ES505556A0 - Un procedimiento para la preparacion de derivados de imida- zol - Google Patents
Un procedimiento para la preparacion de derivados de imida- zolInfo
- Publication number
- ES505556A0 ES505556A0 ES505556A ES505556A ES505556A0 ES 505556 A0 ES505556 A0 ES 505556A0 ES 505556 A ES505556 A ES 505556A ES 505556 A ES505556 A ES 505556A ES 505556 A0 ES505556 A0 ES 505556A0
- Authority
- ES
- Spain
- Prior art keywords
- imida
- zol
- derivatives
- procedure
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7934347 | 1979-10-03 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES505556A0 true ES505556A0 (es) | 1982-12-01 |
| ES8301221A1 ES8301221A1 (es) | 1982-12-01 |
Family
ID=10508267
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES495589A Granted ES495589A0 (es) | 1979-10-03 | 1980-10-02 | Un procedimiento para la preparacion de derivados de imida- lol. |
| ES505555A Granted ES505555A0 (es) | 1979-10-03 | 1981-09-16 | Un procedimiento para la preparacion de derivados de imida- zol |
| ES505556A Expired ES8301221A1 (es) | 1979-10-03 | 1981-09-16 | Un procedimiento para la preparacion de derivados de imida- zol |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES495589A Granted ES495589A0 (es) | 1979-10-03 | 1980-10-02 | Un procedimiento para la preparacion de derivados de imida- lol. |
| ES505555A Granted ES505555A0 (es) | 1979-10-03 | 1981-09-16 | Un procedimiento para la preparacion de derivados de imida- zol |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4324792A (es) |
| JP (1) | JPS5690063A (es) |
| AU (1) | AU6294580A (es) |
| BE (1) | BE885507A (es) |
| DE (1) | DE3037313A1 (es) |
| DK (1) | DK420480A (es) |
| ES (3) | ES495589A0 (es) |
| FI (1) | FI803127L (es) |
| FR (1) | FR2466461A1 (es) |
| GB (1) | GB2062626B (es) |
| IT (1) | IT1144007B (es) |
| NL (1) | NL8005491A (es) |
| NZ (1) | NZ195144A (es) |
| SE (1) | SE8006953L (es) |
| ZA (1) | ZA806146B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT78388B (en) * | 1983-04-12 | 1986-09-15 | Smithkline Beckman Corp | Dopamine-beta-hydroxylase inhibitors |
| US4532331A (en) * | 1983-04-12 | 1985-07-30 | Smithkline Beckman Corporation | 1-Benzyl-2-aminomethyl imidazole derivatives |
| US4602093A (en) * | 1984-02-08 | 1986-07-22 | Merck & Co., Inc. | Novel substituted imidazoles, their preparation and use |
| US4661602A (en) * | 1985-03-29 | 1987-04-28 | G. D. Searle & Co. | Substituted alkyl imidazole derivatives |
| NZ238688A (en) * | 1990-06-28 | 1992-05-26 | Smithkline Beecham Corp | Substituted histidines: pharmaceutical compositions, preparation and uses thereof |
| US5807872A (en) * | 1992-12-16 | 1998-09-15 | Schering Corporation | Imidazoylalkyl substituted with a six membered nitrogen containing heterocyclic ring |
| US5972984A (en) * | 1995-06-06 | 1999-10-26 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| ES2163295T3 (es) | 1997-10-22 | 2002-01-16 | Astrazeneca Ab | Derivados de imidazol y su uso como inhibidores de la farnesil-protein-transferasa. |
| WO1999020612A1 (en) * | 1997-10-22 | 1999-04-29 | Astrazeneca Uk Limited | Imidazole derivatives and their use as farnesyl protein transferase inhibitors |
| EP2447263A1 (en) * | 2010-09-27 | 2012-05-02 | Bioprojet | Benzazole derivatives as histamine H4 receptor ligands |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2532547A (en) * | 1950-12-05 | Z-aminoalkyl-glyoxaline derivatives | ||
| GB1421792A (en) * | 1973-05-17 | 1976-01-21 | Smith Kline French Lab | Heterocyclic substituted-1, 1-diamino-ethylene derivatives methods for their preparation and compositions containing them |
| US4152443A (en) * | 1973-07-13 | 1979-05-01 | Smith Kline & French Laboratories Limited | Imidazolyl thioureas, ureas and guanidines |
| US4006137A (en) * | 1975-08-21 | 1977-02-01 | E. R. Squibb & Sons, Inc. | 2-Ethenyl imidazolium derivatives |
-
1980
- 1980-10-01 FI FI803127A patent/FI803127L/fi not_active Application Discontinuation
- 1980-10-02 BE BE0/202313A patent/BE885507A/fr unknown
- 1980-10-02 DE DE19803037313 patent/DE3037313A1/de not_active Withdrawn
- 1980-10-02 ES ES495589A patent/ES495589A0/es active Granted
- 1980-10-03 FR FR8021246A patent/FR2466461A1/fr active Granted
- 1980-10-03 DK DK420480A patent/DK420480A/da not_active Application Discontinuation
- 1980-10-03 JP JP13861880A patent/JPS5690063A/ja active Pending
- 1980-10-03 GB GB8032001A patent/GB2062626B/en not_active Expired
- 1980-10-03 NL NL8005491A patent/NL8005491A/nl not_active Application Discontinuation
- 1980-10-03 US US06/193,846 patent/US4324792A/en not_active Expired - Lifetime
- 1980-10-03 IT IT49815/80A patent/IT1144007B/it active
- 1980-10-03 ZA ZA00806146A patent/ZA806146B/xx unknown
- 1980-10-03 AU AU62945/80A patent/AU6294580A/en not_active Abandoned
- 1980-10-03 NZ NZ195144A patent/NZ195144A/xx unknown
- 1980-10-03 SE SE8006953A patent/SE8006953L/xx not_active Application Discontinuation
-
1981
- 1981-09-16 ES ES505555A patent/ES505555A0/es active Granted
- 1981-09-16 ES ES505556A patent/ES8301221A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| IT8049815A0 (it) | 1980-10-03 |
| SE8006953L (sv) | 1981-04-04 |
| FR2466461A1 (fr) | 1981-04-10 |
| JPS5690063A (en) | 1981-07-21 |
| FR2466461B1 (es) | 1983-05-20 |
| BE885507A (fr) | 1981-04-02 |
| DK420480A (da) | 1981-04-04 |
| ES8203855A1 (es) | 1981-12-16 |
| NZ195144A (en) | 1983-02-15 |
| GB2062626B (en) | 1983-10-05 |
| US4324792A (en) | 1982-04-13 |
| ES8205204A1 (es) | 1982-06-01 |
| ZA806146B (en) | 1982-01-27 |
| GB2062626A (en) | 1981-05-28 |
| NL8005491A (nl) | 1981-04-07 |
| ES8301221A1 (es) | 1982-12-01 |
| ES505555A0 (es) | 1982-06-01 |
| DE3037313A1 (de) | 1981-04-23 |
| FI803127A7 (fi) | 1981-04-04 |
| AU6294580A (en) | 1981-04-16 |
| IT1144007B (it) | 1986-10-29 |
| FI803127L (fi) | 1981-04-04 |
| ES495589A0 (es) | 1981-12-16 |
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