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EE200000328A - Bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod ja kasutamine ning farmatseutiline kompositsioon ja selle valmistamismeetod - Google Patents

Bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod ja kasutamine ning farmatseutiline kompositsioon ja selle valmistamismeetod

Info

Publication number
EE200000328A
EE200000328A EEP200000328A EEP200000328A EE200000328A EE 200000328 A EE200000328 A EE 200000328A EE P200000328 A EEP200000328 A EE P200000328A EE P200000328 A EEP200000328 A EE P200000328A EE 200000328 A EE200000328 A EE 200000328A
Authority
EE
Estonia
Prior art keywords
preparation
benzodioxane
benzofuran
pharmaceutical compositions
benzopyran derivatives
Prior art date
Application number
EEP200000328A
Other languages
English (en)
Inventor
Tom Bert Paul Wigerinck Piet
Gaston Verschueren Wim
Francis Josephine Schroven Marc
Frans Leopold De Bruyn Marcel
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of EE200000328A publication Critical patent/EE200000328A/et
Publication of EE04438B1 publication Critical patent/EE04438B1/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
EEP200000328A 1997-12-05 1998-11-27 Bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod ja kasutamine ning farmatseutiline kompositsioon ja selle valmistamismeetod EE04438B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP97203808 1997-12-05
PCT/EP1998/007771 WO1999029687A1 (en) 1997-12-05 1998-11-27 (benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties

Publications (2)

Publication Number Publication Date
EE200000328A true EE200000328A (et) 2001-08-15
EE04438B1 EE04438B1 (et) 2005-02-15

Family

ID=8229014

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200000328A EE04438B1 (et) 1997-12-05 1998-11-27 Bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod ja kasutamine ning farmatseutiline kompositsioon ja selle valmistamismeetod

Country Status (31)

Country Link
US (4) US6133277A (et)
EP (1) EP1036073B8 (et)
JP (1) JP2001525407A (et)
KR (1) KR100591605B1 (et)
CN (1) CN1155597C (et)
AR (1) AR017195A1 (et)
AT (1) ATE334125T1 (et)
AU (1) AU748669B2 (et)
BG (1) BG64624B1 (et)
BR (1) BR9814256A (et)
CA (1) CA2311669C (et)
CO (1) CO5011114A1 (et)
CZ (1) CZ297895B6 (et)
DE (1) DE69835372T2 (et)
EA (1) EA003365B1 (et)
EE (1) EE04438B1 (et)
ES (1) ES2270541T3 (et)
HR (1) HRP20000340B1 (et)
HU (1) HU224813B1 (et)
ID (1) ID24616A (et)
IL (1) IL136529A (et)
MY (1) MY124586A (et)
NO (1) NO320727B1 (et)
NZ (1) NZ503603A (et)
PL (1) PL191144B1 (et)
SK (1) SK286268B6 (et)
TR (1) TR200001542T2 (et)
TW (1) TW577886B (et)
UA (1) UA70308C2 (et)
WO (1) WO1999029687A1 (et)
ZA (1) ZA9811081B (et)

