ES503019A0 - A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS - Google Patents

A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS

Info

Publication number: ES503019A0
Authority: ES; Spain
Prior art keywords: phenylacete; benzoil; midas; approvals; cyclic
Prior art date: 1979-09-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

ES503019A

Other languages

Spanish (es)

Other versions

ES8204715A1 (en

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

AH Robins Co Inc

Original Assignee

AH Robins Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-09-26

Filing date

1981-06-12

Publication date

1982-05-01

1981-06-12 Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc

1982-05-01 Publication of ES8204715A1 publication Critical patent/ES8204715A1/en

1982-05-01 Publication of ES503019A0 publication Critical patent/ES503019A0/en

Status Granted legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Hematology (AREA)
Diabetes (AREA)
Rheumatology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

ES503019A 1979-09-26 1981-06-12 A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS Granted ES503019A0 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US7886079A	1979-09-26	1979-09-26

Publications (2)

Publication Number	Publication Date
ES8204715A1 ES8204715A1 (en)	1982-05-01
ES503019A0 true ES503019A0 (en)	1982-05-01

Family

ID=22146633

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
ES495329A Expired ES8200329A1 (en)	1979-09-26	1980-09-25	A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS
ES503019A Granted ES503019A0 (en)	1979-09-26	1981-06-12	A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
ES495329A Expired ES8200329A1 (en)	1979-09-26	1980-09-25	A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS

Country Status (36)

Country	Link
JP (1)	JPS5657751A (en)
KR (1)	KR840000763B1 (en)
AT (1)	AT374170B (en)
AU (1)	AU532359B2 (en)
BE (1)	BE885393A (en)
BR (1)	BR8006042A (en)
CA (1)	CA1128512A (en)
CH (1)	CH646138A5 (en)
CS (1)	CS227012B2 (en)
DE (1)	DE3035688A1 (en)
DK (1)	DK154136C (en)
EG (1)	EG15020A (en)
ES (2)	ES8200329A1 (en)
FI (1)	FI72967C (en)
FR (1)	FR2465710A1 (en)
GB (1)	GB2059963B (en)
GR (1)	GR70049B (en)
HK (1)	HK59383A (en)
HU (1)	HU183215B (en)
IE (1)	IE50268B1 (en)
IL (1)	IL60999A (en)
IN (3)	IN151313B (en)
IT (1)	IT1133823B (en)
KE (1)	KE3307A (en)
LU (1)	LU82797A1 (en)
MX (1)	MX7159E (en)
NL (1)	NL8005346A (en)
NO (1)	NO152128C (en)
NZ (1)	NZ195061A (en)
PH (1)	PH22628A (en)
PL (1)	PL128998B1 (en)
PT (1)	PT71839B (en)
SE (1)	SE448626B (en)
SG (1)	SG42983G (en)
YU (3)	YU41734B (en)
ZA (1)	ZA805476B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL61945A (en) *	1980-02-19	1984-09-30	Robins Co Inc A H	2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them
US6066671A (en)	1997-12-19	2000-05-23	Alcon Laboratories, Inc.	Treatment of GLC1A glaucoma with 3-benzoyl-phenylacetic acids, esters, or amides
US6646001B2 (en)	1997-12-19	2003-11-11	Alcon Manufacturing, Ltd.	Use of non-steroidal anti-inflammatory agents in combination with prostaglandin FP receptor agonists to treat glaucoma and ocular hypertension
GB9727523D0 (en) *	1997-12-31	1998-02-25	Pharmacia & Upjohn Spa	Alpha-aminoamide derivatives useful as analgesic agents
AR030345A1 (en) *	2000-08-14	2003-08-20	Alcon Inc	METHOD OF TREATMENT OF DISORDERS RELATED TO ANGIOGENESIS
ATE317280T1 (en)	2001-09-03	2006-02-15	Newron Pharm Spa	PHARMACEUTICAL COMPOSITION CONTAINING GABAPENTIN OR ITS ANALOGUE AND AN ALPHA-AMINOAMIDE AND ANALGESIC USE OF THIS COMPOSITION
EP1438956A1 (en)	2003-01-16	2004-07-21	Newron Pharmaceuticals S.p.A.	Alpha-aminoamide derivatives useful as antimigraine agents
CZ301776B6 (en) *	2009-06-08	2010-06-16	Farmak, A.S.	Process for preparing 2-amino-3-benzoylphenylacetamide (nepafenac) with minimum by-products
CN112794809B (en) *	2019-11-14	2023-12-29	南京济群医药科技股份有限公司	Preparation method of high-purity nepafenac intermediate

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1226344A (en) *	1967-07-31	1971-03-24
SE400966B (en) *	1975-08-13	1978-04-17	Robins Co Inc A H	PROCEDURE FOR PREPARING 2-AMINO-3- (OR 5-) BENZOYL-PHENYLETIC ACIDS
IL61945A (en) *	1980-02-19	1984-09-30	Robins Co Inc A H	2-amino-3-(hydroxy(phenyl)methyl)phenylacetic acids,esters and amides and pharmaceutical compositions containing them

