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ES2011727A6 - Aqueous formulations of piperidinylcyclopentylheptenoic acid derivatives - Google Patents

Aqueous formulations of piperidinylcyclopentylheptenoic acid derivatives

Info

Publication number
ES2011727A6
ES2011727A6 ES8803876A ES8803876A ES2011727A6 ES 2011727 A6 ES2011727 A6 ES 2011727A6 ES 8803876 A ES8803876 A ES 8803876A ES 8803876 A ES8803876 A ES 8803876A ES 2011727 A6 ES2011727 A6 ES 2011727A6
Authority
ES
Spain
Prior art keywords
aqueous formulations
acid derivatives
substituted
acid
formulation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
ES8803876A
Other languages
Spanish (es)
Inventor
Harry Finch
Anthony John Phillips
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB878729823A external-priority patent/GB8729823D0/en
Priority claimed from GB888804422A external-priority patent/GB8804422D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of ES2011727A6 publication Critical patent/ES2011727A6/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6564Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
    • C07F9/6581Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms
    • C07F9/6584Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms having one phosphorus atom as ring hetero atom
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08BPOLYSACCHARIDES; DERIVATIVES THEREOF
    • C08B37/00Preparation of polysaccharides not provided for in groups C08B1/00 - C08B35/00; Derivatives thereof
    • C08B37/0006Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid
    • C08B37/0009Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid alpha-D-Glucans, e.g. polydextrose, alternan, glycogen; (alpha-1,4)(alpha-1,6)-D-Glucans; (alpha-1,3)(alpha-1,4)-D-Glucans, e.g. isolichenan or nigeran; (alpha-1,4)-D-Glucans; (alpha-1,3)-D-Glucans, e.g. pseudonigeran; Derivatives thereof
    • C08B37/0012Cyclodextrin [CD], e.g. cycle with 6 units (alpha), with 7 units (beta) and with 8 units (gamma), large-ring cyclodextrin or cycloamylose with 9 units or more; Derivatives thereof
    • C08B37/0015Inclusion compounds, i.e. host-guest compounds, e.g. polyrotaxanes

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nanotechnology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medical Informatics (AREA)
  • Materials Engineering (AREA)
  • Polymers & Plastics (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • General Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Pulmonology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA PREPARAR FORMULACIONES ACUOSAS QUECONTIENEN UN DERIVADO DE ACIDO PIPERIDINILCICLOPENTILHEPTENOICO. CONSISTE EN MEZCLAR EN AGUA ACIDO **FORMULA** (B)-7- 5-(1,1K-BIFENIL)-4-IL METOXI -3-HIDROXI-2-(1-PIPERIDINIL) CICLOPENTIL -4-HEPTENOICO, O SU SAL HIDROCLORURO, COMO INGREDIENTE ACTIVO, CON UNA CICLODEXTRINA SUSTITUIDA O NO SUSTITUIDA, O UN HIDRATO DE LA MISMA, TRAS LO CUAL SE AÑADEN LOS RESTANTES CONSTITUYENTES QUE EVENTUALMENTE FORMEN PARTE DE LA FORMULACION FINAL, QUE PUEDE PRESENTARSE EN FORMA DE JARABES, CAPSULAS Y PREPARADOS PARA INYECCION E INHALACION. EL PRODUCTO OBTENIDO ES UTIL PARA TRATAR O PREVENIR ENFERMEDADES CARDIOVASCULARES MEDIADAS POR TROMBOXANOPROCEDURE FOR PREPARING AQUEOUS FORMULATIONS CONTAINING A DERIVATIVE OF PIPERIDINYL CYCLOPENTILHEPTENOIC ACID. CONSISTS OF MIXING IN WATER ACID ** FORMULA ** (B) -7- 5- (1,1K-BIPHENYL) -4-IL METOXY -3-HYDROXY-2- (1-PIPERIDINIL) CYCLOPENTIL -4-HEPTENOICO, OR ITS HYDROCHLORIDE SALT, AS AN ACTIVE INGREDIENT, WITH A SUBSTITUTED OR NON-SUBSTITUTED CYCLODEXTRINE, OR A HYDRATE OF THE SAME, AFTER WHICH THE REMAINING CONSTITUENTS ARE ADDED THAT EVENTUALLY FORM PART OF THE FORMULATION AND FINAL FORMULATION, WHICH MAY BE PRESENTED PREPARED FOR INJECTION AND INHALATION. THE PRODUCT OBTAINED IS USEFUL TO TREAT OR PREVENT CARDIOVASCULAR DISEASES MEDIATED BY THROMBOXANE

ES8803876A 1987-12-22 1988-12-21 Aqueous formulations of piperidinylcyclopentylheptenoic acid derivatives Expired - Fee Related ES2011727A6 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB878729823A GB8729823D0 (en) 1987-12-22 1987-12-22 Complexes
GB888804422A GB8804422D0 (en) 1988-02-25 1988-02-25 Complexes

Publications (1)

Publication Number Publication Date
ES2011727A6 true ES2011727A6 (en) 1990-02-01

Family

ID=26293226

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8803876A Expired - Fee Related ES2011727A6 (en) 1987-12-22 1988-12-21 Aqueous formulations of piperidinylcyclopentylheptenoic acid derivatives

Country Status (29)

