EE200400016A - Protsess 1,5-diarüül-3-trifluorometüül-delta²-pürasoliinide ratseemiliste ja enantiomeerselt puhaste derivaatide valmistamiseks - Google Patents

Protsess 1,5-diarüül-3-trifluorometüül-delta²-pürasoliinide ratseemiliste ja enantiomeerselt puhaste derivaatide valmistamiseks

Info

Publication number: EE200400016A
Authority: EE; Estonia
Prior art keywords: delta2; pyrazolines; diaryl; racemic; trifluoromethyl
Prior art date: 2001-06-18

Application number

EEP200400016A

Other languages

English (en)

Inventor

Alc�n-Marrugat Montserrat

Angel Pericas-Brondo Miguel

Rosa Cuberes-Altisen Mar�a

Frigola-Constansa Jordi

Original Assignee

Laboratorios Del Dr. Esteve, S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-06-18

Filing date

2002-06-06

Publication date

2004-04-15

2002-06-06 Application filed by Laboratorios Del Dr. Esteve, S.A. filed Critical Laboratorios Del Dr. Esteve, S.A.

2004-04-15 Publication of EE200400016A publication Critical patent/EE200400016A/et

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

EEP200400016A 2001-06-18 2002-06-06 Protsess 1,5-diarüül-3-trifluorometüül-delta²-pürasoliinide ratseemiliste ja enantiomeerselt puhaste derivaatide valmistamiseks EE200400016A (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
ES200101412A ES2183720B1 (es)	2001-06-18	2001-06-18	Procedimiento para la preparacion de derivados de 1,5-diaril-3-trifluorometil-delta2-pirazolinas racemicas y enantiomericamente puras.
PCT/ES2002/000274 WO2002102781A1 (es)	2001-06-18	2002-06-06	Procedimiento para la preparación de derivados de 1,5-diaril-3-trifluorometil-delta2-pirazolinas racémicas y enantioméricamente puras

Publications (1)

Publication Number	Publication Date
EE200400016A true EE200400016A (et)	2004-04-15

Family

ID=8498105

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200400016A EE200400016A (et)	2001-06-18	2002-06-06	Protsess 1,5-diarüül-3-trifluorometüül-delta²-pürasoliinide ratseemiliste ja enantiomeerselt puhaste derivaatide valmistamiseks

Country Status (26)

Country	Link
US (3)	US6846935B2 (et)
EP (1)	EP1408035B1 (et)
JP (1)	JP2005502604A (et)
KR (1)	KR20040018275A (et)
CN (1)	CN1275946C (et)
AR (1)	AR036050A1 (et)
AT (1)	ATE315030T1 (et)
BG (1)	BG108524A (et)
BR (1)	BR0211009A (et)
CA (1)	CA2451132C (et)
CZ (1)	CZ200481A3 (et)
DE (1)	DE60208551T2 (et)
DK (1)	DK1408035T3 (et)
EE (1)	EE200400016A (et)
ES (2)	ES2183720B1 (et)
HU (1)	HUP0401715A3 (et)
IL (1)	IL159367A0 (et)
MX (1)	MXPA03011783A (et)
NO (1)	NO20035642L (et)
PL (1)	PL367773A1 (et)
PT (1)	PT1408035E (et)
RU (1)	RU2288915C2 (et)
SI (1)	SI1408035T1 (et)
SK (1)	SK422004A3 (et)
WO (1)	WO2002102781A1 (et)
ZA (1)	ZA200400343B (et)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2183720B1 (es) *	2001-06-18	2004-01-16	Esteve Labor Dr	Procedimiento para la preparacion de derivados de 1,5-diaril-3-trifluorometil-delta2-pirazolinas racemicas y enantiomericamente puras.
US20080138282A1 (en) *	2004-06-03	2008-06-12	The Trustees Of Columbia University In The City Of New York	Radiolabeled Arylsulfonyl Compounds and Uses Thereof
DE102004057303A1 (de) *	2004-11-26	2006-06-01	Merck Patent Gmbh	Stabile Kristallmodifikationen von DOTAP Chlorid
EP1757587A1 (en) *	2005-07-15	2007-02-28	Laboratorios Del Dr. Esteve, S.A.	Substituted pyrazoline compounds, their preparation and use as medicaments
WO2014065575A1 (ko) *	2012-10-25	2014-05-01	주식회사유한양행	4,5-다이하이드로-1h-피라졸 유도체 또는 그의 염 및 이를 포함하는 약학 조성물

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE788658R (fr) *	1971-09-09	1973-03-12	Hoechst Ag	Derives de 3-(3', 4'-dichloro-6'-alkylphenyl) -delta2-pyrazolines, leurpreparation et leur utilisation comme agents d'azurage
ES2137138B1 (es) *	1998-05-29	2000-09-16	Esteve Labor Dr	Derivados de pirazolinas, su preparacion y su aplicacion como medicamentos.
US6376519B1 (en) *	1999-06-16	2002-04-23	Temple University-Of The Commonwealth Of Higher Education	1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines and inhibitors of cyclooxygenase-2
ES2183720B1 (es) *	2001-06-18	2004-01-16	Esteve Labor Dr	Procedimiento para la preparacion de derivados de 1,5-diaril-3-trifluorometil-delta2-pirazolinas racemicas y enantiomericamente puras.

