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FI823757L - Cis-endo-2-azabicyklo/3,3.0/oktan-3-karboxylsyraderivat, foerfarande foer deras framstaellning, desinnehaollande aemnen och deras anvaendning - Google Patents

Cis-endo-2-azabicyklo/3,3.0/oktan-3-karboxylsyraderivat, foerfarande foer deras framstaellning, desinnehaollande aemnen och deras anvaendning

Info

Publication number
FI823757L
FI823757L FI823757A FI823757A FI823757L FI 823757 L FI823757 L FI 823757L FI 823757 A FI823757 A FI 823757A FI 823757 A FI823757 A FI 823757A FI 823757 L FI823757 L FI 823757L
Authority
FI
Finland
Prior art keywords
syraderated
foreigned
desinnehaollande
azabicyclo
endo
Prior art date
Application number
FI823757A
Other languages
English (en)
Other versions
FI81087C (fi
FI81087B (fi
FI823757A0 (fi
Inventor
Volker Teetz
Rolf Geiger
Hansjoerg Urbach
Reinhard Becker
Benrward Schoelkens
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25797115&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI823757(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoechst Ag filed Critical Hoechst Ag
Priority to FI895951A priority Critical patent/FI895951A0/fi
Publication of FI823757A0 publication Critical patent/FI823757A0/fi
Publication of FI823757L publication Critical patent/FI823757L/fi
Priority to FI863401A priority patent/FI83633C/fi
Priority to FI863400A priority patent/FI80442C/fi
Application granted granted Critical
Publication of FI81087B publication Critical patent/FI81087B/fi
Publication of FI81087C publication Critical patent/FI81087C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Cardiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI823757A 1981-11-05 1982-11-03 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1-acyl-2-azabicyklo/3.3.0/-3-karboxylsyror. FI81087C (fi)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FI895951A FI895951A0 (fi) 1981-11-05 1982-11-03 Foerfarande foer framstaellning av cis, endo-2-azabicyklo/3.3.0/oktan-3-karboxylsyraderivat.
FI863401A FI83633C (fi) 1981-11-05 1986-08-22 Foerfarande foer framstaellning av aminosyraderivat och i foerfarandet anvaend mellanprodukt.
FI863400A FI80442C (fi) 1981-11-05 1986-08-22 Cis, endo-2-azabicyklo/3.3.0/oktan-3 -karboxylsyror och deras estrar, samt foerfarande foer deras framstaellning.

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3143946 1981-11-05
DE3143946 1981-11-05
DE3226768 1982-07-17
DE19823226768 DE3226768A1 (de) 1981-11-05 1982-07-17 Derivate der cis, endo-2-azabicyclo-(3.3.0)-octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung

Publications (4)

Publication Number Publication Date
FI823757A0 FI823757A0 (fi) 1982-11-03
FI823757L true FI823757L (fi) 1983-05-06
FI81087B FI81087B (fi) 1990-05-31
FI81087C FI81087C (fi) 1990-09-10

Family

ID=25797115

Family Applications (1)

Application Number Title Priority Date Filing Date
FI823757A FI81087C (fi) 1981-11-05 1982-11-03 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 1-acyl-2-azabicyklo/3.3.0/-3-karboxylsyror.

Country Status (31)

Country Link
US (4) US4727160A (fi)
EP (2) EP0150263B1 (fi)
JP (3) JPH02104573A (fi)
KR (1) KR890000007B1 (fi)
AR (1) AR240675A1 (fi)
AU (3) AU565200B2 (fi)
BG (1) BG60532B2 (fi)
CA (1) CA1187087A (fi)
CS (1) CS247159B2 (fi)
CZ (1) CZ416291A3 (fi)
DD (2) DD203047A5 (fi)
DE (3) DE3226768A1 (fi)
DK (2) DK166624C (fi)
DZ (1) DZ473A1 (fi)
ES (3) ES8307746A1 (fi)
FI (1) FI81087C (fi)
GR (1) GR77381B (fi)
HK (1) HK74889A (fi)
HU (2) HU186594B (fi)
IE (1) IE56476B1 (fi)
IL (1) IL67172A (fi)
JO (1) JO1224B1 (fi)
LU (1) LU88260I2 (fi)
MA (1) MA19639A1 (fi)
NL (1) NL930039I2 (fi)
NO (2) NO156940C (fi)
NZ (1) NZ202378A (fi)
PH (2) PH22417A (fi)
PT (1) PT75792A (fi)
SG (1) SG1189G (fi)
SU (1) SU1277895A3 (fi)

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US4879403A (en) 1989-11-07
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IE56476B1 (en) 1991-08-14
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NL930039I1 (nl) 1993-08-02
FI81087B (fi) 1990-05-31
DE3226768A1 (de) 1983-05-26
FI823757A0 (fi) 1982-11-03
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AU586316B2 (en) 1989-07-06
PT75792A (de) 1982-12-01
MA19639A1 (fr) 1983-07-01
ES8307746A1 (es) 1983-08-01
PH22417A (en) 1988-09-12
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SU1277895A3 (ru) 1986-12-15
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