ECSP11011211A - Tratamiento de atrofia vaginal en mujeres con riesgo de patología cardiovascular - Google Patents
Tratamiento de atrofia vaginal en mujeres con riesgo de patología cardiovascularInfo
- Publication number
- ECSP11011211A ECSP11011211A EC2011011211A ECSP11011211A ECSP11011211A EC SP11011211 A ECSP11011211 A EC SP11011211A EC 2011011211 A EC2011011211 A EC 2011011211A EC SP11011211 A ECSP11011211 A EC SP11011211A EC SP11011211 A ECSP11011211 A EC SP11011211A
- Authority
- EC
- Ecuador
- Prior art keywords
- women
- treatment
- cardiovascular pathology
- risk
- vaginal atrophy
- Prior art date
Links
- 230000002526 effect on cardiovascular system Effects 0.000 title abstract 3
- 230000007170 pathology Effects 0.000 title abstract 3
- 206010003694 Atrophy Diseases 0.000 title 1
- 230000037444 atrophy Effects 0.000 title 1
- PROQIPRRNZUXQM-UHFFFAOYSA-N (16alpha,17betaOH)-Estra-1,3,5(10)-triene-3,16,17-triol Natural products OC1=CC=C2C3CCC(C)(C(C(O)C4)O)C4C3CCC2=C1 PROQIPRRNZUXQM-UHFFFAOYSA-N 0.000 abstract 2
- PROQIPRRNZUXQM-ZXXIGWHRSA-N estriol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H]([C@H](O)C4)O)[C@@H]4[C@@H]3CCC2=C1 PROQIPRRNZUXQM-ZXXIGWHRSA-N 0.000 abstract 2
- 229960001348 estriol Drugs 0.000 abstract 2
- 206010071018 Urogenital atrophy Diseases 0.000 abstract 1
- 238000010521 absorption reaction Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Inorganic Chemistry (AREA)
- Urology & Nephrology (AREA)
- Pregnancy & Childbirth (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
Abstract
La presente invención se refiere al uso de estriol en la preparación de una formulación farmacéutica para administración vaginal con la capacidad de autolimitar la absorción de estriol, para la prevención y/o el tratamiento de atrofia urogenital en mujeres, teniendo dichas mujeres una probabilidad elevada de padecer una patología cardiovascular o que padecen o han padecido una patología cardiovascular.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES200803623A ES2344675B1 (es) | 2008-12-19 | 2008-12-19 | Uso de estriol en la preparacion de una formulacion farrmaceutica para el tratamiento de atrofia vaginal en mujeres con riesgo de patologiacardiovascular. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP11011211A true ECSP11011211A (es) | 2011-08-31 |
Family
ID=41050933
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2011011211A ECSP11011211A (es) | 2008-12-19 | 2011-07-15 | Tratamiento de atrofia vaginal en mujeres con riesgo de patología cardiovascular |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US8835414B2 (es) |
| EP (1) | EP2376086B1 (es) |
| JP (1) | JP2012512818A (es) |
| KR (1) | KR101734380B1 (es) |
| CN (1) | CN102325533A (es) |
| CA (1) | CA2747314C (es) |
| CL (1) | CL2011001493A1 (es) |
| CO (1) | CO6382128A2 (es) |
| CY (1) | CY1120971T1 (es) |
| DK (1) | DK2376086T3 (es) |
| EC (1) | ECSP11011211A (es) |
| ES (2) | ES2344675B1 (es) |
| HR (1) | HRP20182022T1 (es) |
| HU (1) | HUE040394T2 (es) |
| LT (1) | LT2376086T (es) |
| MA (1) | MA32984B1 (es) |
| MX (1) | MX2011006696A (es) |
| PE (1) | PE20120496A1 (es) |
| PL (1) | PL2376086T3 (es) |
| PT (1) | PT2376086T (es) |
| RU (1) | RU2555752C2 (es) |
| SI (1) | SI2376086T1 (es) |
| SM (1) | SMT201800648T1 (es) |
| WO (1) | WO2010069621A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11246934B2 (en) * | 2015-01-05 | 2022-02-15 | B.G. Negev Technologies & Applications Ltd. At Ben-Gurion University | Nanoparticles and methods for preparation thereof |
Family Cites Families (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1866M (fr) | 1961-04-07 | 1963-06-17 | Vismara Francesco Spa | Nouveaux éthers des hormones oestrogenes. |