1980
- 1980-09-04 ZA ZA00805476A patent/ZA805476B/en unknown
- 1980-09-08 IL IL60999A patent/IL60999A/en unknown
- 1980-09-08 AU AU62116/80A patent/AU532359B2/en not_active Ceased
- 1980-09-11 CS CS806196A patent/CS227012B2/en unknown
- 1980-09-17 IE IE1946/80A patent/IE50268B1/en unknown
- 1980-09-20 EG EG80573A patent/EG15020A/en active
- 1980-09-22 BR BR8006042A patent/BR8006042A/en unknown
- 1980-09-22 DE DE19803035688 patent/DE3035688A1/en active Granted
- 1980-09-22 GR GR62936A patent/GR70049B/el unknown
- 1980-09-23 PH PH24613A patent/PH22628A/en unknown
- 1980-09-23 AT AT0474580A patent/AT374170B/en not_active IP Right Cessation
- 1980-09-24 LU LU82797A patent/LU82797A1/en unknown
- 1980-09-24 FI FI803002A patent/FI72967C/en not_active IP Right Cessation
- 1980-09-24 SE SE8006668A patent/SE448626B/en not_active IP Right Cessation
- 1980-09-25 CH CH719180A patent/CH646138A5/en not_active IP Right Cessation
- 1980-09-25 BE BE0/202226A patent/BE885393A/en not_active IP Right Cessation
- 1980-09-25 NL NL8005346A patent/NL8005346A/en not_active Application Discontinuation
- 1980-09-25 YU YU2450/80A patent/YU41734B/en unknown
- 1980-09-25 FR FR8020596A patent/FR2465710A1/en active Granted
- 1980-09-25 CA CA361,068A patent/CA1128512A/en not_active Expired
- 1980-09-25 MX MX809050U patent/MX7159E/en unknown
- 1980-09-25 DK DK405780A patent/DK154136C/en not_active IP Right Cessation
- 1980-09-25 HU HU802347A patent/HU183215B/en not_active IP Right Cessation
- 1980-09-25 PL PL1980226919A patent/PL128998B1/en unknown
- 1980-09-25 KR KR1019800003740A patent/KR840000763B1/en not_active Expired
- 1980-09-25 GB GB8030955A patent/GB2059963B/en not_active Expired
- 1980-09-25 NO NO802834A patent/NO152128C/en unknown
- 1980-09-25 ES ES495329A patent/ES8200329A1/en not_active Expired
- 1980-09-25 PT PT71839A patent/PT71839B/en unknown
- 1980-09-26 NZ NZ195061A patent/NZ195061A/en unknown
- 1980-09-26 IT IT24948/80A patent/IT1133823B/en active
- 1980-09-26 JP JP13415280A patent/JPS5657751A/en active Granted
- 1980-09-26 IN IN1092/CAL/80A patent/IN151313B/en unknown
1981
- 1981-06-12 ES ES503019A patent/ES503019A0/en active Granted
1982
- 1982-12-30 IN IN1508/CAL/82A patent/IN156254B/en unknown
- 1982-12-30 IN IN1509/CAL/82A patent/IN156255B/en unknown
1983
- 1983-03-28 YU YU730/83A patent/YU43305B/en unknown
- 1983-03-28 YU YU731/83A patent/YU43306B/en unknown
- 1983-07-19 SG SG42983A patent/SG42983G/en unknown
- 1983-07-21 KE KE3307A patent/KE3307A/en unknown
- 1983-11-24 HK HK593/83A patent/HK59383A/en unknown

