FI843219L - Nya karboxylsyraestrar. - Google Patents

Nya karboxylsyraestrar. Download PDF

Info

Publication number: FI843219L
Authority: FI; Finland
Prior art keywords: acid esters; carboxyl acid; new carboxyl; new; esters
Prior art date: 1983-08-18

Application number

FI843219A

Other languages

English (en)

Other versions

FI843219A0 (fi

FI80888B (fi

FI80888C (fi

Inventor

Julius Schmidlin

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-08-18

Filing date

1984-08-15

Publication date

1985-02-19

1984-08-15 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1984-08-15 Publication of FI843219A0 publication Critical patent/FI843219A0/fi

1985-02-19 Publication of FI843219L publication Critical patent/FI843219L/fi

1990-04-30 Publication of FI80888B publication Critical patent/FI80888B/fi

1990-08-10 Application granted granted Critical

1990-08-10 Publication of FI80888C publication Critical patent/FI80888C/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/74—Esters of carboxylic acids having an esterified carboxyl group bound to a carbon atom of a ring other than a six-membered aromatic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
- C07J71/0015—Oxiranes at position 9(11)
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Pain & Pain Management (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Rheumatology (AREA)
Engineering & Computer Science (AREA)
Steroid Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Measuring Pulse, Heart Rate, Blood Pressure Or Blood Flow (AREA)
Ultra Sonic Daignosis Equipment (AREA)
Heat Sensitive Colour Forming Recording (AREA)
Photoreceptors In Electrophotography (AREA)
Fats And Perfumes (AREA)

FI843219A 1983-08-18 1984-08-15 Foerfarande foer framstaellning av terapeutiskt verkande steroida karboxylsyraestrar. FI80888C (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH451283		1983-08-18
CH451283		1983-08-18

Publications (4)

Publication Number	Publication Date
FI843219A0 FI843219A0 (fi)	1984-08-15
FI843219L true FI843219L (fi)	1985-02-19
FI80888B FI80888B (fi)	1990-04-30
FI80888C FI80888C (fi)	1990-08-10

Family

ID=4277476

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI843219A FI80888C (fi)	1983-08-18	1984-08-15	Foerfarande foer framstaellning av terapeutiskt verkande steroida karboxylsyraestrar.

Country Status (21)

Country	Link
US (1)	US4607028A (fi)
EP (1)	EP0135476B1 (fi)
JP (1)	JPS6058999A (fi)
KR (1)	KR850001725A (fi)
AT (1)	ATE37186T1 (fi)
AU (1)	AU3204484A (fi)
CA (1)	CA1234564A (fi)
CY (1)	CY1593A (fi)
DD (1)	DD227966A5 (fi)
DE (1)	DE3474025D1 (fi)
DK (1)	DK160993C (fi)
ES (1)	ES535242A0 (fi)
FI (1)	FI80888C (fi)
GR (1)	GR80131B (fi)
HK (1)	HK42791A (fi)
HU (1)	HUT34991A (fi)
IL (1)	IL72702A0 (fi)
NO (1)	NO160212C (fi)
PT (1)	PT79106B (fi)
SG (1)	SG32091G (fi)
ZA (1)	ZA846406B (fi)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL78144A0 (en) *	1985-04-04	1986-07-31	Draco Ab	Novel androstane-17beta-carboxylic acid esters
JPH04506066A (ja) *	1989-06-16	1992-10-22	ジ・アップジョン・カンパニー	脈管形成を抑制するためのスラミン・タイプの化合物および脈管形成抑止ステロイド類
FR2701262B1 (fr) *	1993-02-05	1995-03-24	Roussel Uclaf	Nouveau procédé de préparation de stéroïdes 6 alpa, 9 alpha-difluorés et nouveaus intermédiaires.
JPH07119308A (ja) *	1993-10-27	1995-05-09	Koa:Kk	移動作業床による外壁貼りの吊り支え工法並にその装置
GB9501286D0 (en) *	1995-01-24	1995-03-15	Ciba Geigy Ag	Pharmaceutical compositions and preparations thereof
US5981517A (en) *	1996-05-09	1999-11-09	Soft Drugs, Inc.	Androstene derivatives
AUPP583198A0 (en) *	1998-09-11	1998-10-01	Soltec Research Pty Ltd	Mousse composition
GB0015876D0 (en) *	2000-06-28	2000-08-23	Novartis Ag	Organic compounds
US6777400B2 (en) *	2000-08-05	2004-08-17	Smithkline Beecham Corporation	Anti-inflammatory androstane derivative compositions
US6759398B2 (en)	2000-08-05	2004-07-06	Smithkline Beecham Corporation	Anti-inflammatory androstane derivative
US6750210B2 (en) *	2000-08-05	2004-06-15	Smithkline Beecham Corporation	Formulation containing novel anti-inflammatory androstane derivative
US6858593B2 (en) *	2000-08-05	2005-02-22	Smithkline Beecham Corporation	Anti-inflammatory androstane derivative compositions
GB0019172D0 (en) *	2000-08-05	2000-09-27	Glaxo Group Ltd	Novel compounds
US6777399B2 (en) *	2000-08-05	2004-08-17	Smithkline Beecham Corporation	Anti-inflammatory androstane derivative compositions
US6858596B2 (en) *	2000-08-05	2005-02-22	Smithkline Beecham Corporation	Formulation containing anti-inflammatory androstane derivative
US6787532B2 (en) *	2000-08-05	2004-09-07	Smithkline Beecham Corporation	Formulation containing anti-inflammatory androstane derivatives
KR100889426B1 (ko) *	2000-08-05	2009-03-23	글락소 그룹 리미티드	항염증제로서의 6.알파.,9.알파.-디플루오로-17.알파.-'(2-푸라닐카르복실)옥시-11.베타.-히드록시-16.알파.-메틸-3-옥소-안드로스트-1,4-디엔-17-카르보티오산 ｓ-플루오로메틸 에스테르
GB0029562D0 (en) *	2000-12-04	2001-01-17	Novartis Ag	Organic compounds
UA77656C2 (en) *	2001-04-07	2007-01-15	Glaxo Group Ltd	S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent
AU2002253342B2 (en) *	2001-04-30	2007-01-04	Glaxo Group Limited	Novel anti-inflammatory androstane derivatives
JP2003095382A (ja) *	2001-09-25	2003-04-03	Ishikawajima Harima Heavy Ind Co Ltd	タンクのマンホール構造
GB0202216D0 (en) *	2002-01-31	2002-03-20	Glaxo Group Ltd	Novel compounds
US20050175545A1 (en) *	2002-02-04	2005-08-11	Keith Biggadike	Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist
GB0202635D0 (en) *	2002-02-05	2002-03-20	Glaxo Wellcome Mfg Pte Ltd	Formulation containing novel anti-inflammatory androstane derivative
GB2389530B (en)	2002-06-14	2007-01-10	Cipla Ltd	Pharmaceutical compositions
GB0507165D0 (en) *	2005-04-08	2005-05-18	Glaxo Group Ltd	Novel crystalline pharmaceutical product
GB0615108D0 (en) *	2006-07-28	2006-09-06	Glaxo Group Ltd	Novel formulations

