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FI912499L - Pyrido/3,4-b/pyrrolo/1,2-e//1,4,5/ oxadiazepiner och daermed naerbeslaektade analoger, foerfarande foer deras framstaellning och deras anvaendning som laekemedel. - Google Patents

Pyrido/3,4-b/pyrrolo/1,2-e//1,4,5/ oxadiazepiner och daermed naerbeslaektade analoger, foerfarande foer deras framstaellning och deras anvaendning som laekemedel. Download PDF

Info

Publication number
FI912499L
FI912499L FI912499A FI912499A FI912499L FI 912499 L FI912499 L FI 912499L FI 912499 A FI912499 A FI 912499A FI 912499 A FI912499 A FI 912499A FI 912499 L FI912499 L FI 912499L
Authority
FI
Finland
Prior art keywords
och
deras
oxadiazepiner
naerbeslaektade
daermed
Prior art date
Application number
FI912499A
Other languages
English (en)
Other versions
FI912499A7 (fi
FI912499A0 (fi
Inventor
Richard C Effland
Larry Davis
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI912499A0 publication Critical patent/FI912499A0/fi
Publication of FI912499L publication Critical patent/FI912499L/fi
Publication of FI912499A7 publication Critical patent/FI912499A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI912499A 1990-05-25 1991-05-23 Pyrido/3,4-b/pyrrolo/1,2-e//1,4,5/oksadiatsepiineja ja niille läheisiäanalogeja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä FI912499A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/529,082 US5015637A (en) 1990-05-25 1990-05-25 Pyrido[3,4-b]pyrrolo[1,2-e][1,4,5]oxadiazepines

Publications (3)

Publication Number Publication Date
FI912499A0 FI912499A0 (fi) 1991-05-23
FI912499L true FI912499L (fi) 1991-11-26
FI912499A7 FI912499A7 (fi) 1991-11-26

Family

ID=24108456

Family Applications (1)

Application Number Title Priority Date Filing Date
FI912499A FI912499A7 (fi) 1990-05-25 1991-05-23 Pyrido/3,4-b/pyrrolo/1,2-e//1,4,5/oksadiatsepiineja ja niille läheisiäanalogeja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä

Country Status (22)

Country Link
US (1) US5015637A (fi)
EP (1) EP0458331B1 (fi)
JP (1) JP3090500B2 (fi)
KR (1) KR100286405B1 (fi)
AT (1) ATE183746T1 (fi)
AU (1) AU638572B2 (fi)
CA (1) CA2043229C (fi)
CS (1) CS157191A3 (fi)
DE (1) DE69131546T2 (fi)
DK (1) DK0458331T3 (fi)
ES (1) ES2135383T3 (fi)
FI (1) FI912499A7 (fi)
GR (1) GR3031538T3 (fi)
HU (1) HU207520B (fi)
IE (1) IE911788A1 (fi)
IL (1) IL98231A (fi)
MX (1) MX25922A (fi)
NO (1) NO911998L (fi)
NZ (1) NZ238238A (fi)
PL (1) PL290405A1 (fi)
PT (1) PT97762B (fi)
ZA (1) ZA913951B (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69426804D1 (de) * 1993-05-27 2001-04-12 Icos Corp Cyclisch gmp bindende cyclisch gmp spezifische phosphodiesterase materialien und verfahren.
TWI316939B (en) * 2001-12-18 2009-11-11 Syngenta Participations Ag Process for the preparation of organic compounds
WO2011133291A2 (en) 2010-04-18 2011-10-27 Chang Jun Yu Pillow with positionable inserts

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4029672A (en) * 1976-02-26 1977-06-14 American Hoechst Corporation Aminoalkylpyrrolobenzoxazalkanes
US4045448A (en) * 1976-02-26 1977-08-30 American Hoechst Corporation Pyrrolo[2,1-c][1,4]benzoxazepine and benzoxazocine derivatives
FI803908L (fi) * 1979-12-21 1981-06-22 Sandoz Ag Nya pyrrolobenszotriazepiner deras framstaellning och dessa innehaollande farmaceutiska foereningar
US4608374A (en) * 1983-11-07 1986-08-26 Hoechst-Roussel Pharmaceuticals Inc. 11-substituted 5H,11H-pyrrolo[2,1-c][1,4]benzoxazepines as antipsychotic and analgesic agents
US4794110A (en) * 1987-07-20 1988-12-27 Hoechst-Roussel Pharmaceuticals, Inc. 5-Aryl-11-substituted-5H,11H-pyrrolo[2,1-c][1,4]benzoxazepined as analgesic and hypotensive agents
US4879382A (en) * 1988-07-25 1989-11-07 Hoechst-Roussel Pharmaceuticals, Inc. Pyrido(3,4-f)pyrrolo(1,2-b)(1,2,5)triazepines

Also Published As

Publication number Publication date
DK0458331T3 (da) 2000-03-13
DE69131546T2 (de) 2000-03-23
DE69131546D1 (de) 1999-09-30
KR910020018A (ko) 1991-12-19
AU638572B2 (en) 1993-07-01
IL98231A (en) 1994-11-28
NO911998L (no) 1991-11-26
NZ238238A (en) 1993-06-25
AU7621391A (en) 1991-11-28
JPH04235186A (ja) 1992-08-24
EP0458331B1 (en) 1999-08-25
PT97762A (pt) 1992-02-28
KR100286405B1 (ko) 2001-04-16
JP3090500B2 (ja) 2000-09-18
ATE183746T1 (de) 1999-09-15
EP0458331A1 (en) 1991-11-27
IE911788A1 (en) 1991-12-04
MX25922A (es) 1993-10-01
HUT60744A (en) 1992-10-28
PL290405A1 (en) 1992-08-24
ES2135383T3 (es) 1999-11-01
GR3031538T3 (en) 2000-01-31
CA2043229A1 (en) 1991-11-26
US5015637A (en) 1991-05-14
CA2043229C (en) 2003-02-11
CS157191A3 (en) 1992-01-15
HU207520B (en) 1993-04-28
FI912499A7 (fi) 1991-11-26
PT97762B (pt) 1998-10-30
HU911755D0 (en) 1991-12-30
NO911998D0 (no) 1991-05-24
ZA913951B (en) 1992-03-25
FI912499A0 (fi) 1991-05-23
IL98231A0 (en) 1992-06-21

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