| WO1985002092A1 (en) | 1983-11-14 | 1985-05-23 | Bio-Mimetics Inc. | Bioadhesive compositions and methods of treatment therewith |
| US5719197A (en) | 1988-03-04 | 1998-02-17 | Noven Pharmaceuticals, Inc. | Compositions and methods for topical administration of pharmaceutically active agents |
| ES2050096T3 (es) | 1989-10-31 | 1995-01-16 | Columbia Lab Inc | Composicion humidificante del tejido vaginal. |
| FI913127A0 (fi) | 1989-10-31 | 1991-06-27 | Watson Lab | Vid slemhinnan haeftade stoedsystem foer frigoerande av ett terapeutiskt aemne. |
| US5340586A (en) * | 1991-04-12 | 1994-08-23 | University Of Southern California | Methods and formulations for use in treating oophorectomized women |
| US5543150A (en) | 1993-09-15 | 1996-08-06 | Columbia Laboratories, Inc. | Method of progesterone delivery and affect thereof |
| US5667492A (en) | 1994-10-07 | 1997-09-16 | Columbia Laboratories, Inc. | Use and composition of an anti-sexually transmitted diseases formulation |
| AT408067B (de) | 1995-03-17 | 2001-08-27 | Gebro Pharma Gmbh | Pharmazeutische zusammensetzung zur topischen applizierung und verfahren zu ihrer herstellung |
| US5741525A (en) | 1995-10-24 | 1998-04-21 | Marshall University Research Corporation | Vaginal pharmaceutical hydrogen peroxide composition |
| IT1275816B1 (it) | 1995-10-27 | 1997-10-17 | Montefarmaco Spa | Composizioni farmaceutiche solide per uso vaginale |
| AU714797B2 (en) | 1996-06-14 | 2000-01-13 | Mcneil-Ppc, Inc. | Moisture containing compositions that are spreadable onto and adherable to biomembranes, methods of making and use thereof |
| IT1284874B1 (it) | 1996-08-02 | 1998-05-22 | Farmigea Spa | Complessi bioadesivi di polycarbophil e farmaci antifungini o antiprotozoari azolici |
| US5942243A (en) | 1996-11-12 | 1999-08-24 | Polytherapeutics, Inc. | Mucoadhesive compositions for administration of biologically active agents to animal tissue |
| WO1998020872A1 (en) | 1996-11-14 | 1998-05-22 | Halldor Thormar | Topical formulations containing as a therapeutic active agent fatty acids or fatty alcohols or monoglyceride derivatives thereof for treating of mucosa infections |
| DE69819748T2 (de) | 1997-09-12 | 2004-09-30 | Columbia Laboratories (Bermuda) Ltd. | Arzneimittel zur behandlung von dysmenorrhöe und verfrühten wehen |
| US6159491A (en) | 1999-02-12 | 2000-12-12 | Biovector Technologies, Inc. | Prolonged release bioadhesive vaginal gel dosage form |
| ES2350306T3 (es) | 1999-02-26 | 2011-01-20 | Novartis Vaccines And Diagnostics, Inc. | Uso de bioadhesivos y adyuvantes para la administración de antígenos por vía mucosa. |
| UA74168C2 (uk) | 1999-10-05 | 2005-11-15 | Коламбіа Леборетеріс (Бермуда) Лімітед | Лікування ендометріозу або безпліддя, або покращення плідності та застосування бета-адренергічного агоніста для виробництва лікарського засобу |
| EP1267826B1 (en) | 1999-10-22 | 2007-01-03 | Lif-Hlaup Ehf. Bio-Gels Pharmaceuticals Inc. | Pharmaceutical composition for treatment of mucosal epithelial ulceration and/or erosion |
| SI1611892T1 (sl) * | 2000-01-18 | 2010-01-29 | Bayer Schering Pharma Ag | Farmacevtski sestavki, ki obsegajo drospirenon |
| EP1307232B1 (en) | 2000-08-03 | 2007-03-07 | Antares Pharma IPL AG | Novel composition for transdermal and/or transmucosal administration of active compounds that ensures adequate therapeutic levels |
| US20040092494A9 (en) | 2000-08-30 | 2004-05-13 | Dudley Robert E. | Method of increasing testosterone and related steroid concentrations in women |
| JP3655846B2 (ja) | 2001-06-27 | 2005-06-02 | 埼玉日本電気株式会社 | Cdma移動通信システム、及びその呼切断防止方法 |
| ES2237298B1 (es) * | 2003-07-16 | 2006-11-01 | Italfarmaco, S.A. | Formulaciones mucoadhesivas semisolidas. |