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US6133277A (en) 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
PL198552B1 (pl) * 1999-06-02 2008-06-30 Janssen Pharmaceutica Nv Pochodna benzopiranu podstawionego aminoalkilem i sposób jej otrzymywania oraz kompozycja farmaceutyczna i sposób jej otrzymywania
HUP0201344A3 (en) * 1999-06-02 2005-09-28 Janssen Pharmaceutica Nv Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives, process for their preparation and pharmaceutical compositions containing the compounds
JO2352B1 (en) * 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus
JO2654B1 (en) * 2000-09-04 2012-06-17 شركة جانسين فارماسوتيكا ان. في Multiple aryl caroxa amides are useful as lipid - lowering agents
JO2409B1 (en) * 2000-11-21 2007-06-17 شركة جانسين فارماسوتيكا ان. في Second-phenyl carboxy amides are useful as lipid-lowering agents
US6688079B2 (en) 2001-04-18 2004-02-10 Kraft Foods Holdings, Inc. Method for manufacturing flexible packages having slide closures
EP1445324A4 (en) * 2001-11-09 2005-02-16 Kaneka Corp PROCESS FOR PRODUCING OPTICALLY ACTIVE CHROMAN DERIVATIVE AND INTERMEDIATE PRODUCT
ES2199086B1 (es) 2002-07-31 2005-06-01 Cepa Schwarz Pharma Sl Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
US7071821B2 (en) * 2003-05-14 2006-07-04 Bellsouth Intellectual Property Corporation Method and system for alerting a person to a situation
ITTO20030140U1 (it) * 2003-09-16 2005-03-17 Interfila Srl Matita cosmetica
US7514461B2 (en) 2003-09-19 2009-04-07 Edison Pharmaceuticals, Inc. Chroman derivatives
AU2004295058B9 (en) 2003-11-20 2011-06-30 Janssen Pharmaceutica N.V. 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(ADP-ribose) polymerase inhibitors
BRPI0416817A (pt) 2003-11-20 2007-03-06 Janssen Pharmaceutica Nv 2-quinolinonas e 2-quinoxalinonas 7-fenilalquila substituìdas como inibidores da poli(adp-ribose)polimerase
ES2238015B1 (es) * 2004-01-30 2006-11-01 Cepa Schwarz Pharma, S.L. Derivados de cicloalcanodionas con actividad neuroprotectora.
NZ551799A (en) 2004-06-30 2009-11-27 Janssen Pharmaceutica Nv Phthalazine derivatives as PARP inhibitors
BRPI0512790A (pt) 2004-06-30 2008-04-08 Janssen Pharmaceutica Nv derivados de 2-alquil quinazolinona substituìdos como inibidores de parp
WO2006003148A1 (en) 2004-06-30 2006-01-12 Janssen Pharmaceutica N.V. Quinazolinedione derivatives as parp inhibitors
RU2391350C2 (ru) * 2004-07-02 2010-06-10 Базелль Полиолефине Гмбх Способ рацемоселективного синтеза анса-металлоценов
DE102004032277A1 (de) * 2004-07-02 2006-01-19 Basell Polyolefine Gmbh Verfahren zur racemoselektiven Synthese von ansa-Metallocenen
EP1856126A2 (en) 2005-02-17 2007-11-21 Wyeth a Corporation of the State of Delaware Cycloalkylfused indole, benzothiophene, benzofuran and indene derivatives
CN101203505A (zh) * 2005-04-22 2008-06-18 惠氏公司 苯并二氢吡喃和苯并吡喃衍生物及其用途
WO2008015538A2 (en) * 2006-07-31 2008-02-07 Schwarz Pharma S.L. Use of diaza- and thiaza-cycloalkanediones for preventing and/or treating pain and /or migraine
US20080033050A1 (en) 2006-08-04 2008-02-07 Richards Patricia Allison Tewe Method of treating thermoregulatory disfunction with paroxetine
US8503431B2 (en) * 2006-08-25 2013-08-06 Wireless Wonders Ltd. Mobile phone related indirect communication system and method
DK2134691T3 (da) 2007-03-08 2012-05-07 Janssen Pharmaceutica Nv Quinolinonderivativer som parp- og tank-inhibitorer
JP5017703B2 (ja) * 2007-05-16 2012-09-05 住友ゴム工業株式会社 ビードエイペックスおよびタイヤ
US8404713B2 (en) 2007-10-26 2013-03-26 Janssen Pharmaceutica Nv Quinolinone derivatives as PARP inhibitors
AU2009228943B2 (en) 2008-03-27 2013-04-04 Janssen Pharmaceutica Nv Tetrahydrophenanthridinones and tetrahydrocyclopentaquinolinones as PARP and tubulin polymerization inhibitors
ES2367760T3 (es) 2008-03-27 2011-11-08 Janssen Pharmaceutica, N.V. Derivados de quinazolinona como inhibidores de la polimerización de la tubulina.
UA112679C2 (uk) 2012-02-24 2016-10-10 Люпін Лімітед Заміщені хроманові сполуки як модулятори рецептора, чутливого до кальцію
DE102012206062B4 (de) 2012-04-13 2019-09-12 Adidas Ag Schuhoberteil
US9040533B2 (en) 2012-12-27 2015-05-26 Purdue Pharma L.P. Oxime-substituted-quinoxaline-type piperidine compounds as ORL-1 modulators
DE102013207163B4 (de) 2013-04-19 2022-09-22 Adidas Ag Schuhoberteil
DE102014220087B4 (de) 2014-10-02 2016-05-12 Adidas Ag Flachgestricktes Schuhoberteil für Sportschuhe
CN108713021A (zh) 2015-12-30 2018-10-26 耶路撒冷希伯来大学伊森姆研究发展有限公司 Pt(IV)前药
CN119462701A (zh) * 2024-10-11 2025-02-18 合肥工业大学 一种四吡啶草酸铜金属配合物的制备及用途

