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FI943421L - 1,5-bentsodiatsepiinijohdannaiset ja niiden käyttö lääkkeenä - Google Patents

1,5-bentsodiatsepiinijohdannaiset ja niiden käyttö lääkkeenä Download PDF

Info

Publication number
FI943421L
FI943421L FI943421A FI943421A FI943421L FI 943421 L FI943421 L FI 943421L FI 943421 A FI943421 A FI 943421A FI 943421 A FI943421 A FI 943421A FI 943421 L FI943421 L FI 943421L
Authority
FI
Finland
Prior art keywords
medicine
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
FI943421A
Other languages
English (en)
Swedish (sv)
Other versions
FI111632B (fi
FI943421A0 (fi
Inventor
Harry Finch
David Gordon Trist
Giorgio Tarzia
Aldo Feriani
Original Assignee
Glaxo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Spa filed Critical Glaxo Spa
Publication of FI943421L publication Critical patent/FI943421L/fi
Publication of FI943421A0 publication Critical patent/FI943421A0/fi
Application granted granted Critical
Publication of FI111632B publication Critical patent/FI111632B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/121,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI943421A 1992-01-21 1994-07-19 Menetelmä CCK-B-antagonistisesti vaikuttavien 1,5-bentsodiatsepiinijohdannaisten valmistamiseksi FI111632B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB9201180 1992-01-21
GB929201180A GB9201180D0 (en) 1992-01-21 1992-01-21 Chemical compounds
PCT/EP1993/000098 WO1993014074A1 (en) 1992-01-21 1993-01-19 1,5-benzodiazepine derivatives and their use in medicine
EP9300098 1993-01-19

Publications (3)

Publication Number Publication Date
FI943421L true FI943421L (fi) 1994-07-19
FI943421A0 FI943421A0 (fi) 1994-07-19
FI111632B FI111632B (fi) 2003-08-29

Family

ID=10708914

Family Applications (1)

Application Number Title Priority Date Filing Date
FI943421A FI111632B (fi) 1992-01-21 1994-07-19 Menetelmä CCK-B-antagonistisesti vaikuttavien 1,5-bentsodiatsepiinijohdannaisten valmistamiseksi

Country Status (29)

Country Link
US (2) US5580895A (fi)
JP (1) JP3253723B2 (fi)
KR (1) KR100263625B1 (fi)
CN (1) CN1049217C (fi)
AP (1) AP369A (fi)
AU (2) AU3450193A (fi)
BG (1) BG61876B1 (fi)
CA (1) CA2087672C (fi)
CZ (1) CZ283950B6 (fi)
FI (1) FI111632B (fi)
GB (1) GB9201180D0 (fi)
GE (1) GEP20001968B (fi)
HU (2) HU221297B1 (fi)
IL (1) IL104447A (fi)
IS (1) IS3970A (fi)
MX (1) MX9300261A (fi)
MY (1) MY131307A (fi)
NO (1) NO305952B1 (fi)
NZ (1) NZ245715A (fi)
OA (1) OA09964A (fi)
PH (1) PH30894A (fi)
PL (1) PL175340B1 (fi)
RO (1) RO114128B1 (fi)
RU (1) RU2124009C1 (fi)
SK (1) SK280173B6 (fi)
TW (1) TW226013B (fi)
UA (1) UA29416C2 (fi)
WO (1) WO1993014074A1 (fi)
ZA (1) ZA93375B (fi)