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1384372A (en) *	1971-01-20	1975-02-19	Glaxo Lab Ltd	Dereivatives of 17alpha-hydroxyandrost-4-ene-17beta-carboxylic acids
GB1514476A (en) *	1974-08-30	1978-06-14	Glaxo Lab Ltd	Alkyl and haloalkyl androst-4-ene and androsta-1,4-diene-17beta-carboxylates
JPS5297597A (en) *	1976-02-09	1977-08-16	Walt Disney Prod	Guide device of ship
JPS5938239B2 (ja) *	1976-02-12	1984-09-14	グラクソ・ラボラトリ−ス・リミテツド	新規ステロイド化合物
CH628355A5 (de) *	1976-02-24	1982-02-26	Ciba Geigy Ag	Verfahren zur herstellung neuer androstadien-17beta-carbonsaeuren und ihrer ester und salze.
CH634081A5 (en) *	1977-04-13	1983-01-14	Ciba Geigy Ag	Process for the preparation of novel androstadiene-17beta-carboxylic acid esters
ZA814440B (en) *	1980-07-10	1982-10-27	Otsuka Pharma Co Ltd	Soft steroids having anti-inflammatory activity

1984
- 1984-08-09 US US06/639,033 patent/US4607028A/en not_active Expired - Lifetime
- 1984-08-13 DE DE8484810397T patent/DE3474025D1/de not_active Expired
- 1984-08-13 EP EP84810397A patent/EP0135476B1/de not_active Expired
- 1984-08-13 AT AT84810397T patent/ATE37186T1/de active
- 1984-08-15 FI FI843219A patent/FI80888C/fi not_active IP Right Cessation
- 1984-08-16 IL IL72702A patent/IL72702A0/xx unknown
- 1984-08-16 CA CA000461216A patent/CA1234564A/en not_active Expired
- 1984-08-17 JP JP59170498A patent/JPS6058999A/ja active Granted
- 1984-08-17 HU HU843129A patent/HUT34991A/hu unknown
- 1984-08-17 AU AU32044/84A patent/AU3204484A/en not_active Abandoned
- 1984-08-17 DK DK396284A patent/DK160993C/da not_active IP Right Cessation
- 1984-08-17 KR KR1019840004956A patent/KR850001725A/ko not_active Withdrawn
- 1984-08-17 ES ES535242A patent/ES535242A0/es active Granted
- 1984-08-17 PT PT79106A patent/PT79106B/pt not_active IP Right Cessation
- 1984-08-17 DD DD84266390A patent/DD227966A5/de unknown
- 1984-08-17 GR GR80131A patent/GR80131B/el unknown
- 1984-08-17 ZA ZA846406A patent/ZA846406B/xx unknown
- 1984-08-17 NO NO843298A patent/NO160212C/no unknown
1991
- 1991-05-02 SG SG320/91A patent/SG32091G/en unknown
- 1991-05-30 HK HK427/91A patent/HK42791A/xx not_active IP Right Cessation
1992
- 1992-04-03 CY CY1593A patent/CY1593A/xx unknown

