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DK2938194T3 - N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater - Google Patents

N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater Download PDF

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Publication number
DK2938194T3
DK2938194T3 DK13868013.7T DK13868013T DK2938194T3 DK 2938194 T3 DK2938194 T3 DK 2938194T3 DK 13868013 T DK13868013 T DK 13868013T DK 2938194 T3 DK2938194 T3 DK 2938194T3
Authority
DK
Denmark
Prior art keywords
dihydropyrimidine
fluor
imino
oxo
substituted
Prior art date
Application number
DK13868013.7T
Other languages
English (en)
Inventor
Beth Lorsbach
W John Owen
Chenglin Yao
Lindsay Stelzer
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Application granted granted Critical
Publication of DK2938194T3 publication Critical patent/DK2938194T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22O-Aryl or S-Aryl esters thereof
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK13868013.7T 2012-12-28 2013-12-23 N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater DK2938194T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261747086P 2012-12-28 2012-12-28
PCT/US2013/077540 WO2014105844A1 (en) 2012-12-28 2013-12-23 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives

Publications (1)

Publication Number Publication Date
DK2938194T3 true DK2938194T3 (da) 2020-01-02

Family

ID=51022033

Family Applications (1)

Application Number Title Priority Date Filing Date
DK13868013.7T DK2938194T3 (da) 2012-12-28 2013-12-23 N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater

Country Status (18)

Country Link
US (2) US9622474B2 (da)
EP (1) EP2938194B1 (da)
JP (1) JP6324994B2 (da)
KR (1) KR20150103096A (da)
CN (2) CN110003118A (da)
AU (1) AU2013370493B2 (da)
BR (1) BR102013033709B1 (da)
CA (1) CA2893778A1 (da)
CR (1) CR20150382A (da)
DK (1) DK2938194T3 (da)
EC (1) ECSP15032859A (da)
HU (1) HUE047711T2 (da)
IL (1) IL239561B (da)
MX (1) MX2015008441A (da)
PL (1) PL2938194T3 (da)
RU (1) RU2638556C2 (da)
UA (1) UA115462C2 (da)
WO (1) WO2014105844A1 (da)

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CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
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KR102805798B1 (ko) 2014-12-30 2025-05-15 코르테바 애그리사이언스 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
KR20210136961A (ko) 2018-11-05 2021-11-17 아다마 마켓심 리미티드 5-플루오로-4-이미노-3-메틸-1-토실-3,4-디하이드로피리미딘-2-온을 포함하는 혼합물들과 조성물들 및 이들을 사용하는 방법들
CN114599639A (zh) 2019-09-23 2022-06-07 阿达玛马克西姆有限公司 用于制备5-(氟-4-亚氨基-3-甲基)-1-甲苯磺酰基-3,4-二氢嘧啶-(1h)-酮的方法

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DK2938194T3 (da) 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
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CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
WO2015103144A1 (en) 2013-12-31 2015-07-09 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
MA41272A (fr) 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences

Also Published As

Publication number Publication date
MX2015008441A (es) 2015-09-23
US9908855B2 (en) 2018-03-06
EP2938194A4 (en) 2016-08-31
CA2893778A1 (en) 2014-07-03
UA115462C2 (uk) 2017-11-10
KR20150103096A (ko) 2015-09-09
JP2016507512A (ja) 2016-03-10
BR102013033709B1 (pt) 2019-05-14
RU2638556C2 (ru) 2017-12-14
BR102013033709A2 (pt) 2015-10-06
CN104902757A (zh) 2015-09-09
AU2013370493A1 (en) 2015-07-02
AU2013370493B2 (en) 2017-08-17
ECSP15032859A (es) 2015-11-30
US20170204069A1 (en) 2017-07-20
PL2938194T3 (pl) 2020-09-21
HK1214475A1 (en) 2016-07-29
EP2938194A1 (en) 2015-11-04
HUE047711T2 (hu) 2020-05-28
EP2938194B1 (en) 2019-11-27
JP6324994B2 (ja) 2018-05-16
RU2015131095A (ru) 2017-02-06
CR20150382A (es) 2015-08-21
US9622474B2 (en) 2017-04-18
CN104902757B (zh) 2019-01-08
IL239561A0 (en) 2015-08-31
IL239561B (en) 2018-01-31
US20160192653A1 (en) 2016-07-07
CN110003118A (zh) 2019-07-12
WO2014105844A1 (en) 2014-07-03

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