EE200300435A - 4-(2-butüülamino)-2,7-dimetüül-8-(2-metüül-6-metoksüpürid-3-üül)[1,5-a]pürasolo-1, 3,5-triasiin, selle farmatseutiliselt vastuvõetavad eelravimid võifarmatseutiliselt vastuvõetavad soolad ning nendekasutamine - Google Patents

4-(2-butüülamino)-2,7-dimetüül-8-(2-metüül-6-metoksüpürid-3-üül)[1,5-a]pürasolo-1, 3,5-triasiin, selle farmatseutiliselt vastuvõetavad eelravimid võifarmatseutiliselt vastuvõetavad soolad ning nendekasutamine

Info

Publication number: EE200300435A
Authority: EE; Estonia
Prior art keywords: pharmaceutically acceptable; methoxypyrid; pyrazolo; butylamino; triazine
Prior art date: 2001-03-13

Application number

EEP200300435A

Other languages

English (en)

Inventor

J. Gilligan Paul

Original Assignee

Bristol-Myers Squibb Pharma Company

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-03-13

Filing date

2002-03-06

Publication date

2003-12-15

2002-03-06 Application filed by Bristol-Myers Squibb Pharma Company filed Critical Bristol-Myers Squibb Pharma Company

2003-12-15 Publication of EE200300435A publication Critical patent/EE200300435A/et

2011-06-15 Publication of EE05433B1 publication Critical patent/EE05433B1/et

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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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EEP200300435A 2001-03-13 2002-03-06 4-(2-butlamino)-2,7-dimetl-8-(2-metl-6-metoksprid-3-l)[1,5-a]prasolo-1,3,5-triasiin, selle farmatseutiliselt vastuv?etavad eelravimid v?i farmatseutiliselt vastuv?etavad soolad ning nende kasutamine EE05433B1 (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US27540301P	2001-03-13	2001-03-13
PCT/US2002/006837 WO2002072202A1 (en)	2001-03-13	2002-03-06	4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands

Publications (2)

Publication Number	Publication Date
EE200300435A true EE200300435A (et)	2003-12-15
EE05433B1 EE05433B1 (et)	2011-06-15

Family

ID=23052141

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200300435A EE05433B1 (et)	2001-03-13	2002-03-06	4-(2-butlamino)-2,7-dimetl-8-(2-metl-6-metoksprid-3-l)[1,5-a]prasolo-1,3,5-triasiin, selle farmatseutiliselt vastuv?etavad eelravimid v?i farmatseutiliselt vastuv?etavad soolad ning nende kasutamine

Country Status (35)

Country	Link
US (4)	US20030125330A1 (et)
EP (1)	EP1368094B1 (et)
JP (1)	JP4549630B2 (et)
KR (1)	KR100875595B1 (et)
CN (1)	CN100427093C (et)
AR (1)	AR032986A1 (et)
AT (1)	ATE355102T1 (et)
AU (1)	AU2002245605B2 (et)
BG (1)	BG66331B1 (et)
BR (1)	BR0208357A (et)
CA (1)	CA2440553C (et)
CY (1)	CY1106607T1 (et)
CZ (1)	CZ20032481A3 (et)
DE (1)	DE60218434T2 (et)
DK (1)	DK1368094T3 (et)
EE (1)	EE05433B1 (et)
ES (1)	ES2282401T3 (et)
GE (1)	GEP20053608B (et)
HR (1)	HRP20030822B1 (et)
HU (1)	HU229317B1 (et)
IL (2)	IL157615A0 (et)
IS (1)	IS2839B (et)
MX (1)	MXPA03008185A (et)
MY (1)	MY146935A (et)
NO (1)	NO328580B1 (et)
NZ (1)	NZ528207A (et)
PL (1)	PL208278B1 (et)
PT (1)	PT1368094E (et)
RS (1)	RS50863B (et)
RU (1)	RU2292347C2 (et)
SK (1)	SK287603B6 (et)
TW (1)	TWI257388B (et)
UA (1)	UA74634C2 (et)
WO (1)	WO2002072202A1 (et)
ZA (1)	ZA200306995B (et)

