GB1330071A - Oestrone derivative and a process for its manufacture - Google Patents
Oestrone derivative and a process for its manufactureInfo
- Publication number
- GB1330071A GB1330071A GB1042771*[A GB1042771A GB1330071A GB 1330071 A GB1330071 A GB 1330071A GB 1042771 A GB1042771 A GB 1042771A GB 1330071 A GB1330071 A GB 1330071A
- Authority
- GB
- United Kingdom
- Prior art keywords
- april
- methyl
- manufacture
- methylestrone
- uterotropic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/168—Steroids
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/184—Hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Polymers & Plastics (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Husbandry (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Food Science & Technology (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1330071 The 3-cyclopentyl ether of 7α-methylestrone CIBA-GEIGY AG 21 April 1971 [24 April 1970] 10427/71 Heading C2U The title compound is prepared by etherification, using a reactive ester of cyclopentanol, of 7α-methyl-estrone or a salt thereof or of a corresponding compound containing in the 17- position a ketalized oxo group or a free or esterified hydroxyl group with subsequent conversion to a 17-one by known methods. In one example the primary product is 3-cyclopentyloxy - 7α - methyl - 17# - hydroxy - #<SP>1,3,5(10)</SP> - estratriene which is converted by oxidation to the required product. The novel steroid is stated to have estrogenic, uterotropic and blastocyte implantation inhibiting action, and it may be made up into pharmaceutical and veterinary compositions with suitable carriers.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH621770A CH536826A (en) | 1970-04-24 | 1970-04-24 | Process for the production of a new, highly estrogenic steroid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1330071A true GB1330071A (en) | 1973-09-12 |
Family
ID=4306123
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB1042771*[A Expired GB1330071A (en) | 1970-04-24 | 1971-04-21 | Oestrone derivative and a process for its manufacture |
Country Status (17)
| Country | Link |
|---|---|
| AT (1) | AT307639B (en) |
| BE (1) | BE766182A (en) |
| CA (1) | CA925852A (en) |
| CH (2) | CH534140A (en) |
| CS (1) | CS151091B2 (en) |
| DE (1) | DE2118996A1 (en) |
| DK (2) | DK129451B (en) |
| ES (1) | ES390459A1 (en) |
| FI (1) | FI48827C (en) |
| FR (1) | FR2092080B1 (en) |
| GB (1) | GB1330071A (en) |
| IE (1) | IE35071B1 (en) |
| IL (1) | IL36652A (en) |
| NL (1) | NL7105576A (en) |
| PL (1) | PL73563B1 (en) |
| SE (1) | SE385588B (en) |
| SU (1) | SU399117A3 (en) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1866M (en) * | 1961-04-07 | 1963-06-17 | Vismara Francesco Spa | New ethers of estrogen hormones. |
| FR1434172A (en) * | 1963-12-24 | 1966-04-08 | Ciba Geigy | Process for preparing new substituted estrones |
| BE755689A (en) * | 1969-09-03 | 1971-03-03 | Upjohn Co | NEW 7 BETA-ALKYL-19- NORTESTOSTERONES MANUFACTURING PROCESS |
-
1970
- 1970-04-24 CH CH1870072A patent/CH534140A/en not_active IP Right Cessation
- 1970-04-24 CH CH621770A patent/CH536826A/en not_active IP Right Cessation
-
1971
- 1971-04-16 CA CA110524A patent/CA925852A/en not_active Expired
- 1971-04-19 IL IL36652A patent/IL36652A/en unknown
- 1971-04-20 DE DE19712118996 patent/DE2118996A1/en active Pending
- 1971-04-20 IE IE489/71A patent/IE35071B1/en unknown
- 1971-04-21 GB GB1042771*[A patent/GB1330071A/en not_active Expired
- 1971-04-22 PL PL1971147685A patent/PL73563B1/pl unknown
- 1971-04-22 FR FR7114320A patent/FR2092080B1/fr not_active Expired
- 1971-04-22 ES ES390459A patent/ES390459A1/en not_active Expired
- 1971-04-23 BE BE766182A patent/BE766182A/en unknown
- 1971-04-23 CS CS2984A patent/CS151091B2/cs unknown
- 1971-04-23 DK DK196971AA patent/DK129451B/en unknown
- 1971-04-23 NL NL7105576A patent/NL7105576A/xx unknown
- 1971-04-23 FI FI711129A patent/FI48827C/en active
- 1971-04-23 AT AT350971A patent/AT307639B/en not_active IP Right Cessation
- 1971-04-23 SE SE7105301A patent/SE385588B/en unknown
- 1971-04-23 SU SU1649255A patent/SU399117A3/ru active
-
1972
- 1972-08-18 DK DK411972AA patent/DK128110B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2092080B1 (en) | 1974-10-18 |
| DK128110B (en) | 1974-03-04 |
| IE35071B1 (en) | 1975-10-29 |
| IE35071L (en) | 1971-10-24 |
| CH534140A (en) | 1973-02-28 |
| DK129451B (en) | 1974-10-14 |
| AT307639B (en) | 1973-05-25 |
| PL73563B1 (en) | 1974-10-30 |
| SU399117A3 (en) | 1973-09-27 |
| FR2092080A1 (en) | 1972-01-21 |
| IL36652A (en) | 1974-07-31 |
| CS151091B2 (en) | 1973-09-17 |
| SE385588B (en) | 1976-07-12 |
| FI48827C (en) | 1975-01-10 |
| DE2118996A1 (en) | 1971-11-11 |
| ES390459A1 (en) | 1973-06-01 |
| FI48827B (en) | 1974-09-30 |
| CA925852A (en) | 1973-05-08 |
| CH536826A (en) | 1973-05-15 |
| DK129451C (en) | 1975-04-28 |
| IL36652A0 (en) | 1971-06-23 |
| NL7105576A (en) | 1971-10-26 |
| BE766182A (en) | 1971-10-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PCNP | Patent ceased through non-payment of renewal fee |