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FI20040657A7 - Kortikotropiinia vapauttavan tekijän antagonisteja - Google Patents

Kortikotropiinia vapauttavan tekijän antagonisteja Download PDF

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Publication number
FI20040657A7
FI20040657A7 FI20040657A FI20040657A FI20040657A7 FI 20040657 A7 FI20040657 A7 FI 20040657A7 FI 20040657 A FI20040657 A FI 20040657A FI 20040657 A FI20040657 A FI 20040657A FI 20040657 A7 FI20040657 A7 FI 20040657A7
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FI
Finland
Prior art keywords
corticotropin
releasing factor
factor antagonists
antagonists
releasing
Prior art date
Application number
FI20040657A
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English (en)
Swedish (sv)
Other versions
FI20040657L (fi
Inventor
Yuhpyng L Chen
Original Assignee
Pfizer
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Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI20040657A7 publication Critical patent/FI20040657A7/fi
Publication of FI20040657L publication Critical patent/FI20040657L/fi

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/69—Two or more oxygen atoms
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    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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FI20040657A 1994-06-08 2004-05-10 Kortikotropiinia vapauttavan tekijän antagonisteja FI20040657L (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25551494A 1994-06-08 1994-06-08
PCT/IB1995/000439 WO1995033750A1 (en) 1994-06-08 1995-06-06 Corticotropin releasing factor antagonists

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FI20040657A7 true FI20040657A7 (fi) 2004-05-10
FI20040657L FI20040657L (fi) 2004-05-10

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FI964894A FI114469B (fi) 1994-06-08 1996-12-05 Kortikotropiinia vapauttavan tekijän antagonisteja
FI20040657A FI20040657L (fi) 1994-06-08 2004-05-10 Kortikotropiinia vapauttavan tekijän antagonisteja

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EP (1) EP0764166B1 (fi)
JP (3) JP3193055B2 (fi)
KR (2) KR100418240B1 (fi)
CN (2) CN1049659C (fi)
AT (1) ATE196295T1 (fi)
AU (1) AU692548B2 (fi)
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WO (1) WO1995033750A1 (fi)
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Families Citing this family (188)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995029909A1 (en) * 1994-04-29 1995-11-09 Pfizer Inc. Novel acyclic and cyclic amides as neurotransmitter release enhancers
EP0729758A3 (en) * 1995-03-02 1997-10-29 Pfizer Pyrazolopyrimidines and pyrrolopyrimidines for the treatment of neuronal and other diseases
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NO310234B1 (no) 2001-06-11
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DE69518841T2 (de) 2001-01-11
CN1150428A (zh) 1997-05-21
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FI114469B (fi) 2004-10-29
FI964894A0 (fi) 1996-12-05
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DK0764166T3 (da) 2000-10-09
CN1246475A (zh) 2000-03-08
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PE32596A1 (es) 1996-08-07
NO965237L (no) 1997-02-06
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