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EE200000441A - 2-(puriin-9-üül) tetrahüdrofuraan-3,4-diooli derivaadid - Google Patents

2-(puriin-9-üül) tetrahüdrofuraan-3,4-diooli derivaadid

Info

Publication number
EE200000441A
EE200000441A EEP200000441A EEP200000441A EE200000441A EE 200000441 A EE200000441 A EE 200000441A EE P200000441 A EEP200000441 A EE P200000441A EE P200000441 A EEP200000441 A EE P200000441A EE 200000441 A EE200000441 A EE 200000441A
Authority
EE
Estonia
Prior art keywords
purin
tetrahydrofuran
diol derivatives
diol
derivatives
Prior art date
Application number
EEP200000441A
Other languages
English (en)
Estonian (et)
Inventor
Peter Charles Cousins Richard
Chan Chuen
Cox Brian
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9802066.2A external-priority patent/GB9802066D0/en
Priority claimed from GBGB9813528.8A external-priority patent/GB9813528D0/en
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of EE200000441A publication Critical patent/EE200000441A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EEP200000441A 1998-01-31 1999-01-29 2-(puriin-9-üül) tetrahüdrofuraan-3,4-diooli derivaadid EE200000441A (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9802066.2A GB9802066D0 (en) 1998-01-31 1998-01-31 Chemical compounds
GBGB9813528.8A GB9813528D0 (en) 1998-06-23 1998-06-23 Chemical compounds
PCT/EP1999/000503 WO1999038877A2 (fr) 1998-01-31 1999-01-29 Derives de 2-(purine-9-yl)-tetrahydrofurane-3,4-diol

Publications (1)

Publication Number Publication Date
EE200000441A true EE200000441A (et) 2001-12-17

Family

ID=26313042

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200000441A EE200000441A (et) 1998-01-31 1999-01-29 2-(puriin-9-üül) tetrahüdrofuraan-3,4-diooli derivaadid

Country Status (38)

Country Link
US (1) US6762170B1 (fr)
EP (1) EP1051425B1 (fr)
JP (1) JP2002501928A (fr)
KR (1) KR20010034473A (fr)
CN (1) CN1289338A (fr)
AP (1) AP2000001875A0 (fr)
AR (1) AR014508A1 (fr)
AT (1) ATE226957T1 (fr)
AU (1) AU757183B2 (fr)
BG (1) BG63783B1 (fr)
BR (1) BR9907270A (fr)
CA (1) CA2318278A1 (fr)
CO (1) CO4980872A1 (fr)
DE (1) DE69903708T2 (fr)
DK (1) DK1051425T3 (fr)
EA (1) EA003194B1 (fr)
EE (1) EE200000441A (fr)
ES (1) ES2186330T3 (fr)
GE (1) GEP20022839B (fr)
HR (1) HRP20000511A2 (fr)
HU (1) HUP0101305A3 (fr)
ID (1) ID26326A (fr)
IL (1) IL137042A0 (fr)
IS (1) IS5550A (fr)
MA (1) MA26601A1 (fr)
NO (1) NO20003867L (fr)
NZ (1) NZ505452A (fr)
OA (1) OA11447A (fr)
PE (1) PE20000280A1 (fr)
PL (1) PL342670A1 (fr)
PT (1) PT1051425E (fr)
SI (1) SI1051425T1 (fr)
SK (1) SK11192000A3 (fr)
SV (1) SV1999000009A (fr)
TR (1) TR200002218T2 (fr)
TW (1) TW434250B (fr)
WO (1) WO1999038877A2 (fr)
YU (1) YU44900A (fr)

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GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
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UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
WO2012034095A1 (fr) 2010-09-09 2012-03-15 Irm Llc Composés et compositions comme inhibiteurs de trk
EP2673277A1 (fr) 2011-02-10 2013-12-18 Novartis AG Composés de [1, 2, 4]triazolo [4, 3 -b]pyridazine en tant qu'inhibiteurs de la tyrosine kinase c-met
JP5808826B2 (ja) 2011-02-23 2015-11-10 インテリカイン， エルエルシー 複素環化合物およびその使用
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Also Published As

Publication number Publication date
HUP0101305A2 (hu) 2002-04-29
CA2318278A1 (fr) 1999-08-05
EA200000723A1 (ru) 2001-04-23
HUP0101305A3 (en) 2002-08-28
PL342670A1 (en) 2001-07-02
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