GB1116795A - An oral contraceptive preparation - Google Patents
An oral contraceptive preparationInfo
- Publication number
- GB1116795A GB1116795A GB4191865A GB4191865A GB1116795A GB 1116795 A GB1116795 A GB 1116795A GB 4191865 A GB4191865 A GB 4191865A GB 4191865 A GB4191865 A GB 4191865A GB 1116795 A GB1116795 A GB 1116795A
- Authority
- GB
- United Kingdom
- Prior art keywords
- oral contraceptive
- dosage unit
- progesterone
- contraceptive preparation
- quantity equivalent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229940127234 oral contraceptive Drugs 0.000 title 1
- 239000003539 oral contraceptive agent Substances 0.000 title 1
- RJKFOVLPORLFTN-LEKSSAKUSA-N Progesterone Chemical compound C1CC2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](C(=O)C)[C@@]1(C)CC2 RJKFOVLPORLFTN-LEKSSAKUSA-N 0.000 abstract 2
- DVMAUGGKVWJBDV-FXXCCUJSSA-N (8s,9s,13r,14s,16r)-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthrene-3,16-diol Chemical compound C1CC2=CC(O)=CC=C2[C@@H]2[C@@H]1[C@@H]1C[C@@H](O)C[C@@]1(C)CC2 DVMAUGGKVWJBDV-FXXCCUJSSA-N 0.000 abstract 1
- VOXZDWNPVJITMN-ZBRFXRBCSA-N 17β-estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 VOXZDWNPVJITMN-ZBRFXRBCSA-N 0.000 abstract 1
- 239000011149 active material Substances 0.000 abstract 1
- 239000003433 contraceptive agent Substances 0.000 abstract 1
- 230000002254 contraceptive effect Effects 0.000 abstract 1
- 229930182833 estradiol Natural products 0.000 abstract 1
- 229960005309 estradiol Drugs 0.000 abstract 1
- 230000001076 estrogenic effect Effects 0.000 abstract 1
- 230000003152 gestagenic effect Effects 0.000 abstract 1
- IMSSROKUHAOUJS-MJCUULBUSA-N mestranol Chemical compound C1C[C@]2(C)[C@@](C#C)(O)CC[C@H]2[C@@H]2CCC3=CC(OC)=CC=C3[C@H]21 IMSSROKUHAOUJS-MJCUULBUSA-N 0.000 abstract 1
- 229960003387 progesterone Drugs 0.000 abstract 1
- 239000000186 progesterone Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
An orally administerable contraceptive composition in dosage unit form comprises, per dosage unit, an estrogenic component in a quantity equivalent to 2000 I.u. (\sB 300) of estradiol and a gestagenic component in a quantity equivalent to 10 I.u. (+ 1.5) of progesterone. The preferred active materials are ethinyl estradiol 3 - methyl ether and 16 - methylene - 6 - dehydro - 17a - acetoxy progesterone.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS553564 | 1964-10-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1116795A true GB1116795A (en) | 1968-06-12 |
Family
ID=5400420
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB4191865A Expired GB1116795A (en) | 1964-10-06 | 1965-10-04 | An oral contraceptive preparation |
Country Status (3)
| Country | Link |
|---|---|
| BE (1) | BE670438A (en) |
| GB (1) | GB1116795A (en) |
| NL (1) | NL6512823A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5360616A (en) * | 1990-06-14 | 1994-11-01 | Applicaciones Farmaceuticas S.A. De C.V. | Injectable pharmaceutical composition |
-
1965
- 1965-10-01 BE BE670438D patent/BE670438A/xx unknown
- 1965-10-04 NL NL6512823A patent/NL6512823A/xx unknown
- 1965-10-04 GB GB4191865A patent/GB1116795A/en not_active Expired
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5360616A (en) * | 1990-06-14 | 1994-11-01 | Applicaciones Farmaceuticas S.A. De C.V. | Injectable pharmaceutical composition |
| US5633014A (en) * | 1990-06-14 | 1997-05-27 | Aplicaciones Farmaceuticas S.A. De C.V. | Injectable pharmaceutical composition |
Also Published As
| Publication number | Publication date |
|---|---|
| BE670438A (en) | 1966-01-31 |
| NL6512823A (en) | 1966-04-07 |
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