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ES8306739A1 - "procedimiento para la fabricacion de derivados (tienil-2) t (tienil-3)-2 etilaminas". - Google Patents

"procedimiento para la fabricacion de derivados (tienil-2) t (tienil-3)-2 etilaminas".

Info

Publication number
ES8306739A1
ES8306739A1 ES514248A ES514248A ES8306739A1 ES 8306739 A1 ES8306739 A1 ES 8306739A1 ES 514248 A ES514248 A ES 514248A ES 514248 A ES514248 A ES 514248A ES 8306739 A1 ES8306739 A1 ES 8306739A1
Authority
ES
Spain
Prior art keywords
formula
thienyl
products
preparation
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES514248A
Other languages
English (en)
Other versions
ES514248A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9260130&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES8306739(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi SA filed Critical Sanofi SA
Publication of ES514248A0 publication Critical patent/ES514248A0/es
Publication of ES8306739A1 publication Critical patent/ES8306739A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms
    • C07F9/655345—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms the sulfur atom being part of a five-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/32—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/32—Esters thereof
    • C07F9/3205—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/3211—Esters of acyclic saturated acids which can have further substituents on alkyl
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biochemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Developing Agents For Electrophotography (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE (TIENIL-2)- Y (TIENIL-3)-2 ETILAMINAS, DE FORMULA (I), EN LA QUE R , R Y AR PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE CONDENSACION DE UN COMPUESTO DE FORMULA (II) CON UN COMPUESTO CARBONILADO DE FORMULA (III), EN LA QUE R , X E Y PUEDEN SER VARIOS TIPOS DE RADICALES; SEGUIDA DEL TRATAMIENTO CON UNA BASE DE FORMULA B>~P M>~O, A UNA TEMPERATURA ENTRE -78 C Y 150 C; HIDROLISIS Y TRATAMIENTO CON UNA BASE DE FORMULA B >~P M >~O; REACCION CON UN COMPUESTO CARBONILADO DE FORMULA ARCOR , EN LA QUE AR Y R SON LOS MISMOS QUE EN LA FORMULA (I); Y, FINALMENTE REDUCCION CON UN AGENTE REDUCTOR, TAL COMO BOROHIDRURO SODICO. ESTOS COMUESTOS TIENEN APLICACIONES COMO INTERMEDIOS EN PROCESOS DE SINTESIS.
ES514248A 1981-06-30 1982-06-11 "procedimiento para la fabricacion de derivados (tienil-2) t (tienil-3)-2 etilaminas". Expired ES8306739A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8113063A FR2508454A1 (fr) 1981-06-30 1981-06-30 Procede de preparation de derives des (thienyl-2)- et (thienyl-3)-2 ethylamines et produits ainsi obtenus

Publications (2)

Publication Number Publication Date
ES514248A0 ES514248A0 (es) 1983-06-01
ES8306739A1 true ES8306739A1 (es) 1983-06-01

Family

ID=9260130

Family Applications (1)

Application Number Title Priority Date Filing Date
ES514248A Expired ES8306739A1 (es) 1981-06-30 1982-06-11 "procedimiento para la fabricacion de derivados (tienil-2) t (tienil-3)-2 etilaminas".

Country Status (24)

Country Link
US (1) US4487931A (es)
EP (1) EP0068979B1 (es)
JP (1) JPS5810576A (es)
KR (1) KR840000537A (es)
AT (1) ATE15801T1 (es)
AU (1) AU567283B2 (es)
CA (1) CA1205809A (es)
CS (1) CS239926B2 (es)
DD (1) DD202710A5 (es)
DE (1) DE3266524D1 (es)
DK (1) DK152364C (es)
ES (1) ES8306739A1 (es)
FI (1) FI822316A7 (es)
FR (1) FR2508454A1 (es)
GR (1) GR78254B (es)
HU (1) HU194859B (es)
IE (1) IE53241B1 (es)
IL (1) IL65981A (es)
NO (1) NO155291C (es)
NZ (1) NZ200853A (es)
PT (1) PT75153B (es)
SU (1) SU1145930A3 (es)
YU (1) YU143282A (es)
ZA (1) ZA824615B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2622191B1 (fr) * 1987-10-22 1991-06-21 Sanofi Sa Procede de preparation de la n-(chloro-2 benzyl)-2 ethylamine et produits intermediaires dans cette preparation
US4900539A (en) * 1988-12-22 1990-02-13 The United States Of America As Represented By The United States Department Of Energy Radiohalogenated thienylethylamine derivatives for evaluating local cerebral blood flow
WO1992000964A1 (fr) * 1990-07-05 1992-01-23 Nippon Soda Co., Ltd. Derive d'amine
WO1993003025A1 (en) * 1991-08-09 1993-02-18 Yoshitomi Pharmaceutical Industries, Ltd. Thiophene compound

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4127580A (en) * 1975-02-07 1978-11-28 Parcor Process for the preparation of thieno-pyridine derivatives
FR2300090A1 (fr) * 1975-02-07 1976-09-03 Parcor Procede de preparation de derives de la thienopyridine
IT1082336B (it) * 1977-01-27 1985-05-21 Medea Res Srl Processo per la preparazione della 5.2.clorobenzil.4 5 6 7.tetraidro tien 3 2.c.piridina
FR2508453A1 (fr) * 1981-06-30 1982-12-31 Sanofi Sa Procede de preparation de derives des (thienyl-2)- et thienyl-3)-2 ethylamines et produits ainsi obtenus

Also Published As

Publication number Publication date
AU567283B2 (en) 1987-11-19
YU143282A (en) 1984-12-31
CA1205809A (en) 1986-06-10
FI822316A0 (fi) 1982-06-29
FI822316L (fi) 1982-12-31
ATE15801T1 (de) 1985-10-15
FR2508454B1 (es) 1983-12-23
DE3266524D1 (en) 1985-10-31
DD202710A5 (de) 1983-09-28
IE53241B1 (en) 1988-09-14
IL65981A0 (en) 1982-09-30
NO155291C (no) 1987-03-11
NO822225L (no) 1983-01-03
KR840000537A (ko) 1984-02-25
CS239926B2 (en) 1986-01-16
ES514248A0 (es) 1983-06-01
ZA824615B (en) 1983-04-27
AU8475382A (en) 1983-01-06
US4487931A (en) 1984-12-11
JPS5810576A (ja) 1983-01-21
IL65981A (en) 1986-04-29
DK152364B (da) 1988-02-22
IE821311L (en) 1982-12-30
SU1145930A3 (ru) 1985-03-15
GR78254B (es) 1984-09-26
FI822316A7 (fi) 1982-12-31
PT75153A (fr) 1982-07-01
DK284082A (da) 1982-12-31
DK152364C (da) 1988-08-15
HU194859B (en) 1988-03-28
FR2508454A1 (fr) 1982-12-31
EP0068979B1 (fr) 1985-09-25
NZ200853A (en) 1985-09-13
EP0068979A1 (fr) 1983-01-05
NO155291B (no) 1986-12-01
PT75153B (fr) 1984-05-29

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