| BRPI0614625A2 (pt) | 2005-08-12 | 2011-04-12 | Drugtech Corp | composição farmacêutica que compreende pelo menos um composto estrogênico, sistema de distribuição de estrogênio vaginal, uso de uma composição e kit que compreende uma pluralidade de cremes vaginais |
| US20090124584A1 (en) | 2005-12-16 | 2009-05-14 | Lyle Corporate Development, Inc. | Regeneration of vaginal tissue with non-systemic vaginal administration of estrogen |
| EP1983998A2 (en) * | 2006-01-20 | 2008-10-29 | Pear Tree Pharmaceuticals, Inc. | Method of treating atrophic vaginitis |
| EP1872775A1 (en) * | 2006-06-29 | 2008-01-02 | Polichem S.A. | Use of a hydrophilic matrix comprising a polyacrylic acid derivative, a cellulose ether and a disintegrant for the manufacture of a medicament for treating female genital disorders |
| WO2008089405A1 (en) | 2007-01-19 | 2008-07-24 | Neurosci, Inc. | Composition of multiple hormones delivered vaginally in a single cream |
| ES2310968B1 (es) * | 2007-06-25 | 2010-02-08 | Italfarmaco, S.A. | Uso de estriol en bajas dosis. |
-
2008
- 2008-12-19 ES ES200803623A patent/ES2344675B1/es active Active
-
2009
- 2009-08-07 SM SM20180648T patent/SMT201800648T1/it unknown
- 2009-08-07 RU RU2011127702/15A patent/RU2555752C2/ru active
- 2009-08-07 CA CA2747314A patent/CA2747314C/en active Active
- 2009-08-07 KR KR1020117016748A patent/KR101734380B1/ko active Active
- 2009-08-07 US US13/140,602 patent/US8835414B2/en active Active
- 2009-08-07 MA MA34038A patent/MA32984B1/fr unknown
- 2009-08-07 CN CN2009801571799A patent/CN102325533A/zh active Pending
- 2009-08-07 PL PL09781638T patent/PL2376086T3/pl unknown
- 2009-08-07 LT LTEP09781638.3T patent/LT2376086T/lt unknown
- 2009-08-07 PT PT09781638T patent/PT2376086T/pt unknown
- 2009-08-07 MX MX2011006696A patent/MX2011006696A/es active IP Right Grant
- 2009-08-07 WO PCT/EP2009/060304 patent/WO2010069621A1/en not_active Ceased
- 2009-08-07 SI SI200931909T patent/SI2376086T1/sl unknown
- 2009-08-07 ES ES09781638T patent/ES2707873T3/es active Active
- 2009-08-07 DK DK09781638.3T patent/DK2376086T3/en active
- 2009-08-07 HR HRP20182022TT patent/HRP20182022T1/hr unknown
- 2009-08-07 JP JP2011541240A patent/JP2012512818A/ja active Pending
- 2009-08-07 HU HUE09781638A patent/HUE040394T2/hu unknown
- 2009-08-07 EP EP09781638.3A patent/EP2376086B1/en active Active
- 2009-08-07 PE PE2011001250A patent/PE20120496A1/es not_active Application Discontinuation
-
2011
- 2011-06-17 CL CL2011001493A patent/CL2011001493A1/es unknown
- 2011-07-15 EC EC2011011211A patent/ECSP11011211A/es unknown
- 2011-07-19 CO CO11090537A patent/CO6382128A2/es not_active Application Discontinuation
-
2018
- 2018-12-07 CY CY181101306T patent/CY1120971T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK2376086T3 (en) | 2018-12-10 |
| WO2010069621A1 (en) | 2010-06-24 |
| KR20110108358A (ko) | 2011-10-05 |
| SMT201800648T1 (it) | 2019-01-11 |
| ES2707873T3 (es) | 2019-04-05 |
| PE20120496A1 (es) | 2012-05-04 |
| CN102325533A (zh) | 2012-01-18 |
| LT2376086T (lt) | 2019-01-10 |
| HUE040394T2 (hu) | 2019-03-28 |
| CA2747314C (en) | 2017-04-18 |
| CO6382128A2 (es) | 2012-02-15 |
| RU2555752C2 (ru) | 2015-07-10 |
| MA32984B1 (fr) | 2012-01-02 |
| MX2011006696A (es) | 2011-07-28 |
| CA2747314A1 (en) | 2010-06-24 |
| US8835414B2 (en) | 2014-09-16 |
| KR101734380B1 (ko) | 2017-05-11 |
| PL2376086T3 (pl) | 2019-05-31 |
| EP2376086B1 (en) | 2018-09-19 |
| EP2376086A1 (en) | 2011-10-19 |
| HRP20182022T1 (hr) | 2019-01-25 |
| ES2344675A1 (es) | 2010-09-02 |
| WO2010069621A8 (en) | 2011-07-21 |
| RU2011127702A (ru) | 2013-01-27 |
| SI2376086T1 (sl) | 2019-02-28 |
| PT2376086T (pt) | 2018-12-18 |
| US20110312929A1 (en) | 2011-12-22 |
| CL2011001493A1 (es) | 2012-01-13 |
| ES2344675B1 (es) | 2011-04-28 |
| CY1120971T1 (el) | 2019-12-11 |
| JP2012512818A (ja) | 2012-06-07 |
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