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FI955304L - (1,2,4)triatsoli(4,3-a)kinoksaliiniyhdisteitä, niiden valmistus ja käyttö - Google Patents

(1,2,4)triatsoli(4,3-a)kinoksaliiniyhdisteitä, niiden valmistus ja käyttö Download PDF

Info

Publication number
FI955304L
FI955304L FI955304A FI955304A FI955304L FI 955304 L FI955304 L FI 955304L FI 955304 A FI955304 A FI 955304A FI 955304 A FI955304 A FI 955304A FI 955304 L FI955304 L FI 955304L
Authority
FI
Finland
Prior art keywords
triazolo
preparation
quinoxaline compounds
quinoxaline
compounds
Prior art date
Application number
FI955304A
Other languages
English (en)
Swedish (sv)
Other versions
FI955304A7 (fi
FI955304A0 (fi
Inventor
Poul Jacobsen
Flemming Elmelund Nielsen
Lone Jeppesen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK53593A external-priority patent/DK53593D0/da
Priority claimed from DK128793A external-priority patent/DK128793D0/da
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of FI955304A7 publication Critical patent/FI955304A7/fi
Publication of FI955304L publication Critical patent/FI955304L/fi
Publication of FI955304A0 publication Critical patent/FI955304A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI955304A 1993-05-06 1994-04-28 (1,2,4)triatsoli(4,3-a)kinoksaliiniyhdisteitä, niiden valmistus ja käyttö FI955304A0 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DK53593A DK53593D0 (da) 1993-05-06 1993-05-06 Oe1,2,4aatriazolooe4,3-aaaquinoxalinonforbindelser, deres fremstilling og farmaceutiske praeparater indeholdende disse
DK128793A DK128793D0 (fi) 1993-11-12 1993-11-12
PCT/DK1994/000170 WO1994026746A1 (en) 1993-05-06 1994-04-28 [1,2,4]TRIAZOLO[4,3-a]QUINOXALINE COMPOUNDS, THEIR PREPARATION AND USE

Publications (3)

Publication Number Publication Date
FI955304A7 FI955304A7 (fi) 1995-11-06
FI955304L true FI955304L (fi) 1995-11-06
FI955304A0 FI955304A0 (fi) 1995-11-06

Family

ID=26064177

Family Applications (1)

Application Number Title Priority Date Filing Date
FI955304A FI955304A0 (fi) 1993-05-06 1994-04-28 (1,2,4)triatsoli(4,3-a)kinoksaliiniyhdisteitä, niiden valmistus ja käyttö

Country Status (19)

Country Link
US (1) US5532236A (fi)
EP (1) EP0698024B1 (fi)
JP (1) JPH08509747A (fi)
KR (1) KR100304177B1 (fi)
CN (1) CN1041931C (fi)
AT (1) ATE148120T1 (fi)
AU (1) AU683062B2 (fi)
CA (1) CA2162023A1 (fi)
DE (1) DE69401583T2 (fi)
DK (1) DK0698024T3 (fi)
ES (1) ES2097652T3 (fi)
FI (1) FI955304A0 (fi)
GR (1) GR3023001T3 (fi)
HU (1) HUT73983A (fi)
IL (1) IL109530A (fi)
NO (1) NO305516B1 (fi)
NZ (1) NZ266127A (fi)
TW (1) TW377354B (fi)
WO (1) WO1994026746A1 (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2200055A1 (en) * 1994-09-16 1996-03-21 Novo Nordisk A/S [1,2,4]triazolo[4,3-a]quinoxalinone derivatives, their preparation and use
AU694554B2 (en) * 1994-09-16 1998-07-23 Novo Nordisk A/S {1,2,4}triazolo{4,3-a}quinoxalinone derivatives, their preparation and use
DE19510965A1 (de) * 1995-03-24 1996-09-26 Asta Medica Ag Neue Pyrido/3,2-e/pyrazinone mit antiasthmatischer Wirksamkeit und Verfahren zu deren Herstellung
AU730503B2 (en) 1996-05-15 2001-03-08 Pfizer Inc. Novel 2,3 disubstituted-4(3H)-quinazolinones
WO1998027097A1 (en) * 1996-12-16 1998-06-25 Warner-Lambert Company Tricyclic quinoxaline derivatives as neuroprotective agents
US6015800A (en) * 1997-09-03 2000-01-18 Warner-Lambert Company Substituted quinoxaline-2-ones as glutamate receptor antagonists
IL125950A0 (en) * 1997-09-05 1999-04-11 Pfizer Prod Inc Methods of administering ampa receptor antagonists to treat dyskinesias associated with dopamine agonist therapy
US6323208B1 (en) 1997-09-05 2001-11-27 Pfizer Inc Atropisomers of 2,3-disubstituted-(5.6)-heteroaryl fused-pyrimidin-4-ones
AU9651198A (en) 1997-11-11 1999-05-31 Ono Pharmaceutical Co. Ltd. Fused pyrazine compounds
US20040152694A1 (en) * 2003-02-04 2004-08-05 Istvan Kurucz Methods and compositions for treating inflammatory disorders of the airways
US7781478B2 (en) 2004-07-14 2010-08-24 Ptc Therapeutics, Inc. Methods for treating hepatitis C
EP2338492A1 (en) 2009-12-24 2011-06-29 Universidad del Pais Vasco Methods and compositions for the treatment of alzheimer
WO2016199943A1 (en) * 2015-06-11 2016-12-15 Takeda Pharmaceutical Company Limited Heterocyclic compounds
CA3106752A1 (en) * 2018-07-20 2020-01-23 Grunenthal Gmbh Substituted triazolo quinoxaline derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4400382A (en) * 1980-05-09 1983-08-23 Usv Pharmaceutical Corporation Thiazoloquinoxalin-1,4-diones for treating allergy
DK162491D0 (da) * 1991-09-20 1991-09-20 Novo Nordisk As Heterocycliske forbindelser, deres fremstilling og farmaceutiske praeparater indeholdende forbindelserne

Also Published As

Publication number Publication date
NO954402L (no) 1996-01-05
FI955304A7 (fi) 1995-11-06
DK0698024T3 (da) 1997-07-28
IL109530A (en) 1997-01-10
NO305516B1 (no) 1999-06-14
EP0698024B1 (en) 1997-01-22
KR960701877A (ko) 1996-03-28
TW377354B (en) 1999-12-21
ES2097652T3 (es) 1997-04-01
DE69401583D1 (de) 1997-03-06
DE69401583T2 (de) 1997-06-12
AU683062B2 (en) 1997-10-30
HU9503157D0 (en) 1996-01-29
KR100304177B1 (ko) 2001-11-22
CN1125446A (zh) 1996-06-26
EP0698024A1 (en) 1996-02-28
HUT73983A (en) 1996-10-28
GR3023001T3 (en) 1997-07-30
WO1994026746A1 (en) 1994-11-24
JPH08509747A (ja) 1996-10-15
IL109530A0 (en) 1994-08-26
AU6720094A (en) 1994-12-12
FI955304A0 (fi) 1995-11-06
NZ266127A (en) 1997-11-24
CA2162023A1 (en) 1994-11-24
ATE148120T1 (de) 1997-02-15
CN1041931C (zh) 1999-02-03
NO954402D0 (no) 1995-11-03
US5532236A (en) 1996-07-02

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