FI914071A7 - Uudet hetratsepinoidiset amidit - Google Patents

Uudet hetratsepinoidiset amidit Download PDF

Info

Publication number: FI914071A7
Authority: FI; Finland
Prior art keywords: hetrazepinoid; amides; new; new hetrazepinoid; hetrazepinoid amides
Prior art date: 1990-08-30

Application number

FI914071A

Other languages

English (en)

Swedish (sv)

Other versions

FI914071A0 (fi

FI914071L (fi

Inventor

Karl-Hainz Weber

Ulrike Küfner-Mühl

Wolf-Dietrich Bechtel

Werner Stransky

Hubert Heuer

Franz Birke

Original Assignee

Boehringer Ingelheim Kg

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-08-30

Filing date

1991-08-29

Publication date

1992-03-01

1991-08-29 Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg

1991-08-29 Publication of FI914071A0 publication Critical patent/FI914071A0/fi

1992-03-01 Publication of FI914071A7 publication Critical patent/FI914071A7/fi

1992-03-01 Publication of FI914071L publication Critical patent/FI914071L/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Urology & Nephrology (AREA)
Pulmonology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Hematology (AREA)
Diabetes (AREA)
Vascular Medicine (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

FI914071A 1990-08-30 1991-08-29 Nya hetrazepinoida amider. FI914071L (fi)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE4027470A DE4027470A1 (de)	1990-08-30	1990-08-30	Neue hetrazepinoide amide

Publications (3)

Publication Number	Publication Date
FI914071A0 FI914071A0 (fi)	1991-08-29
FI914071A7 true FI914071A7 (fi)	1992-03-01
FI914071L FI914071L (fi)	1992-03-01

Family

ID=6413254

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI914071A FI914071L (fi)	1990-08-30	1991-08-29	Nya hetrazepinoida amider.

Country Status (17)

Country	Link
US (1)	US5698552A (fi)
EP (1)	EP0475204A3 (fi)
JP (1)	JPH04261181A (fi)
KR (1)	KR920004394A (fi)
AU (1)	AU8346291A (fi)
CA (1)	CA2050268A1 (fi)
CS (1)	CS265391A3 (fi)
DE (1)	DE4027470A1 (fi)
FI (1)	FI914071L (fi)
HU (1)	HUT62007A (fi)
IE (1)	IE913043A1 (fi)
IL (1)	IL99325A0 (fi)
MX (1)	MX9100845A (fi)
NO (1)	NO913391L (fi)
PL (1)	PL291562A1 (fi)
PT (1)	PT98816B (fi)
ZA (1)	ZA916902B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0656004A1 (en) *	1992-08-20	1995-06-07	Cytomed, Inc.	Dual functional anti-inflammatory and immunosuppressive agents
US5821924A (en) *	1992-09-04	1998-10-13	Elonex I.P. Holdings, Ltd.	Computer peripherals low-power-consumption standby system
US5389952A (en) *	1992-12-02	1995-02-14	Cordata Inc.	Low-power-consumption monitor standby system
US5302590A (en) *	1992-12-18	1994-04-12	Hoffmann-La Roche Inc.	Compounds useful as dual antagonists of platelet activating factor and leukotriene D4
EA001732B1 (ru) *	1996-09-13	2001-08-27	Велфайд Корпорейшн	Тиенотриазолодиазепиновые соединения и лекарственное средство
US9249161B2 (en)	2010-12-02	2016-02-02	Constellation Pharmaceuticals, Inc.	Bromodomain inhibitors and uses thereof
AR084070A1 (es)	2010-12-02	2013-04-17	Constellation Pharmaceuticals Inc	Inhibidores del bromodominio y usos de los mismos
US9422292B2 (en)	2011-05-04	2016-08-23	Constellation Pharmaceuticals, Inc.	Bromodomain inhibitors and uses thereof
US9328117B2 (en)	2011-06-17	2016-05-03	Constellation Pharmaceuticals, Inc.	Bromodomain inhibitors and uses thereof
TWI602820B (zh)	2012-06-06	2017-10-21	星宿藥物公司	溴域抑制劑及其用途
WO2013184878A1 (en)	2012-06-06	2013-12-12	Constellation Pharmaceuticals, Inc.	Benzo [b] isoxazoloazepine bromodomain inhibitors and uses thereof
ES2725928T3 (es)	2014-06-20	2019-09-30	Constellation Pharmaceuticals Inc	Formas cristalinas de 2-((4S)-6-(4-clorofenil)-1-metil-4H-benzo[c]isoxazolo[4,5-e]azepin-4-il)acetamida