2001
- 2001-06-18 ES ES200101412A patent/ES2183720B1/es not_active Expired - Fee Related
2002
- 2002-06-06 AT AT02735442T patent/ATE315030T1/de active
- 2002-06-06 PT PT02735442T patent/PT1408035E/pt unknown
- 2002-06-06 HU HU0401715A patent/HUP0401715A3/hu unknown
- 2002-06-06 IL IL15936702A patent/IL159367A0/xx unknown
- 2002-06-06 SI SI200230277T patent/SI1408035T1/sl unknown
- 2002-06-06 WO PCT/ES2002/000274 patent/WO2002102781A1/es not_active Ceased
- 2002-06-06 CZ CZ200481A patent/CZ200481A3/cs unknown
- 2002-06-06 EE EEP200400016A patent/EE200400016A/et unknown
- 2002-06-06 SK SK42-2004A patent/SK422004A3/sk unknown
- 2002-06-06 CN CNB028143280A patent/CN1275946C/zh not_active Expired - Fee Related
- 2002-06-06 JP JP2003505323A patent/JP2005502604A/ja active Pending
- 2002-06-06 US US10/312,194 patent/US6846935B2/en not_active Expired - Fee Related
- 2002-06-06 DK DK02735442T patent/DK1408035T3/da active
- 2002-06-06 PL PL02367773A patent/PL367773A1/xx not_active Application Discontinuation
- 2002-06-06 BR BR0211009-1A patent/BR0211009A/pt not_active IP Right Cessation
- 2002-06-06 CA CA2451132A patent/CA2451132C/en not_active Expired - Fee Related
- 2002-06-06 KR KR10-2003-7016500A patent/KR20040018275A/ko not_active Ceased
- 2002-06-06 DE DE60208551T patent/DE60208551T2/de not_active Expired - Lifetime
- 2002-06-06 RU RU2004101050/04A patent/RU2288915C2/ru not_active IP Right Cessation
- 2002-06-06 EP EP02735442A patent/EP1408035B1/en not_active Expired - Lifetime
- 2002-06-06 ES ES02735442T patent/ES2256483T3/es not_active Expired - Lifetime
- 2002-06-06 MX MXPA03011783A patent/MXPA03011783A/es active IP Right Grant
- 2002-06-12 AR ARP020102218A patent/AR036050A1/es not_active Application Discontinuation
2003
- 2003-12-17 NO NO20035642A patent/NO20035642L/no not_active Application Discontinuation
2004
- 2004-01-13 BG BG108524A patent/BG108524A/bg unknown
- 2004-01-16 ZA ZA2004/00343A patent/ZA200400343B/en unknown
- 2004-12-08 US US11/007,449 patent/US6958403B2/en not_active Expired - Fee Related
- 2004-12-08 US US11/006,931 patent/US20050096474A1/en not_active Abandoned

Also Published As

Publication number	Publication date
US20050096373A1 (en)	2005-05-05
NO20035642D0 (no)	2003-12-17
PT1408035E (pt)	2006-05-31
MXPA03011783A (es)	2004-04-02
KR20040018275A (ko)	2004-03-02
NO20035642L (no)	2004-02-12
IL159367A0 (en)	2004-06-01
US20040019222A1 (en)	2004-01-29
SK422004A3 (en)	2004-07-07
HUP0401715A2 (hu)	2005-01-28
EP1408035A1 (en)	2004-04-14
CN1275946C (zh)	2006-09-20
CZ200481A3 (cs)	2004-07-14
CA2451132A1 (en)	2002-12-27
DK1408035T3 (da)	2006-05-08
CN1610672A (zh)	2005-04-27
US20050096474A1 (en)	2005-05-05
ES2183720A1 (es)	2003-03-16
SI1408035T1 (sl)	2006-04-30
HUP0401715A3 (en)	2005-06-28
DE60208551D1 (de)	2006-03-30
ATE315030T1 (de)	2006-02-15
CA2451132C (en)	2010-10-12
WO2002102781A1 (es)	2002-12-27
RU2288915C2 (ru)	2006-12-10
BG108524A (bg)	2004-08-31
BR0211009A (pt)	2004-11-03
DE60208551T2 (de)	2006-10-19
RU2004101050A (ru)	2005-06-27
PL367773A1 (en)	2005-03-07
HK1077058A1 (en)	2006-02-03
ES2183720B1 (es)	2004-01-16
US6846935B2 (en)	2005-01-25
ES2256483T3 (es)	2006-07-16
JP2005502604A (ja)	2005-01-27
AR036050A1 (es)	2004-08-04
US6958403B2 (en)	2005-10-25
EP1408035B1 (en)	2006-01-04
ZA200400343B (en)	2005-03-30

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