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DE3901814A1 (de) * 1988-07-28 1990-02-01 Bayer Ag Substituierte aminomethylzetraline sowie ihre heterocyclischen analoga
DE4140540A1 (de) * 1991-12-09 1993-06-17 Bayer Ag Neue azaheterocyclylmethyl-chromane
SI9300097B (en) * 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
DE4319038A1 (de) * 1993-06-08 1994-12-15 Bayer Ag Verwendung von teilweise bekannten substituierten Chromanen als Arzneimittel, neue Wirkstoffe und Verfahren zu ihrer Herstellung
WO1995005383A1 (en) * 1993-08-19 1995-02-23 Janssen Pharmaceutica N.V. Vasocontrictive dihydrobenzopyran derivatives
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Also Published As

Publication number Publication date
SK8032000A3 (en) 2001-02-12
IL136529A (en) 2003-03-12
HU224813B1 (en) 2006-02-28
JP2001525407A (ja) 2001-12-11
DE69835372D1 (de) 2006-09-07
US20030149093A1 (en) 2003-08-07
UA70308C2 (uk) 2004-10-15
BG104372A (en) 2000-12-29
US6747045B2 (en) 2004-06-08
WO1999029687A1 (en) 1999-06-17
US6852714B2 (en) 2005-02-08
CA2311669C (en) 2010-04-27
CZ297895B6 (cs) 2007-04-25
US6133277A (en) 2000-10-17
EA003365B1 (ru) 2003-04-24
CN1155597C (zh) 2004-06-30
WO1999029687A8 (en) 2000-04-13
ZA9811081B (en) 2000-06-22
AR017195A1 (es) 2001-08-22
HUP0004492A2 (hu) 2002-03-28
EE04438B1 (et) 2005-02-15
EP1036073B1 (en) 2006-07-26
US6495547B1 (en) 2002-12-17
ATE334125T1 (de) 2006-08-15
ID24616A (id) 2000-07-27
HRP20000340B1 (hr) 2008-12-31
KR100591605B1 (ko) 2006-06-20
ES2270541T3 (es) 2007-04-01
US20030083365A1 (en) 2003-05-01
AU2412799A (en) 1999-06-28
CA2311669A1 (en) 1999-06-17
EA200000616A1 (ru) 2000-12-25
NO20002074D0 (no) 2000-04-19
BR9814256A (pt) 2000-10-03
HRP20000340A2 (en) 2001-04-30
DE69835372T2 (de) 2007-08-09
KR20010031010A (ko) 2001-04-16
NO20002074L (no) 2000-06-02
PL191144B1 (pl) 2006-03-31
BG64624B1 (bg) 2005-09-30
HUP0004492A3 (en) 2002-04-29
EP1036073A1 (en) 2000-09-20
NZ503603A (en) 2001-10-26
IL136529A0 (en) 2001-06-14
PL341007A1 (en) 2001-03-12
MY124586A (en) 2006-06-30
AU748669B2 (en) 2002-06-06
EP1036073B8 (en) 2006-11-15
HK1028400A1 (en) 2001-02-16
CO5011114A1 (es) 2001-02-28
TW577886B (en) 2004-03-01
CZ20002018A3 (cs) 2000-10-11
SK286268B6 (sk) 2008-06-06
CN1280577A (zh) 2001-01-17
NO320727B1 (no) 2006-01-23
TR200001542T2 (tr) 2001-01-22

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