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3435973A1 (de) *	1984-10-01	1986-04-10	Boehringer Ingelheim KG, 6507 Ingelheim	Diazepine enthaltende pharmazeutische zusammensetzungen mit paf-antagonistischer wirkung
DE3502392A1 (de) *	1985-01-25	1986-07-31	Boehringer Ingelheim KG, 6507 Ingelheim	Neue thieno-triazolo-1,4-diazepino-2- carbonsaeureamide, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen
ES2037013T3 (es) *	1986-01-21	1993-06-16	Boehringer Ingelheim Kg	Procedimiento para preparar tieno-1,4-diazepinas.
PH30676A (en) *	1986-07-22	1997-09-16	Boehringer Ingelhein Kg	Hetrazepine compounds which have useful pharmaceutical utility
CA1324863C (en) *	1988-01-30	1993-11-30	Minoru Moriwaki	Thienotriazolodiazepine compounds and pharmaceutical uses thereof
FI95708C (fi) *	1988-10-31	1996-03-11	Eisai Co Ltd	Analogiamenetelmä 1,4-diatsepiinijohdannaisen ja sen farmaseuttisesti sopivan suolan valmistamiseksi
EP0368175A1 (de) *	1988-11-06	1990-05-16	Boehringer Ingelheim Kg	3S,7S-3-(Morpholinocarbonyl)-5-(2-chlorphenyl)-7,10-dimethyl-3,4-dihydro-2H,7H-cyclopenta[4,5]thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin.
DE3909012A1 (de) *	1989-03-18	1990-09-20	Boehringer Ingelheim Kg	Verbessertes verfahren zur herstellung von enantiomerenreinen hetrazepinen
GB8907256D0 (en) *	1989-03-31	1989-05-17	Rech Et D Applic Scient Scras	New derivatives of hetrazepine as anti-asthmatic anti-allergic and gastro-intestinal protectors
EP0407955A1 (de) *	1989-07-12	1991-01-16	Boehringer Ingelheim Kg	Neue Hetrazepine mit PAF-antagonistischer Wirkung, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE4010528A1 (de) *	1990-04-02	1991-10-17	Boehringer Ingelheim Kg	Praeparativ chromatographisches trennverfahren zur herstellung enantiomerenreiner hetrazepine

1990
- 1990-08-30 DE DE4027470A patent/DE4027470A1/de not_active Withdrawn
1991
- 1991-08-28 IL IL99325A patent/IL99325A0/xx unknown
- 1991-08-28 MX MX9100845A patent/MX9100845A/es unknown
- 1991-08-28 CS CS912653A patent/CS265391A3/cs unknown
- 1991-08-29 NO NO91913391A patent/NO913391L/no unknown
- 1991-08-29 EP EP19910114518 patent/EP0475204A3/de not_active Withdrawn
- 1991-08-29 IE IE304391A patent/IE913043A1/en unknown
- 1991-08-29 PL PL29156291A patent/PL291562A1/xx unknown
- 1991-08-29 HU HU912821A patent/HUT62007A/hu unknown
- 1991-08-29 FI FI914071A patent/FI914071L/fi not_active Application Discontinuation
- 1991-08-29 JP JP3218916A patent/JPH04261181A/ja active Pending
- 1991-08-29 PT PT98816A patent/PT98816B/pt active IP Right Grant
- 1991-08-29 CA CA002050268A patent/CA2050268A1/en not_active Abandoned
- 1991-08-30 KR KR1019910015086A patent/KR920004394A/ko not_active Withdrawn
- 1991-08-30 ZA ZA916902A patent/ZA916902B/xx unknown
- 1991-08-30 AU AU83462/91A patent/AU8346291A/en not_active Abandoned
1995
- 1995-05-31 US US08/453,038 patent/US5698552A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
EP0475204A2 (de)	1992-03-18
FI914071A0 (fi)	1991-08-29
HU912821D0 (en)	1993-03-29
CS265391A3 (en)	1992-03-18
MX9100845A (es)	1992-04-01
IL99325A0 (en)	1992-07-15
PT98816A (pt)	1992-07-31
AU8346291A (en)	1992-03-05
FI914071L (fi)	1992-03-01
CA2050268A1 (en)	1992-03-01
EP0475204A3 (en)	1992-05-13
JPH04261181A (ja)	1992-09-17
PT98816B (pt)	1999-01-29
KR920004394A (ko)	1992-03-27
US5698552A (en)	1997-12-16
HUT62007A (en)	1993-03-29
NO913391D0 (no)	1991-08-29
IE913043A1 (en)	1992-03-11
PL291562A1 (en)	1992-10-05
NO913391L (no)	1992-03-02
DE4027470A1 (de)	1992-03-05
ZA916902B (en)	1992-04-29

Publication	Publication Date	Title
FI914071A7 (fi)	1992-03-01	Uudet hetratsepinoidiset amidit
ATA210290A (de)	1991-10-15	Lotpille
BR9102325A (pt)	1992-01-07	Ebulidor
FI911351A7 (fi)	1991-09-22	Uusia 8-sulfamyylimetyleeni-2-aminotetraliineja
DE69118732D1 (de)	1996-05-23	Elektrophotorezeptor
ATA80690A (de)	1997-12-15	Alpinschi
ATA200090A (de)	1991-06-15	Pianino
NO932219D0 (no)	1993-06-16	Skadedyrdrepende forbindelser
ATA209290A (de)	1992-10-15	Diaraehmchen
BR9103647A (pt)	1992-05-19	Tioesteres
ATA237490A (de)	1991-12-15	Rinnenstein
BR9101437A (pt)	1991-11-26	Copoliester
SE9002439D0 (sv)	1990-07-16	New amides ii
IS3664A7 (is)	1991-06-23	Ný amíð
BR9003611A (pt)	1992-02-18	Hidrobaliador
BR9002505A (pt)	1991-01-08	Venturbo
SE9002698D0 (sv)	1990-08-20	New use
BR7002609U (pt)	1992-08-04	Camelomovel
ATA70290A (de)	1991-08-15	Anzeigetafel
BR7001467U (pt)	1992-03-03	Halleybus
BR7001392U (pt)	1992-01-21	Lixa
BR7001143U (pt)	1991-01-22	Minitecnigrafo
BR7000887U (pt)	1991-11-19	Informapa
BR7000857U (pt)	1991-11-19	Acucareiro dosador
BR7000792U (pt)	1992-11-03	Microbebedouro

Legal Events

Date	Code	Title	Description
1994-03-07	FD	Application lapsed