Families Citing this family (48)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9225492D0 (en) * 1992-12-05 1993-01-27 Glaxo Group Ltd Amine derivatives
WO1994024151A1 (en) * 1993-04-15 1994-10-27 Glaxo Inc. 1,5 benzodiazepine derivatives having cck and/or gastrin antagonistic activity
GB9307833D0 (en) * 1993-04-15 1993-06-02 Glaxo Inc Modulators of cholecystokinin and gastrin
GB9308431D0 (en) * 1993-04-23 1993-06-09 Glaxo Spa Chemical compounds
GB9308421D0 (en) * 1993-04-23 1993-06-09 Glaxo Spa Chemical compounds
GB2280182A (en) * 1993-07-20 1995-01-25 Glaxo Spa Benzodiazepine derivatives
GB9314977D0 (en) * 1993-07-20 1993-09-01 Glaxo Spa Chemical compounds
GB9314981D0 (en) * 1993-07-20 1993-09-01 Glaxo Spa Chemical compounds
GB9315018D0 (en) * 1993-07-20 1993-09-01 Glaxo Spa Chemical compounds
US5739129A (en) * 1994-04-14 1998-04-14 Glaxo Wellcome Inc. CCK or gastrin modulating 5-heterocyclic-1, 5 benzodiazepines
JPH09511223A (ja) * 1994-04-14 1997-11-11 グラクソ、ウェルカム、インコーポレーテッド Cckまたはガストリンを調節する5−ヘテロシクロ−1,5−ベンゾジアゼピン
PE27497A1 (es) * 1994-04-15 1997-08-07 Glaxo Inc Derivados de 1,5 benzodiazepina
GB9420748D0 (en) * 1994-10-14 1994-11-30 Glaxo Inc 1,5 benzodiazepine derivatives
US5780464A (en) * 1994-10-14 1998-07-14 Glaxo Wellcome Inc. Enteric coated compositions of 1,5-benzodiazepine derivatives having CCK antagonistic or agonistic activity
CA2239293A1 (en) 1995-12-11 1997-06-19 New England Medical Center Hosptials, Inc. Assay for and uses of peptide hormone receptor ligands
US5750353A (en) * 1995-12-11 1998-05-12 New England Medical Center Hospitals, Inc. Assay for non-peptide agonists to peptide hormone receptors
DE69724644T4 (de) * 1996-12-10 2006-08-10 Zeria Pharmaceutical Co., Ltd. 1,5-benzodiazepin-derivate
RU2321583C2 (ru) * 2001-01-22 2008-04-10 Мемори Фармасьютиклз Корпорейшн Применение производных анилина в качестве ингибиторов фосфодиэстеразы 4
JP4613157B2 (ja) * 2003-01-14 2011-01-12 サイトキネティクス・インコーポレーテッド 化合物、組成物および方法
GB0307918D0 (en) * 2003-04-05 2003-05-14 Astrazeneca Ab Therapeutic use
RU2377987C2 (ru) * 2003-11-18 2010-01-10 Бёрингер Ингельхайм Интернациональ Гмбх Твердая лекарственная форма
PL216049B1 (pl) 2004-06-17 2014-02-28 Cytokinetics Inc Pochodne mocznika, kompozycje zawierajace pochodne mocznika oraz zastosowanie pochodnych mocznika do wytwarzania leku do leczenia niewydolnosci serca
US7538223B2 (en) 2005-08-04 2009-05-26 Cytokinetics, Inc. Compounds, compositions and methods
US7825120B2 (en) 2005-12-15 2010-11-02 Cytokinetics, Inc. Certain substituted ((piperazin-1-ylmethyl)benzyl)ureas
US20070161617A1 (en) 2005-12-15 2007-07-12 Morgan Bradley P Certain chemical entities, compositions and methods
WO2007078815A2 (en) 2005-12-16 2007-07-12 Cytokinetics, Inc. Certain chemical entities, compositions, and methods
JP5178526B2 (ja) 2005-12-19 2013-04-10 サイトキネティクス・インコーポレーテッド 化合物、組成物および方法
CU20090172A6 (es) 2009-10-09 2011-10-05 Facultad De Quimica Universidad De La Habana Sistemas tricíclicos y tetracíclicos con actividad sobre el sistema nervioso central y vascular
JP6014904B2 (ja) 2011-07-29 2016-10-26 国立大学法人徳島大学 Erap1由来ペプチド及びその使用
CN103435562B (zh) * 2013-08-26 2016-02-24 华东理工大学 6-取代苯并二氮卓-2,4-二酮类化合物及其用途
CN108200760B (zh) 2015-07-22 2022-04-01 英安塔制药有限公司 作为rsv抑制剂的苯并二氮杂䓬衍生物
EP3402799B1 (en) 2016-01-15 2022-05-04 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
ES2923521T3 (es) 2017-02-16 2022-09-28 Enanta Pharm Inc Procesos para la preparación de derivados de benzodiazepina