Country Link
JP (1) JPH02210A (en)
KR (1) KR890009402A (en)
CN (1) CN1034132A (en)
AT (1) AT395943B (en)
AU (1) AU615245B2 (en)
BE (1) BE1001704A3 (en)
CA (1) CA1328078C (en)
CH (1) CH676665A5 (en)
DE (1) DE3843059A1 (en)
DK (1) DK712888A (en)
ES (1) ES2011727A6 (en)
FI (1) FI885920L (en)
FR (1) FR2624731B1 (en)
GB (1) GB2211737B (en)
GR (1) GR880100854A (en)
HU (1) HU204700B (en)
IE (1) IE61995B1 (en)
IL (1) IL88764A0 (en)
IT (1) IT1224835B (en)
LU (1) LU87411A1 (en)
MY (1) MY103952A (en)
NL (1) NL8803126A (en)
NO (1) NO885689L (en)
NZ (1) NZ227446A (en)
PH (1) PH24982A (en)
PL (1) PL276595A1 (en)
PT (1) PT89301B (en)
SE (1) SE502288C2 (en)
ZW (1) ZW18088A1 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8814725D0 (en) * 1988-06-21 1988-07-27 Glaxo Group Ltd Medicaments
AU616571B2 (en) * 1988-10-28 1991-10-31 Shiseido Company Ltd. Cosmetic composition containing inclusion product with hydroxyalkylated cyclodextrin
IT1269578B (en) * 1994-04-22 1997-04-08 Chiesi Farma Spa MULTI-COMPONENT INCLUSION COMPLEXES WITH HIGH SOLUBILITY CONSISTING OF AN ACID TYPE DRUG, A CYCLODESTRINE AND A BASE.
KR100825736B1 (en) * 2005-12-07 2008-04-29 한국전자통신연구원 Apparatus for providing XML signnature in mobile environment and method thereof
KR100832740B1 (en) * 2007-01-17 2008-05-27 한국과학기술원 Mutant microorganism with improved branched chain amino acid production ability and method for producing branched chain amino acid using the same

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS503362B1 (en) * 1970-06-10 1975-02-04
JPS5443569B2 (en) * 1972-07-05 1979-12-20
HU181703B (en) * 1980-05-09 1983-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing aqueus solutuins of water insoluble or hardly soluble vitamines, steroides, localanesthetics, prostanoides and non-steroid and antiphlogistic agents
JPS57183772A (en) * 1981-04-29 1982-11-12 Glaxo Group Ltd Aminocyclopentanol acids and esters, manufacture and medicinal composition
JPS58116423A (en) * 1981-12-28 1983-07-11 Sumitomo Chem Co Ltd Methanoprostacycline pharmaceutical composition
JPS58192821A (en) * 1982-04-30 1983-11-10 Dainippon Pharmaceut Co Ltd Remedy for anoxia of cranial nerve cells
JPS5946228A (en) * 1982-09-08 1984-03-15 Zeria Shinyaku Kogyo Kk Method for producing water-soluble and lymphatic drug of biologically active organic compound
JPS5973576A (en) * 1982-09-16 1984-04-25 グラクソ・グル−プ・リミテツド Piperidinylcyclopentanolheptanoate
GB2127406B (en) * 1982-09-16 1986-03-05 Glaxo Group Ltd Piperidinlycyclopentanolheptenoic acid salt
DE3346123A1 (en) * 1983-12-21 1985-06-27 Janssen Pharmaceutica, N.V., Beerse PHARMACEUTICAL PREPARATIONS OF SUBSTANCES MEDICAL OR UNSTABLE IN WATER AND METHOD FOR THE PRODUCTION THEREOF
JPS60150039A (en) * 1984-01-17 1985-08-07 Minolta Camera Co Ltd Amphibious fixed-focus camera
DE3504044A1 (en) * 1985-02-04 1986-08-07 Schering AG, Berlin und Bergkamen, 1000 Berlin 9-HALOGEN PROSTAGLANDIN CLATHRATE AND THEIR USE AS A MEDICINAL PRODUCT
JPS6327440A (en) * 1986-07-18 1988-02-05 Sanraku Inc Glucosylated branched cyclodextrin-containing composition

Also Published As

Publication number Publication date
HUT50040A (en) 1989-12-28
IE883820L (en) 1989-06-22
CH676665A5 (en) 1991-02-28
DE3843059A1 (en) 1989-07-13
NL8803126A (en) 1989-07-17
FR2624731A1 (en) 1989-06-23
SE8804607D0 (en) 1988-12-21
PH24982A (en) 1990-12-26
AU615245B2 (en) 1991-09-26
NZ227446A (en) 1991-08-27
PT89301A (en) 1990-06-29
PT89301B (en) 1995-07-03
IE61995B1 (en) 1994-12-14
DK712888D0 (en) 1988-12-21
GB2211737B (en) 1991-12-11
AT395943B (en) 1993-04-26
IL88764A0 (en) 1989-07-31
GB2211737A (en) 1989-07-12
GR880100854A (en) 1994-03-31
DK712888A (en) 1989-06-23
SE502288C2 (en) 1995-09-25
AU2735688A (en) 1989-06-22
LU87411A1 (en) 1989-07-07
CN1034132A (en) 1989-07-26
ATA313088A (en) 1992-09-15
GB8829793D0 (en) 1989-02-15
IT1224835B (en) 1990-10-24
IT8848702A0 (en) 1988-12-21
SE8804607L (en) 1989-06-23
CA1328078C (en) 1994-03-29
JPH02210A (en) 1990-01-05
KR890009402A (en) 1989-08-01
FI885920A7 (en) 1989-06-23
PL276595A1 (en) 1989-08-21
HU204700B (en) 1992-02-28
FI885920L (en) 1989-06-23
NO885689D0 (en) 1988-12-21
NO885689L (en) 1989-06-23
MY103952A (en) 1993-10-30
BE1001704A3 (en) 1990-02-13
FR2624731B1 (en) 1992-10-23
ZW18088A1 (en) 1989-07-26

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Legal Events

Date Code Title Description
SA6 Expiration date (snapshot 920101)

Free format text: 2008-12-21

FD1A Patent lapsed

Effective date: 20010402