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EE200300504A - 3,7-diasabitsüklo[3.3.1]preparaadid, nende valmistamise meetod ja nimetatud preparaatide kasutaminesüdame arütmiate profülaktikas või ravis - Google Patents

3,7-diasabitsüklo[3.3.1]preparaadid, nende valmistamise meetod ja nimetatud preparaatide kasutaminesüdame arütmiate profülaktikas või ravis

Info

Publication number
EE200300504A
EE200300504A EEP200300504A EEP200300504A EE200300504A EE 200300504 A EE200300504 A EE 200300504A EE P200300504 A EEP200300504 A EE P200300504A EE P200300504 A EEP200300504 A EE P200300504A EE 200300504 A EE200300504 A EE 200300504A
Authority
EE
Estonia
Prior art keywords
diazabicyclo
prophylaxis
preparations
preparation
treatment
Prior art date
Application number
EEP200300504A
Other languages
English (en)
Inventor
Barnwell Neil
Bj�re Annika
Cheema Lal
Cladingboel David
Herring Adam
L�vqvist Karin
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of EE200300504A publication Critical patent/EE200300504A/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
EEP200300504A 2001-04-12 2002-04-12 3,7-diasabitsüklo[3.3.1]preparaadid, nende valmistamise meetod ja nimetatud preparaatide kasutaminesüdame arütmiate profülaktikas või ravis EE200300504A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0101327A SE0101327D0 (sv) 2001-04-12 2001-04-12 New crystalline forms
PCT/SE2002/000725 WO2002083688A1 (en) 2001-04-12 2002-04-12 3,7-diazabicyclo [3.3.1] formulations as antiarhythmic compounds

Publications (1)

Publication Number Publication Date
EE200300504A true EE200300504A (et) 2003-12-15

Family

ID=20283783

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300504A EE200300504A (et) 2001-04-12 2002-04-12 3,7-diasabitsüklo[3.3.1]preparaadid, nende valmistamise meetod ja nimetatud preparaatide kasutaminesüdame arütmiate profülaktikas või ravis

Country Status (29)

Country Link
US (1) US7217708B2 (et)
EP (2) EP1389213B1 (et)
JP (1) JP2004525970A (et)
KR (1) KR20030087078A (et)
CN (1) CN1269823C (et)
AR (1) AR035452A1 (et)
AT (1) ATE323095T1 (et)
BR (1) BR0208829A (et)
CA (1) CA2443470A1 (et)
CZ (1) CZ20032760A3 (et)
DE (1) DE60210598T2 (et)
DK (1) DK1389213T3 (et)
EE (1) EE200300504A (et)
ES (1) ES2261721T3 (et)
HU (1) HUP0303487A3 (et)
IL (1) IL158250A0 (et)
IS (1) IS6980A (et)
MX (1) MXPA03009206A (et)
NO (1) NO20034527L (et)
NZ (1) NZ528560A (et)
PL (1) PL367179A1 (et)
PT (1) PT1389213E (et)
RU (1) RU2286993C2 (et)
SE (1) SE0101327D0 (et)
SK (1) SK12572003A3 (et)
TW (1) TWI237025B (et)
UA (1) UA74629C2 (et)
WO (1) WO2002083688A1 (et)
ZA (1) ZA200307759B (et)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI259836B (en) * 2001-04-12 2006-08-11 Astrazeneca Ab Modified release formulation suitable for antiarrhythmic compounds
SE0401539D0 (sv) * 2004-06-15 2004-06-15 Astrazeneca Ab New compounds
SE0401540D0 (sv) * 2004-06-15 2004-06-15 Astrazeneca Ab New compounds
EP1893619A1 (en) * 2005-06-13 2008-03-05 AstraZeneca AB New oxabispidine compounds for the treatment of cardiac arrhytmias
WO2006137772A1 (en) * 2005-06-20 2006-12-28 Astrazeneca Ab New physical form of n,n´- disubstituted oxabispidines
CA2610089A1 (en) * 2005-06-20 2006-12-28 Astrazeneca Ab Process for the preparation of n,n´- disubstituted oxabispidines
TW200734342A (en) * 2005-12-15 2007-09-16 Astrazeneca Ab New compounds for the treatment of cardiac arrhythmias
EP2001881A2 (en) * 2006-03-07 2008-12-17 Endacea, Inc. Compositions and methods for treating respiratory disorders
PT3357911T (pt) 2006-06-26 2022-07-11 Akebia Therapeutics Inc Inibidores da prolil-hidroxilase e métodos de utilização
WO2012170442A1 (en) 2011-06-06 2012-12-13 Akebia Therapeutics Inc. Compounds and compositions for stabilizing hypoxia inducible factor-2 alpha as a method for treating cancer
NO2686520T3 (et) 2011-06-06 2018-03-17
EP3007695B1 (en) 2013-06-13 2024-02-07 Akebia Therapeutics, Inc. Compositions and methods for treating anemia
CR20160222U (es) 2013-11-15 2016-08-26 Akebia Therapeutics Inc Formas solidas de acido { [ -(3- clorofenil) -3- hidroxipiridin -2-carbonil] amino} acetico, composiciones, y usos de las mismas
CA2974691A1 (en) 2015-01-23 2016-07-28 Akebia Therapeutics, Inc. Solid forms of 2-(5-(3-fluorophenyl)-3-hydroxypicolinamido)acetic acid, compositions, and uses thereof
UA123308C2 (uk) 2015-04-01 2021-03-17 Екебіа Терапьютікс, Інк. Композиції і способи для лікування анемії
JP7440989B2 (ja) 2018-05-09 2024-02-29 アケビア セラピューティクス インコーポレイテッド 2-[5-(3-クロロフェニル)-3-ヒドロキシピリジン-2-カルボニル]アミノ]酢酸を調製するための方法
US12304905B2 (en) 2019-03-28 2025-05-20 1ST Biotherapeutics, Inc. Pharmaceutical salts of benzothiazol compounds, polymorphs and methods for preparation thereof
US11524939B2 (en) 2019-11-13 2022-12-13 Akebia Therapeutics, Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino} acetic acid

