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ES480121A0 - Un procedimiento para la preparacion de nuevos derivados de quinazolina. - Google Patents

Un procedimiento para la preparacion de nuevos derivados de quinazolina.

Info

Publication number
ES480121A0
ES480121A0 ES480121A ES480121A ES480121A0 ES 480121 A0 ES480121 A0 ES 480121A0 ES 480121 A ES480121 A ES 480121A ES 480121 A ES480121 A ES 480121A ES 480121 A0 ES480121 A0 ES 480121A0
Authority
ES
Spain
Prior art keywords
procedure
preparation
quinazoline derivatives
new quinazoline
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES480121A
Other languages
English (en)
Other versions
ES8308559A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Original Assignee
Pfizer Corp Belgium
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium filed Critical Pfizer Corp Belgium
Publication of ES480121A0 publication Critical patent/ES480121A0/es
Publication of ES8308559A1 publication Critical patent/ES8308559A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/201,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
ES480121A 1977-11-05 1979-04-30 Un procedimiento para la preparacion de nuevos derivados de quinazolina. Expired ES8308559A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4612877 1977-11-05

Publications (2)

Publication Number Publication Date
ES480121A0 true ES480121A0 (es) 1980-07-16
ES8308559A1 ES8308559A1 (es) 1980-07-16

Family

ID=10439957

Family Applications (2)

Application Number Title Priority Date Filing Date
ES474805A Expired ES474805A1 (es) 1977-11-05 1978-11-03 Un procedimiento para la preparacion de nuevos derivados de quinazolina
ES480121A Expired ES8308559A1 (es) 1977-11-05 1979-04-30 Un procedimiento para la preparacion de nuevos derivados de quinazolina.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES474805A Expired ES474805A1 (es) 1977-11-05 1978-11-03 Un procedimiento para la preparacion de nuevos derivados de quinazolina

Country Status (36)

Country Link
JP (1) JPS5498792A (es)
AR (2) AR219562A1 (es)
AT (1) AT365186B (es)
AU (1) AU509329B2 (es)
BE (1) BE871771A (es)
CA (1) CA1088059A (es)
CH (1) CH643255A5 (es)
CS (2) CS207671B2 (es)
DD (1) DD139850A5 (es)
DE (1) DE2847623C2 (es)
DK (1) DK154082C (es)
EG (1) EG13594A (es)
ES (2) ES474805A1 (es)
FI (1) FI64366C (es)
FR (1) FR2407929A1 (es)
GR (1) GR81514B (es)
HK (1) HK94284A (es)
HU (1) HU176306B (es)
IE (1) IE47888B1 (es)
IL (1) IL55857A (es)
IN (1) IN148828B (es)
IT (1) IT1100919B (es)
KE (1) KE3350A (es)
LU (2) LU80470A1 (es)
MY (1) MY8500286A (es)
NL (2) NL174549C (es)
NO (1) NO150158C (es)
NZ (1) NZ188813A (es)
PH (1) PH13966A (es)
PL (2) PL119586B1 (es)
PT (1) PT68735A (es)
SE (1) SE437518B (es)
SU (1) SU816403A3 (es)
UA (1) UA8324A1 (es)
YU (2) YU40204B (es)
ZA (1) ZA786184B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985002617A1 (fr) * 1983-12-14 1985-06-20 Takeda Chemical Industries. Ltd. Derives de 1,5-benzoxathiepine et leur procede de preparation
WO1986002644A1 (fr) * 1984-11-01 1986-05-09 Takeda Chemical Industries, Ltd. Derives de 1,5-benzoxathiepines et leur procede de preparation
WO1985004658A1 (fr) * 1984-04-04 1985-10-24 Takeda Chemical Industries, Ltd. Derives de 1,5 benzoxathiepine et leur preparation
EP0849265A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von Doxazosin-Mesylat (Form II)
EP0849264A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von doxazosinmesylat (Form I)
PT849266E (pt) * 1996-12-20 2007-03-30 Heumann Pcs Gmbh Nova forma polimorfa de mesilato de doxazosina (forma iii)
TW448155B (en) * 1999-03-29 2001-08-01 Dev Center Biotechnology Method for producing amide compounds and quinazolin derivatives
EP1403263B1 (en) * 2002-09-27 2005-06-22 Council of Scientific and Industrial Research Process for the preparation of N-(2,3-dihydrobenzo 1,4 dioxin-2-carbonyl) piperazine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3663706A (en) * 1969-09-29 1972-05-16 Pfizer Use of 2,4-diaminoquinazolines as hypotensive agents
US3669968A (en) * 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines

Also Published As

Publication number Publication date
NL930062I1 (nl) 1993-09-01
FI64366C (fi) 1983-11-10
DK154082C (da) 1989-02-27
YU40419B (en) 1985-12-31
AR223015A1 (es) 1981-07-15
FR2407929B1 (es) 1981-02-27
IT1100919B (it) 1985-09-28
MY8500286A (en) 1985-12-31
FR2407929A1 (fr) 1979-06-01
IE782179L (en) 1979-05-05
DE2847623C2 (de) 1983-06-01
NL174549C (nl) 1984-07-02
NO150158B (no) 1984-05-21
AU509329B2 (en) 1980-05-08
PL119419B1 (en) 1981-12-31
PT68735A (en) 1978-12-01
ES8308559A1 (es) 1980-07-16
KE3350A (en) 1983-12-16
YU255378A (en) 1983-06-30
DD139850A5 (de) 1980-01-23
CA1088059A (en) 1980-10-21
SU816403A3 (ru) 1981-03-23
NZ188813A (en) 1980-10-08
NL930062I2 (nl) 1993-11-16
IL55857A (en) 1982-07-30
ZA786184B (en) 1979-10-31
LU80470A1 (fr) 1980-06-05
SE7811382L (sv) 1979-05-06
NO150158C (no) 1984-08-29
PH13966A (en) 1980-11-12
SE437518B (sv) 1985-03-04
HU176306B (en) 1981-01-28
NO783705L (no) 1979-05-08
DK154082B (da) 1988-10-10
AR219562A1 (es) 1980-08-29
NL7810909A (nl) 1979-05-08
YU38683A (en) 1983-06-30
HK94284A (en) 1984-12-07
IE47888B1 (en) 1984-07-11
PL119586B1 (en) 1982-01-30
GR81514B (es) 1984-12-11
PL210681A1 (es) 1979-11-05
ATA784378A (de) 1981-05-15
FI783347A7 (fi) 1979-05-06
IT7829434A0 (it) 1978-11-03
UA8324A1 (uk) 1996-03-29
JPS5498792A (en) 1979-08-03
FI64366B (fi) 1983-07-29
JPS5625233B2 (es) 1981-06-11
DE2847623A1 (de) 1979-05-23
NL174549B (nl) 1984-02-01
CH643255A5 (en) 1984-05-30
ES474805A1 (es) 1980-01-16
BE871771A (fr) 1979-05-03
IL55857A0 (en) 1979-01-31
LU88331I2 (fr) 1994-05-04
CS354491A3 (en) 1992-06-17
YU40204B (en) 1985-08-31
DK428678A (da) 1979-05-06
CS207671B2 (en) 1981-08-31
AU4132278A (en) 1979-05-17
EG13594A (en) 1982-03-31
AT365186B (de) 1981-12-28
IN148828B (es) 1981-06-27

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