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US20140206667A1 (en)	2012-11-14	2014-07-24	Michela Gallagher	Methods and compositions for treating schizophrenia
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CN110996943A (zh)	2017-08-14	2020-04-10	云杉生物科学公司	促肾上腺皮质激素释放因子受体拮抗剂
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2002
- 2002-03-06 US US10/092,312 patent/US20030125330A1/en not_active Abandoned
- 2002-03-06 NZ NZ528207A patent/NZ528207A/en not_active IP Right Cessation
- 2002-03-06 DK DK02713776T patent/DK1368094T3/da active
- 2002-03-06 PL PL368644A patent/PL208278B1/pl unknown
- 2002-03-06 HU HU0303480A patent/HU229317B1/hu not_active IP Right Cessation
- 2002-03-06 IL IL15761502A patent/IL157615A0/xx unknown
- 2002-03-06 EP EP02713776A patent/EP1368094B1/en not_active Expired - Lifetime
- 2002-03-06 CA CA2440553A patent/CA2440553C/en not_active Expired - Fee Related
- 2002-03-06 RU RU2003130093/04A patent/RU2292347C2/ru not_active IP Right Cessation
- 2002-03-06 AU AU2002245605A patent/AU2002245605B2/en not_active Ceased
- 2002-03-06 HR HR20030822A patent/HRP20030822B1/xx not_active IP Right Cessation
- 2002-03-06 EE EEP200300435A patent/EE05433B1/et not_active IP Right Cessation
- 2002-03-06 SK SK1157-2003A patent/SK287603B6/sk not_active IP Right Cessation
- 2002-03-06 BR BR0208357-4A patent/BR0208357A/pt active Search and Examination
- 2002-03-06 CN CNB028064151A patent/CN100427093C/zh not_active Expired - Fee Related
- 2002-03-06 RS YUP-715/03A patent/RS50863B/sr unknown
- 2002-03-06 JP JP2002571157A patent/JP4549630B2/ja not_active Expired - Fee Related
- 2002-03-06 MX MXPA03008185A patent/MXPA03008185A/es active IP Right Grant
- 2002-03-06 CZ CZ20032481A patent/CZ20032481A3/cs unknown
- 2002-03-06 DE DE60218434T patent/DE60218434T2/de not_active Expired - Lifetime
- 2002-03-06 GE GE5322A patent/GEP20053608B/en unknown
- 2002-03-06 PT PT02713776T patent/PT1368094E/pt unknown
- 2002-03-06 AT AT02713776T patent/ATE355102T1/de active
- 2002-03-06 WO PCT/US2002/006837 patent/WO2002072202A1/en not_active Ceased
- 2002-03-06 KR KR1020037011913A patent/KR100875595B1/ko not_active Expired - Fee Related
- 2002-03-06 ES ES02713776T patent/ES2282401T3/es not_active Expired - Lifetime
- 2002-03-12 MY MYPI20020879A patent/MY146935A/en unknown
- 2002-03-13 TW TW091104706A patent/TWI257388B/zh not_active IP Right Cessation
- 2002-03-13 AR ARP020100908A patent/AR032986A1/es not_active Application Discontinuation
- 2002-06-03 UA UA2003109244A patent/UA74634C2/uk unknown
2003
- 2003-02-05 US US10/358,652 patent/US7157578B2/en not_active Expired - Lifetime
- 2003-08-27 IL IL157615A patent/IL157615A/en not_active IP Right Cessation
- 2003-09-08 ZA ZA200306995A patent/ZA200306995B/en unknown
- 2003-09-10 IS IS6947A patent/IS2839B/is unknown
- 2003-09-11 NO NO20034023A patent/NO328580B1/no not_active IP Right Cessation
- 2003-09-23 BG BG108189A patent/BG66331B1/bg unknown
2006
- 2006-11-07 US US11/593,715 patent/US7358252B2/en not_active Expired - Lifetime
2007
- 2007-05-18 CY CY20071100678T patent/CY1106607T1/el unknown
2008
- 2008-02-13 US US12/030,439 patent/US7662817B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
WO2002072202A1 (en)	2002-09-19
IS2839B (is)	2013-06-15
KR100875595B1 (ko)	2008-12-23
DE60218434T2 (de)	2007-11-08
CZ20032481A3 (cs)	2007-12-27
US20030125330A1 (en)	2003-07-03
HRP20030822A2 (en)	2004-04-30
PL368644A1 (en)	2005-04-04
HK1057182A1 (en)	2004-03-19
HU229317B1 (en)	2013-10-28
US7358252B2 (en)	2008-04-15
IS6947A (is)	2003-09-10
ATE355102T1 (de)	2006-03-15
AU2002245605B2 (en)	2006-02-02
CN100427093C (zh)	2008-10-22
DK1368094T3 (da)	2007-07-02
IL157615A0 (en)	2004-03-28
UA74634C2 (uk)	2006-01-16
DE60218434D1 (en)	2007-04-12
TWI257388B (en)	2006-07-01
US7157578B2 (en)	2007-01-02
NO328580B1 (no)	2010-03-22
RS50863B (sr)	2010-08-31
YU71503A (sh)	2006-05-25
US20040014760A1 (en)	2004-01-22
AR032986A1 (es)	2003-12-03
CA2440553A1 (en)	2002-09-19
HRP20030822B1 (en)	2008-01-31
GEP20053608B (en)	2005-09-12
SK287603B6 (sk)	2011-03-04
CA2440553C (en)	2010-06-08
SK11572003A3 (sk)	2004-02-03
US20080139567A1 (en)	2008-06-12
EP1368094B1 (en)	2007-02-28
MXPA03008185A (es)	2004-01-29
NZ528207A (en)	2006-02-24
HUP0303480A2 (hu)	2004-01-28
BG66331B1 (bg)	2013-06-28
JP4549630B2 (ja)	2010-09-22
RU2292347C2 (ru)	2007-01-27
HUP0303480A3 (en)	2005-12-28
EE05433B1 (et)	2011-06-15
KR20030080086A (ko)	2003-10-10
NO20034023L (no)	2003-09-11
CN1509196A (zh)	2004-06-30
PL208278B1 (pl)	2011-04-29
ES2282401T3 (es)	2007-10-16
IL157615A (en)	2009-09-01
NO20034023D0 (no)	2003-09-11
US20070054913A1 (en)	2007-03-08
CY1106607T1 (el)	2012-01-25
PT1368094E (pt)	2007-05-31
US7662817B2 (en)	2010-02-16
MY146935A (en)	2012-10-15
EP1368094A4 (en)	2004-03-31
EP1368094A1 (en)	2003-12-10
BG108189A (bg)	2004-09-30
RU2003130093A (ru)	2005-03-20
ZA200306995B (en)	2004-09-08
JP2004530662A (ja)	2004-10-07
BR0208357A (pt)	2004-06-29