Also Published As

Publication number	Publication date
KR840000763B1 (en)	1984-06-08
IL60999A (en)	1984-05-31
GB2059963B (en)	1983-04-20
PL226919A1 (en)	1982-02-01
FI803002A7 (en)	1981-03-27
JPH0141616B2 (en)	1989-09-06
DK154136B (en)	1988-10-17
HU183215B (en)	1984-04-28
YU43305B (en)	1989-06-30
PT71839B (en)	1981-06-25
PH22628A (en)	1988-10-28
IT8024948A0 (en)	1980-09-26
IN156255B (en)	1985-06-08
YU245080A (en)	1983-09-30
PT71839A (en)	1980-10-01
SG42983G (en)	1985-01-11
CA1128512A (en)	1982-07-27
BE885393A (en)	1981-01-16
DE3035688C2 (en)	1990-05-17
FR2465710B1 (en)	1984-10-12
PL128998B1 (en)	1984-03-31
LU82797A1 (en)	1982-05-10
FR2465710A1 (en)	1981-03-27
IE50268B1 (en)	1986-03-19
NO152128C (en)	1985-08-07
MX7159E (en)	1987-12-02
JPS5657751A (en)	1981-05-20
DE3035688A1 (en)	1981-04-16
CS227012B2 (en)	1984-04-16
YU73083A (en)	1983-12-31
NO802834L (en)	1981-03-27
KR830004210A (en)	1983-07-06
DK405780A (en)	1981-03-27
AU532359B2 (en)	1983-09-29
BR8006042A (en)	1981-04-07
ES495329A0 (en)	1981-10-16
NL8005346A (en)	1981-03-30
SE8006668L (en)	1981-03-27
CH646138A5 (en)	1984-11-15
ES8200329A1 (en)	1981-10-16
ES8204715A1 (en)	1982-05-01
YU41734B (en)	1987-12-31
FI72967C (en)	1987-08-10
KE3307A (en)	1983-08-19
YU73183A (en)	1983-12-31
GB2059963A (en)	1981-04-29
AU6211680A (en)	1981-04-02
DK154136C (en)	1989-03-06
NZ195061A (en)	1984-04-27
YU43306B (en)	1989-06-30
AT374170B (en)	1984-03-26
IT1133823B (en)	1986-07-24
ATA474580A (en)	1983-08-15
IL60999A0 (en)	1980-11-30
ZA805476B (en)	1981-11-25
IN156254B (en)	1985-06-08
NO152128B (en)	1985-04-29
HK59383A (en)	1983-12-02
SE448626B (en)	1987-03-09
IE801946L (en)	1981-03-26
IN151313B (en)	1983-03-26
GR70049B (en)	1982-07-26
EG15020A (en)	1985-03-31
FI72967B (en)	1987-04-30

Publication	Publication Date	Title
ES495813A0 (en)	1981-11-16	A PROCEDURE FOR PREPARING A MODIFIED ELASTOMER
AR225301A1 (en)	1982-03-15	PROCEDURE FOR PREPARING NORTROPIL-ALKYL BENZAMIDES
ES493061A0 (en)	1981-06-16	A PROCEDURE FOR PREPARING A LIPOPOLISACARIDE
ES487180A0 (en)	1980-12-16	A PROCEDURE FOR PREPARING MERCAPTOACIL-PROLINAS CETALIC AND THIOCEALIC DERIVATIVES
ES490166A0 (en)	1981-04-01	A PROCEDURE FOR PREPARING MERCAPTOACILDIPEPTIDOS
ES523194A0 (en)	1985-04-16	A PROCEDURE FOR PREPARING N-FORMIL AND N-HYDROXYMETHYL-3-PHENOXI-1-AZETIDINCARBOXAMIDES
ES487847A0 (en)	1980-12-16	A PROCEDURE FOR PREPARING NEW PHENETHANOLAMINS
ES497301A0 (en)	1982-01-01	A PROCEDURE FOR PREPARING 9-AMINOALKYLFLUORENES
MX5431E (en)	1983-08-05	IMPROVED PROCEDURE FOR PREPARING COCO-POLYMERS CONTAINING TRIORGANOESTANE
ES495329A0 (en)	1981-10-16	A PROCEDURE FOR PREPARING 2-AMINO-3-BENZOIL-PHENYLACETE-MIDAS AND CYCLIC APPROVALS
ES493759A0 (en)	1981-08-01	A PROCEDURE FOR PREPARING BENZOXAZEPINES
ES494459A0 (en)	1981-08-16	A PROCEDURE FOR PREPARING CETOXIMINOETERES
AR224149A1 (en)	1981-10-30	A PROCEDURE FOR PRODUCING PIRAN-4-ONAS
IT8048889A0 (en)	1980-06-05	PERFLUOROALKY COMPOUNDS AND PROCEDURE FOR PREPARING THEM
ES487682A0 (en)	1980-12-16	A PROCEDURE FOR PREPARING VINDESINE
ES487349A0 (en)	1981-05-16	A PROCEDURE FOR PREPARING A CHROMOGEN MATERIAL
BR7904285A (en)	1981-01-05	FIT FOR A GAUGE AND GAUGE
MX6013E (en)	1984-09-24	PROCEDURE FOR PREPARING ARILALQUIL AND ARILOXI-ALQUIL-FOSFONATOS
IT7948141A0 (en)	1979-02-27	PROCEDURE FOR PACKING AND PACKING A PARACHUTE
ES498871A0 (en)	1982-06-01	PROCEDURE FOR PREPARING A 2-METHYL-8 (R) OR (S) ERGOTPEPTIDE ALCALOID
ES494705A0 (en)	1981-07-16	A PROCEDURE FOR HYDROLYZING ALIL - ETERES
ES486713A0 (en)	1980-12-16	A PROCEDURE FOR PREPARING FUROPYRIDINONES AND FUROPYRAZI-NONAS
ES493191A0 (en)	1981-06-16	A METHOD FOR PREPARING PHENYLIMINOTIADIAZOLINS
MX5707E (en)	1983-12-16	PROCEDURE FOR PREPARING DIURETHANE
ES481212A0 (en)	1980-12-16	A PROCEDURE FOR PREPARING BENZOXEPINES

Legal Events

Date	Code	Title	Description
1996-06-16	MM4A	Patent lapsed	Effective date: 19960506