
GB (1) GB2111056B (en)
GR (1) GR75996B (en)
IT (1) IT1190794B (en)
LU (1) LU83327A1 (en)
NL (1) NL8220153A (en)
NO (1) NO824398L (en)
PT (1) PT74813B (en)
SE (1) SE8207294D0 (en)
WO (1) WO1982003860A1 (en)
ZA (1) ZA822926B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3436386A1 (en) * 1984-10-04 1986-04-10 Merck Patent Gmbh, 6100 Darmstadt (THIO) MORPHOLINE
FR2618434B1 (en) * 1987-07-21 1991-02-08 Oreal ESTERS OF THIAMORPHOLINONE CARBOXYLIC ACID AND DERIVATIVES THEREOF, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE COSMETIC AND DERMO-PHARMACEUTICAL FIELD
WO1990007111A2 (en) * 1988-12-14 1990-06-28 Hicks, Richard Method for predicting biological activity of antibiotics, and novel non beta-lactam antibacterial agents derived therefrom
RU2650111C2 (en) 2012-02-03 2018-04-09 Санофи Fused pyrroledicarboxamides and their use as pharmaceuticals

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2187327B1 (en) * 1972-06-15 1975-06-20 Rech Pharm Scientifiques
US4179276A (en) * 1977-02-01 1979-12-18 E. I. Du Pont De Nemours And Company Novel imidazothiazine-1,3 (2H)-diones
JPS5540658A (en) * 1978-09-19 1980-03-22 Tanabe Seiyaku Co Ltd 1,4-thiazan-3-carboxylic ester derivative and its preparation

Also Published As

Publication number Publication date
FI66366B (en) 1984-06-29
JPS58500713A (en) 1983-05-06
SE8207294L (en) 1982-12-21
GB2111056B (en) 1985-03-06
GR75996B (en) 1984-08-03
PT74813B (en) 1983-10-26
BE893025A (en) 1982-10-29
FI824279L (en) 1982-12-14
GB2111056A (en) 1983-06-29
FI824279A0 (en) 1982-12-14
IT1190794B (en) 1988-02-24
WO1982003860A1 (en) 1982-11-11
ES511759A0 (en) 1983-07-01
SE8207294D0 (en) 1982-12-21
JPH0330592B2 (en) 1991-04-30
ZA822926B (en) 1983-03-30
KR830010089A (en) 1983-12-26
IT8220998A0 (en) 1982-04-29
PT74813A (en) 1982-05-01
FI66366C (en) 1984-10-10
NL8220153A (en) 1983-03-01
NO824398L (en) 1982-12-28
FR2509303A1 (en) 1983-01-14
LU83327A1 (en) 1983-03-24

Similar Documents

Publication Publication Date Title
GR3005315T3 (en)
ES8306759A1 (en) Cephalosporin derivatives, their preparation and compositions containing them.
ES8302001A1 (en) Cephalosporin derivatives, a process for their preparation and compositions containing them.
ES8507090A1 (en) 1,5-Benzothiazepines with cardiovascular utility, and pharmaceutical compositions containing them
ES486824A1 (en) Neuroleptic-4-(naphthylmethyl)piperidine derivatives
IL63782A0 (en) 2-(1,4-benzodioxan-2-ylalkyl)imidazoles,their preparation and pharmaceutical compositions containing them
ES8106289A1 (en) Derivatives of alpha-phenyl-2-pyrrolidine methanol and their salts, process for their preparation, use as medicines and compositions containing them.
ES8307233A1 (en) Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same
ES8303397A1 (en) 1(4-Quinolyl)ethanol or propanol derivatives, pharmaceutical compositions containing them and processes for their preparation.
ES8305359A1 (en) Bicyclo (3,2,1) octylbenzamides, a process for their preparation and pharmaceutical compositions containing them.
DE3070768D1 (en) 1-((substituted-naphthyl)ethyl)-imidazole derivatives, pharmaceutical compositions containing them and methods of making them
ES8407053A1 (en) Penem derivatives, and composition containing them
ES8400743A1 (en) 1-Phenylindazol-3-one compounds, process and intermediates for their preparation and medicines containing these compounds.
ES8200113A1 (en) Cephalosporin compounds
PT80787A (en) Process for preparing piperidine (or pyrrolidine)-butanamides and compounds relating to them
DE3264556D1 (en) Sulfimines, their salts and their preparation, and pharmaceutical compositions containing them
ES8501382A1 (en) Phenyl-acetic-acid derivatives, their preparation and pharmaceutical compostions containing them.
ES8406442A1 (en) New quinolylacetic acid compounds and pharmaceutical compositions containing them.
ATE19879T1 (en) FURILOXAZOLYLACETIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
IE801382L (en) Piperidines.
ES8502700A1 (en) Derivatives of tetrahydrobenzothiazole and herbicidal compositions containing the same as an active ingredient
ES8205816A1 (en) Cardenolide-bis-digitoxoside derivatives, process for their preparation and their utilization as medicines.
SE8301785L (en) SET TO MAKE 2-THIOPHENIC ACETIC ACID DERIVATIVES AND INTERMEDIATES REQUIRED FOR THEIR PREPARATION
ES488388A1 (en) Thiazole derivatives, their preparation and medicaments containing them.
MY101628A (en) Sulfonamide compounds and salts thereof, herbicidal compositions containing them, and process for producing them.