FI932206A7 - Uusia heterosyklisiä yhdisteitä ekskitatoristen aminohapporeseptorien antagonisteina, menetelmä niiden valmistamiseksi ja niiden käyttö - Google Patents
Uusia heterosyklisiä yhdisteitä ekskitatoristen aminohapporeseptorien antagonisteina, menetelmä niiden valmistamiseksi ja niiden käyttö Download PDFInfo
- Publication number
- FI932206A7 FI932206A7 FI932206A FI932206A FI932206A7 FI 932206 A7 FI932206 A7 FI 932206A7 FI 932206 A FI932206 A FI 932206A FI 932206 A FI932206 A FI 932206A FI 932206 A7 FI932206 A7 FI 932206A7
- Authority
- FI
- Finland
- Prior art keywords
- antagonists
- preparation
- amino acid
- heterocyclic compounds
- excitatory amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6509—Six-membered rings
- C07F9/650952—Six-membered rings having the nitrogen atoms in the positions 1 and 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/59—Hydrogenated pyridine rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Injection Moulding Of Plastics Or The Like (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9003652A SE9003652D0 (sv) | 1990-11-15 | 1990-11-15 | New heterocyclic compounds |
| PCT/SE1991/000753 WO1992008724A1 (en) | 1990-11-15 | 1991-11-07 | New heterocyclic compounds as antagonists of excitatory amino acid receptors, processes for their preparation and their use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI932206A0 FI932206A0 (fi) | 1993-05-14 |
| FI932206A7 true FI932206A7 (fi) | 1993-05-14 |
| FI932206L FI932206L (fi) | 1993-05-14 |
Family
ID=20380925
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI932206A FI932206L (fi) | 1990-11-15 | 1991-11-07 | Nya heterocykliska foereningar som antagonister mot excitatoriska aminosyrareceptorer, foerfaranden foer deras framstaellning och anvaendning av desamma |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP0557375A1 (fi) |
| JP (1) | JPH06502421A (fi) |
| CN (1) | CN1061595A (fi) |
| AU (1) | AU652399B2 (fi) |
| CA (1) | CA2095224A1 (fi) |
| CZ (1) | CZ80993A3 (fi) |
| FI (1) | FI932206L (fi) |
| HU (1) | HU9301417D0 (fi) |
| IE (1) | IE913922A1 (fi) |
| IS (1) | IS3782A7 (fi) |
| LT (1) | LTIP1718A (fi) |
| MX (1) | MX9101979A (fi) |
| NO (1) | NO931679L (fi) |
| PT (1) | PT99515A (fi) |
| SE (1) | SE9003652D0 (fi) |
| SK (1) | SK46993A3 (fi) |
| WO (1) | WO1992008724A1 (fi) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5194430A (en) * | 1990-05-17 | 1993-03-16 | Merrell Dow Pharmaceuticals Inc. | Heterocyclic-nmda antagonists |
| TW281670B (fi) * | 1993-09-02 | 1996-07-21 | Hoffmann La Roche | |
| US5491241A (en) * | 1993-10-18 | 1996-02-13 | Eli Lilly And Company | Bicyclic intermediates for excitatory amino acid receptor antagonists |
| RS62861B1 (sr) | 2016-02-04 | 2022-02-28 | Takeda Pharmaceuticals Co | Supstituisano piperidin jedinjenje i njegova upotreba |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1248531A (en) * | 1984-04-17 | 1989-01-10 | Jeffrey C. Watkins | 4-substituted piperazine-2-carboxylic acids |
| JPS612519A (ja) * | 1984-04-24 | 1986-01-08 | Aron Kasei Co Ltd | 射出成形法 |
| US4906621A (en) * | 1985-05-24 | 1990-03-06 | Ciba-Geigy Corporation | Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade |
| US4740346A (en) * | 1986-02-26 | 1988-04-26 | The Budd Company | Perimeter resin feeding of composite structures |
| JPS63112129A (ja) * | 1986-10-30 | 1988-05-17 | Toyoda Gosei Co Ltd | 多色樹脂成形用金型 |
| ES2031927T3 (es) * | 1986-11-21 | 1993-01-01 | Ciba-Geigy Ag | Procedimiento para la obtencion de acidos fosfonicos insaturados y derivados. |
-
1990
- 1990-11-15 SE SE9003652A patent/SE9003652D0/xx unknown
-
1991
- 1991-11-05 CN CN91110925A patent/CN1061595A/zh active Pending
- 1991-11-07 SK SK46993A patent/SK46993A3/sk unknown
- 1991-11-07 WO PCT/SE1991/000753 patent/WO1992008724A1/en not_active Ceased
- 1991-11-07 FI FI932206A patent/FI932206L/fi not_active Application Discontinuation
- 1991-11-07 CZ CS93809A patent/CZ80993A3/cs unknown
- 1991-11-07 EP EP91920264A patent/EP0557375A1/en not_active Withdrawn
- 1991-11-07 AU AU89391/91A patent/AU652399B2/en not_active Ceased
- 1991-11-07 JP JP4500566A patent/JPH06502421A/ja active Pending
- 1991-11-07 HU HU931417A patent/HU9301417D0/hu unknown
- 1991-11-07 CA CA002095224A patent/CA2095224A1/en not_active Abandoned
- 1991-11-08 MX MX9101979A patent/MX9101979A/es unknown
- 1991-11-12 IE IE392291A patent/IE913922A1/en unknown
- 1991-11-14 PT PT99515A patent/PT99515A/pt not_active Application Discontinuation
- 1991-11-14 IS IS3782A patent/IS3782A7/is unknown
-
1993
- 1993-05-07 NO NO93931679A patent/NO931679L/no unknown
- 1993-12-30 LT LTIP1718A patent/LTIP1718A/xx not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MX9101979A (es) | 1992-07-08 |
| AU8939191A (en) | 1992-06-11 |
| LTIP1718A (en) | 1995-07-25 |
| FI932206A0 (fi) | 1993-05-14 |
| SE9003652D0 (sv) | 1990-11-15 |
| CA2095224A1 (en) | 1992-05-16 |
| HU9301417D0 (en) | 1993-09-28 |
| JPH06502421A (ja) | 1994-03-17 |
| IE913922A1 (en) | 1992-05-20 |
| WO1992008724A1 (en) | 1992-05-29 |
| PT99515A (pt) | 1992-09-30 |
| IS3782A7 (is) | 1992-05-16 |
| NO931679D0 (no) | 1993-05-07 |
| NO931679L (no) | 1993-05-07 |
| EP0557375A1 (en) | 1993-09-01 |
| CN1061595A (zh) | 1992-06-03 |
| FI932206L (fi) | 1993-05-14 |
| SK46993A3 (en) | 1993-10-06 |
| CZ80993A3 (en) | 1994-02-16 |
| AU652399B2 (en) | 1994-08-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application lapsed |