Publication	Publication Date	Title
EE200300435A (et)	2003-12-15	4-(2-butüülamino)-2,7-dimetüül-8-(2-metüül-6-metoksüpürid-3-üül)[1,5-a]pürasolo-1, 3,5-triasiin, selle farmatseutiliselt vastuvõetavad eelravimid võifarmatseutiliselt vastuvõetavad soolad ning nendekasutamine
EE05223B1 (et)	2009-10-15	Triasoloprimidiini hendid, meetod nende valmistamiseks ning nende kasutamine
DK1242425T3 (da)	2004-07-05	N-(5,7-dimethoxy[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)arylsulfonamid-forbindelser og deres anvendelse som herbicider
EE200300544A (et)	2004-02-16	4-anilinokinoliin-3-karboksamiidid, nende kasutamine ning valmistamine
DK1416935T3 (da)	2008-07-07	4-Amino-6-phenyl-pyrrolo[2,3-d]pyrimidinderivater
DK1625847T3 (da)	2010-10-18	Medicinsk anvendelse af tetrahydrotriazolo[4,3-A]pyrazin
EE200300400A (et)	2003-12-15	Pürimidiiniühendid, nende valmistamismeetod ning kasutamine
DE60207241D1 (de)	2005-12-15	5-amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3-d)pyrimidin-derivate
DE50213202D1 (de)	2009-02-26	Cdk inhibitorische pyrimidine, deren herstellung und verwendung als arzneimittel
EE200200704A (et)	2004-08-16	Uued ühendid, meetod nende valmistamiseks ning nende kasutamine
DK1250328T4 (da)	2010-06-28	Dihydro-1,3,5-triazindiaminderivater og terapeutisk anvendelse deraf
EE200300347A (et)	2003-12-15	Aniliini derivaadid, mis on kasulikud kui fosfodiesteraas 4 inhibiitorid
ATE303388T1 (de)	2005-09-15	Substituierte 2-pyridinyl-6,7,8,9- tetrahydropyrimidoc1,2-aöpyrimidin-4-on- und 7- pyridinyl-2,3-dihydroimidazo-c1,2-aöpyrimidin- 5(1h)onderivate
ATE267201T1 (de)	2004-06-15	4-(2-phenylthiazol-5-yl)1,4- diazabicyclo(3.2.2)nonanederivate, ihre herstellung und therapeutische verwendung
DE60127434D1 (de)	2007-05-03	Benzoxazinonderivative, deren herstellung und verwendung
DE60208044D1 (de)	2006-01-19	Acylaminothiazolderivate, deren herstellung und deren therapeutische verwendung
NO20014050D0 (no)	2001-08-20	1-aryl-1,3,5-triazin-4-tion-2,6-dioner, fremstilling derav og anvendelse derav som herbicider
ATE329908T1 (de)	2006-07-15	Arylethene-sulfonamid derivate, deren herstellung und deren verwendung als endothelin-antagonisten
ATE346069T1 (de)	2006-12-15	3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino(4, - b)indol-1-karboxamid-derivate, ihre herstellung und therapeutische verwendung
PT1326866E (pt)	2005-08-31	3,4-di-hidropirido[1,2-a]pirimidinas substituidas
PT1325010E (pt)	2005-08-31	3, 4-di-hidropirimido [1,2-a] pirimidinas e 3, 4-di-hidropirazino [1,2-a] pirimidinas substituidas
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ITMI20002173A0 (it)	2000-10-09	Procedimento per la preparazione di (s)-n-terbutil-1,2,3,4-treraidroisochinolin-3-carbossiammide
ES1049770Y (es)	2002-05-16	Servilleta para pinchos y similares.
ES1048428Y (es)	2001-12-16	Almohada perfeccionada.

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