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3732094A1 (de) * 1987-09-24 1989-04-06 Basf Ag Bispidinderivate als klasse iii-antiarrhythmika
US5110933A (en) 1989-11-13 1992-05-05 Board Of Regents Of Oklahoma State University Salts of 3-azabicyclo[3.3.1]nonanes as antiarrhythmic agents, and precursors thereof
SE9704709D0 (sv) 1997-12-17 1997-12-17 Astra Ab Pharmaceutically active compounds
SE9902268D0 (sv) 1999-06-16 1999-06-16 Astra Ab Pharmaceutically active compounds
SE9903759D0 (sv) * 1999-10-18 1999-10-18 Astra Ab Pharmaceutically active compounds

Also Published As

Publication number Publication date
BR0208829A (pt) 2004-03-09
AR035452A1 (es) 2004-05-26
RU2003129231A (ru) 2005-04-10
PT1389213E (pt) 2006-07-31
SK12572003A3 (sk) 2004-07-07
PL367179A1 (en) 2005-02-21
RU2286993C2 (ru) 2006-11-10
ATE323095T1 (de) 2006-04-15
US20040143000A1 (en) 2004-07-22
EP1389213B1 (en) 2006-04-12
IL158250A0 (en) 2004-05-12
HK1061026A1 (en) 2004-09-03
ZA200307759B (en) 2005-01-03
TWI237025B (en) 2005-08-01
HUP0303487A3 (en) 2005-04-28
CA2443470A1 (en) 2002-10-24
KR20030087078A (ko) 2003-11-12
DK1389213T3 (da) 2006-07-10
UA74629C2 (en) 2006-01-16
US7217708B2 (en) 2007-05-15
JP2004525970A (ja) 2004-08-26
DE60210598D1 (de) 2006-05-24
ES2261721T3 (es) 2006-11-16
CN1514837A (zh) 2004-07-21
CN1269823C (zh) 2006-08-16
CZ20032760A3 (cs) 2004-01-14
NO20034527D0 (no) 2003-10-09
HUP0303487A2 (hu) 2004-01-28
IS6980A (is) 2003-10-08
NO20034527L (no) 2003-12-10
SE0101327D0 (sv) 2001-04-12
EP1389213A1 (en) 2004-02-18
MXPA03009206A (es) 2004-01-29
EP1550663A1 (en) 2005-07-06
NZ528560A (en) 2005-05-27
WO2002083688A1 (en) 2002-10-24
DE60210598T2 (de) 2007-02-08

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