Also Published As

Publication number	Publication date
ES8601234A1 (es)	1985-11-01
HK42791A (en)	1991-06-07
DK396284A (da)	1985-02-19
HUT34991A (en)	1985-05-28
EP0135476A2 (de)	1985-03-27
PT79106A (en)	1984-09-01
CA1234564A (en)	1988-03-29
GR80131B (en)	1984-12-19
IL72702A0 (en)	1984-11-30
NO160212B (no)	1988-12-12
NO160212C (no)	1989-03-22
DK396284D0 (da)	1984-08-17
SG32091G (en)	1991-06-21
US4607028A (en)	1986-08-19
FI843219A0 (fi)	1984-08-15
JPH0253440B2 (fi)	1990-11-16
ES535242A0 (es)	1985-11-01
NO843298L (no)	1985-02-19
FI80888B (fi)	1990-04-30
KR850001725A (ko)	1985-04-01
JPS6058999A (ja)	1985-04-05
EP0135476A3 (en)	1985-12-18
CY1593A (en)	1992-04-03
FI80888C (fi)	1990-08-10
EP0135476B1 (de)	1988-09-14
DD227966A5 (de)	1985-10-02
DK160993C (da)	1991-11-04
DK160993B (da)	1991-05-13
AU3204484A (en)	1985-02-21
PT79106B (en)	1986-11-14
DE3474025D1 (en)	1988-10-20
ATE37186T1 (de)	1988-09-15
ZA846406B (en)	1985-03-27

Publication	Publication Date	Title
FI843219L (fi)	1985-02-19	Nya karboxylsyraestrar.
FI841813L (fi)	1984-11-18	Foerfarande foer framstaellning av n- fosfonometylglycinsyra.
FI844424A0 (fi)	1984-11-09	Nya atriumpeptider.
FI845075A7 (fi)	1985-06-24	Bentsoehappojohdannaisia.
FI841759L (fi)	1984-11-04	Foerfarande foer framstaellning av nya fluoralkoxifoereningar.
FI80885B (fi)	1990-04-30	Framstaellning av nya guaninderivat.
FI881501A7 (fi)	1988-10-03	5-substituerade kinolon- och naftyridonkarboxylsyraderivat.
FI841758L (fi)	1984-11-04	Foerfarande foer framstaellning av nya tricykliska etrar.
FI86987B (fi)	1992-07-31	Foerfarande foer framstaellning av nya terapeutiskt anvaendbara fenylkinolinkarboxylsyraderivat.
FI841259L (fi)	1984-10-01	Nya farmaceutiska foereningar.
FI841738A7 (fi)	1984-11-04	Imidazol-etanolestrar.
FI842960A0 (fi)	1984-07-25	Nya herbicider i form av aminoetylfosfoner tillhoerande sulfonimiderna.
FI841925A0 (fi)	1984-05-14	Nya indolfoereningar.
FI862462A7 (fi)	1986-12-14	Nya sulfonsyraestrar.
FI842547A0 (fi)	1984-06-25	Foerfarande foer framstaellning av nya spirosuckinimider.
ATE42751T1 (de)	1989-05-15	Carboxylsaeureesterderivate von deglucoteicoplanin.
FI841619A0 (fi)	1984-04-25	Nya pyrimidonderivat.
DE3463654D1 (de)	1987-06-19	Pyridinylmethylamino-arylic acids
ATE16806T1 (de)	1985-12-15	3-methylflavon-8-carboxylsaeureester.
FI843332A0 (fi)	1984-08-23	Nya pesticidala heterocykliska foereningar.
FI844466A0 (fi)	1984-11-14	Nya amidfoereningar.
FI73988B (fi)	1987-08-31	Foerfarande foer framstaellning av nya kardiotoniskt verkande pyridinyl-2-pyrimidinaminderivat.
FI814059A7 (fi)	1982-06-19	Propionihappoesterit.
FI841376L (fi)	1985-06-24	Nya oralt administrerbara galeniska former av sulpirid.
FI841461A7 (fi)	1984-10-29	Foerfarande foer framstaellning av nya substituerade piperazin-1-yl-aettiksyra-amider.

Legal Events

Date	Code	Title	Description
1997-08-26	PC	Transfer of assignment of patent	Owner name: NOVARTIS AG
2004-08-31	MM	Patent lapsed	Owner name: NOVARTIS AG