ES485652A2 - Procedimiento para la obtencion de derivados de la hidroxi-4tiazolidinationa-2 - Google Patents
Procedimiento para la obtencion de derivados de la hidroxi-4tiazolidinationa-2Info
- Publication number
- ES485652A2 ES485652A2 ES485652A ES485652A ES485652A2 ES 485652 A2 ES485652 A2 ES 485652A2 ES 485652 A ES485652 A ES 485652A ES 485652 A ES485652 A ES 485652A ES 485652 A2 ES485652 A2 ES 485652A2
- Authority
- ES
- Spain
- Prior art keywords
- radical
- radicals
- substituted
- atom
- atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 4-substituted-4-hydroxy-3-pyridyl-thiazolidine-2-thione Chemical class 0.000 title abstract 7
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 4
- 239000005864 Sulphur Chemical group 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 125000005842 heteroatom Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 229910052757 nitrogen Inorganic materials 0.000 abstract 2
- 229910052760 oxygen Chemical group 0.000 abstract 2
- 239000001301 oxygen Chemical group 0.000 abstract 2
- 229920006395 saturated elastomer Polymers 0.000 abstract 2
- 125000001541 3-thienyl group Chemical group S1C([H])=C([*])C([H])=C1[H] 0.000 abstract 1
- 241000244206 Nematoda Species 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 1
- 125000005115 alkyl carbamoyl group Chemical group 0.000 abstract 1
- MDFFNEOEWAXZRQ-UHFFFAOYSA-N aminyl Chemical compound [NH2] MDFFNEOEWAXZRQ-UHFFFAOYSA-N 0.000 abstract 1
- 230000000507 anthelmentic effect Effects 0.000 abstract 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- JEVCWSUVFOYBFI-UHFFFAOYSA-N cyanyl Chemical compound N#[C] JEVCWSUVFOYBFI-UHFFFAOYSA-N 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- LEVJVKGPFAQPOI-UHFFFAOYSA-N phenylmethanone Chemical compound O=[C]C1=CC=CC=C1 LEVJVKGPFAQPOI-UHFFFAOYSA-N 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/46—Oxygen atoms
- C07D213/50—Ketonic radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Mejoras introducidas en el objeto de la patente principal nº 469.883, concedida el 13 de Junio de 1979, por PROCEDIMIENTO PARA LA OBTENCIÓN DE DERIVADOS DE LA HIDROXI-4 TIAZOLIDINATIONA-2, de fórmula general: **(Formula)** en la que: R1 representa un átomo de hidrógeno o de halógeno situado en posición -4, -5 ó -6, y R2 representa un radical alquilo que contenga de 2 a 4 átomos de carbono sustituido en posición diferente de la -1 (por un radical amino, alquilamino, dialquilamino, carbamoilo, alquilcarbamoilo, dialquilcarcarbamoilo ó ciano) o un radical dialquiloximetilo, fenil-1 ciclopropilo, metil-1 ciclohexilo, fenilo sustituido (por un radical amino en posición -2 o por dos radicales idénticos elegidos de entre hidroxi, metilo o metoxi), naftilo-1, heterocíclico (elegido de entre ditiolano-1,3 il-2, dihidro-5,6 ditiino-1,4 il-2, tienilo-3 ó piridilo-2, -3 ó - 4)alcanoilo o benzoilo; entendiéndose que las porciones alquilo y el radical alcanoilo citados anteriormente son rectos o ramificados y que, salvo mención especial, contienen de 1 a 4 átomos de carbono, y eventualmente sus sales cuando R2 representa un radical alquilo sustituido (por un radical amino, alquilamino, dialquilamino o dialquilcarbamoilo cuyas partes alquilo forman con el átomo de nitrógeno al cual están enlazadas, un heterociclo saturado con 5 ó 6 eslabones que contiene otro átomo de nitrógeno, secundario o terciario) o amino-2 fenilo.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7831039A FR2440368A2 (fr) | 1978-11-02 | 1978-11-02 | Nouveaux derives de la thiazolidine, leur preparation et les compositions qui les contiennent |
| FR7922793A FR2464954A2 (fr) | 1979-09-12 | 1979-09-12 | Nouveaux derives de la thiazolidine, leur preparation et les compositions qui les contiennent |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES485652A2 true ES485652A2 (es) | 1980-06-16 |
Family
ID=26220831
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES485652A Expired ES485652A2 (es) | 1978-11-02 | 1979-11-02 | Procedimiento para la obtencion de derivados de la hidroxi-4tiazolidinationa-2 |
Country Status (10)
| Country | Link |
|---|---|
| AT (1) | ATA706679A (es) |
| AU (1) | AU5237779A (es) |
| DE (1) | DE2944342A1 (es) |
| ES (1) | ES485652A2 (es) |
| GB (1) | GB2034712A (es) |
| IL (1) | IL58610A0 (es) |
| IT (1) | IT1125602B (es) |
| LU (1) | LU81843A1 (es) |
| NL (1) | NL7907862A (es) |
| SE (1) | SE7909082L (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE152102T1 (de) * | 1991-05-10 | 1997-05-15 | Takeda Chemical Industries Ltd | Pyridinderivate, deren herstellung und anwendung |
-
1979
- 1979-10-25 NL NL7907862A patent/NL7907862A/nl not_active Application Discontinuation
- 1979-10-31 GB GB7937711A patent/GB2034712A/en not_active Withdrawn
- 1979-10-31 AU AU52377/79A patent/AU5237779A/en not_active Abandoned
- 1979-10-31 LU LU81843A patent/LU81843A1/fr unknown
- 1979-11-01 SE SE7909082A patent/SE7909082L/xx unknown
- 1979-11-01 IL IL58610A patent/IL58610A0/xx unknown
- 1979-11-02 ES ES485652A patent/ES485652A2/es not_active Expired
- 1979-11-02 IT IT27015/79A patent/IT1125602B/it active
- 1979-11-02 DE DE19792944342 patent/DE2944342A1/de not_active Ceased
- 1979-11-02 AT AT706679A patent/ATA706679A/de unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ATA706679A (de) | 1981-04-15 |
| DE2944342A1 (de) | 1980-05-08 |
| IL58610A0 (en) | 1980-02-29 |
| LU81843A1 (fr) | 1980-05-07 |
| IT1125602B (it) | 1986-05-14 |
| NL7907862A (nl) | 1980-05-07 |
| SE7909082L (sv) | 1980-05-03 |
| IT7927015A0 (it) | 1979-11-02 |
| AU5237779A (en) | 1980-05-08 |
| GB2034712A (en) | 1980-06-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD2A | Announcement of lapse in spain |
Effective date: 20170707 |