WO2018226801A1 (en) * 2017-06-07 2018-12-13 Enanta Pharmaceuticals, Inc. Aryldiazepine derivatives as rsv inhibitors
US11091501B2 (en) 2017-06-30 2021-08-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
WO2019006291A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
JP7198811B2 (ja) 2017-09-29 2023-01-04 エナンタ ファーマシューティカルズ インコーポレイテッド Rsv阻害剤としての組み合わせ医薬剤
WO2019094920A1 (en) 2017-11-13 2019-05-16 Enanta Pharmaceuticals, Inc. Azepin-2-one derivatives as rsv inhibitors
WO2019199908A1 (en) 2018-04-11 2019-10-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
US20220098256A1 (en) 2018-11-30 2022-03-31 Tokushima University Therapeutic agent for breast cancer comprising big3-phb2 interaction-inhibiting peptide derived from phb2
CN113710276B (zh) 2019-03-18 2024-03-29 英安塔制药有限公司 苯二氮䓬衍生物作为rsv抑制剂
US11179400B2 (en) 2019-04-09 2021-11-23 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
US11505558B1 (en) 2019-10-04 2022-11-22 Enanta Pharmaceuticals, Inc. Antiviral heterocyclic compounds
UY39032A (es) 2020-01-24 2021-07-30 Enanta Pharm Inc Compuestos heterocíclicos como agentes antivirales
WO2022010882A1 (en) 2020-07-07 2022-01-13 Enanta Pharmaceuticals, Inc, Dihydroquinoxaline and dihydropyridopyrazine derivatives as rsv inhibitors
US11945824B2 (en) 2020-10-19 2024-04-02 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as anti-viral agents
AR129003A1 (es) 2022-04-07 2024-07-03 Enanta Pharm Inc Compuestos heterocíclicos antivirales
US12162857B2 (en) 2022-04-27 2024-12-10 Enanta Pharmaceuticals, Inc. Antiviral compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3984398A (en) * 1966-12-14 1976-10-05 Roussel-Uclaf 1,5-Benzodiazepine-2,4-diones
US4207228A (en) * 1977-09-21 1980-06-10 The B. F. Goodrich Company UV-Light-stabilized compositions containing substituted 1,5-diazacycloalkanes, novel compounds and synthesis thereof
JPS60158190A (ja) * 1984-01-30 1985-08-19 Eisai Co Ltd ヒダントイン誘導体およびその製法ならびにそれを含有する医薬
US4647561A (en) * 1985-08-05 1987-03-03 E. R. Squibb & Sons, Inc. 1,5-benzodiazepine compounds
FR2641280B1 (fr) * 1988-12-29 1994-01-21 Roussel Uclaf Nouveaux derives de la 2,4-dioxo 2,3,4,5-tetrahydro 1h-1,5-benzodiazepine, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
BG61876B1 (bg) 1998-08-31
OA09964A (en) 1995-12-11
WO1993014074A1 (en) 1993-07-22
CA2087672C (en) 2003-08-05
MY131307A (en) 2007-08-30
RO114128B1 (ro) 1999-01-29
HU9402150D0 (en) 1994-09-28
GEP20001968B (en) 2000-03-05
IS3970A (is) 1993-07-22
CN1049217C (zh) 2000-02-09
FI111632B (fi) 2003-08-29
IL104447A0 (en) 1993-05-13
US5637697A (en) 1997-06-10
MX9300261A (es) 1994-03-31
AU3193593A (en) 1993-07-22
AP9300478A0 (en) 1993-01-31
BG98881A (bg) 1995-03-31
HUT67375A (en) 1995-03-28
AU661749B2 (en) 1995-08-03
NO942720L (no) 1994-07-20
SK280173B6 (sk) 1999-09-10
HU221297B1 (en) 2002-09-28
RU94037768A (ru) 1996-08-10
IL104447A (en) 1998-02-22
HU211295A9 (en) 1995-11-28
ZA93375B (en) 1994-07-18
NZ245715A (en) 1995-07-26
PL175340B1 (pl) 1998-12-31
AP369A (en) 1994-11-06
PH30894A (en) 1997-12-23
TW226013B (fi) 1994-07-01
SK86494A3 (en) 1995-03-08
JPH07118244A (ja) 1995-05-09
CZ173694A3 (en) 1995-09-13
JP3253723B2 (ja) 2002-02-04
CZ283950B6 (cs) 1998-07-15
NO942720D0 (no) 1994-07-20
RU2124009C1 (ru) 1998-12-27
KR100263625B1 (ko) 2000-11-01
CN1074678A (zh) 1993-07-28
FI943421A0 (fi) 1994-07-19
GB9201180D0 (en) 1992-03-11
CA2087672A1 (en) 1993-07-22
NO305952B1 (no) 1999-08-23
UA29416C2 (uk) 2000-11-15
US5580895A (en) 1996-12-03
AU3450193A (en) 1993-08-03

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