DZ3195A1 - Quinolyl propyl piperidine derivatives and their use as antibacterials. - Google Patents

Quinolyl propyl piperidine derivatives and their use as antibacterials.

Info

Publication number: DZ3195A1
Authority: DZ; Algeria
Prior art keywords: antibacterials; piperidine derivatives; propyl piperidine; quinolyl propyl; quinolyl
Prior art date: 1999-09-17

Application number

DZ003195A

Other languages

French (fr)

Inventor

Jean-Luc Malleron

Michel Carry Jean-Chris Tabart

Michel Evers

Ahmad Youssef El

Serge Mignani

Fabrice Viviani

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-09-17

Filing date

2000-09-14

Publication date

2001-04-12

2000-09-14 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2001-04-12 Application granted granted Critical

2001-04-12 Publication of DZ3195A1 publication Critical patent/DZ3195A1/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

DZ003195A 1999-09-17 2000-09-14 Quinolyl propyl piperidine derivatives and their use as antibacterials. DZ3195A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9911679A FR2798656B1 (en)	1999-09-17	1999-09-17	DERIVATIVES OF QUINOLYL PROPYL PIPERIDINE, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM
PCT/FR2000/002541 WO2001025227A2 (en)	1999-09-17	2000-09-14	Quinolyl propyl piperidine derivatives and their use as antibacterial agents

Publications (1)

Publication Number	Publication Date
DZ3195A1 true DZ3195A1 (en)	2001-04-12

Family

ID=9549990

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DZ003195A DZ3195A1 (en)	1999-09-17	2000-09-14	Quinolyl propyl piperidine derivatives and their use as antibacterials.

Country Status (30)

Country	Link
EP (2)	EP1218370B1 (en)
JP (1)	JP2004527448A (en)
KR (1)	KR20020038757A (en)
CN (1)	CN1374959A (en)
AP (1)	AP2002002459A0 (en)
AT (1)	ATE284399T1 (en)
AU (1)	AU7429500A (en)
BG (1)	BG106524A (en)
BR (1)	BR0014060A (en)
CA (1)	CA2383836A1 (en)
CZ (1)	CZ2002940A3 (en)
DE (2)	DE60016611T2 (en)
DZ (1)	DZ3195A1 (en)
EA (1)	EA005183B1 (en)
EE (1)	EE200200138A (en)
FR (1)	FR2798656B1 (en)
GE (1)	GEP20043223B (en)
HR (1)	HRP20020214A2 (en)
HU (1)	HUP0204283A3 (en)
IL (1)	IL148720A0 (en)
MA (1)	MA26820A1 (en)
MX (1)	MXPA02001979A (en)
NO (1)	NO20021253L (en)
OA (1)	OA12022A (en)
PL (1)	PL354809A1 (en)
SK (1)	SK3632002A3 (en)
TN (1)	TNSN00184A1 (en)
WO (1)	WO2001025227A2 (en)
YU (1)	YU19002A (en)
ZA (1)	ZA200202073B (en)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9822440D0 (en)	1998-10-14	1998-12-09	Smithkline Beecham Plc	Medicaments
GB9917406D0 (en)	1999-07-23	1999-09-22	Smithkline Beecham Plc	Compounds
GB9917408D0 (en)	1999-07-23	1999-09-22	Smithkline Beecham Plc	Compounds
NZ523749A (en)	2000-07-26	2005-03-24	Smithkline Beecham P	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0031086D0 (en) *	2000-12-20	2001-01-31	Smithkline Beecham Plc	Medicaments
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
US7109213B2 (en)	2002-01-29	2006-09-19	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
EP1470125A1 (en)	2002-01-29	2004-10-27	Glaxo Group Limited	Aminopiperidine derivatives
TW200409637A (en)	2002-06-26	2004-06-16	Glaxo Group Ltd	Compounds
AR040335A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND
FR2842807A1 (en)	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
FR2844270B1 (en) *	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
FR2844268B1 (en) *	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
CN101817815A (en) *	2002-10-10	2010-09-01	莫弗凯姆联合化学股份公司	Compounds with antibacterial activity
JP4654035B2 (en)	2002-11-05	2011-03-16	グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー	Antibacterial agent
AU2003303956A1 (en)	2002-11-05	2004-11-23	Smithkline Beecham Corporation	Antibacterial agents
US7491714B2 (en)	2002-12-04	2009-02-17	Glaxo Group Limited	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
EP1799674B1 (en) *	2004-10-05	2010-05-05	Actelion Pharmaceuticals Ltd.	New piperidine antibiotics
CN101039935B (en) *	2004-10-05	2011-04-20	埃科特莱茵药品有限公司	piperidine antibiotic
US7592334B2 (en)	2005-01-25	2009-09-22	Glaxo Group Limited	Antibacterial agents
WO2006081179A1 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
JP2008528598A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
JP2008528586A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
WO2007086016A1 (en)	2006-01-26	2007-08-02	Actelion Pharmaceuticals Ltd	Tetrahydropyrane antibiotics
WO2007115947A1 (en)	2006-04-06	2007-10-18	Glaxo Group Limited	Pyrrolo-quinoxalinone derivatives as antibacterials
GB0613208D0 (en)	2006-07-03	2006-08-09	Glaxo Group Ltd	Compounds
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
WO2008139288A2 (en) *	2007-05-09	2008-11-20	Pfizer Inc.	Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
JP2012505866A (en)	2008-10-17	2012-03-08	グラクソグループリミテッド	Tricyclic nitrogen compounds used as antibacterial agents
US8318940B2 (en)	2009-01-15	2012-11-27	Glaxo Group Limited	Naphthyridin-2 (1 H)-one compounds useful as antibacterials
RU2671496C2 (en) *	2013-10-14	2018-11-01	Эйсай Ар Энд Ди Менеджмент Ко., Лтд.	5-piperidin-8-cyanochinoline derivatives
AU2015304847B2 (en)	2014-08-22	2018-10-25	Glaxosmithkline Intellectual Property Development Limited	Tricyclic nitrogen containing compounds for treating Neisseria gonorrhoea infection
TW201722965A (en)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	Compounds for use in antibacterial applications
UA124802C2 (en)	2015-12-17	2021-11-24	Мерк Патент Гмбх	POLYCYCLIC TLR7 / 8 ANTAGONISTS AND THEIR APPLICATIONS IN THE TREATMENT OF IMMUNE DISORDERS
KR20240019867A (en)	2016-08-08	2024-02-14	메르크 파텐트 게엠베하	Tlr7/8 antagonists and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2717899A (en) *	1998-01-26	1999-08-09	Smithkline Beecham Plc	Quinoline derivatives as antibacterials
JP2002535323A (en) *	1999-01-20	2002-10-22	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	Piperidinylquinoline as a protein kinase inhibitor

1999
- 1999-09-17 FR FR9911679A patent/FR2798656B1/en not_active Expired - Fee Related
2000
- 2000-09-14 GE GEAP20006413A patent/GEP20043223B/en unknown
- 2000-09-14 KR KR1020027003547A patent/KR20020038757A/en not_active Ceased
- 2000-09-14 EA EA200200374A patent/EA005183B1/en not_active IP Right Cessation
- 2000-09-14 CA CA002383836A patent/CA2383836A1/en not_active Abandoned
- 2000-09-14 IL IL14872000A patent/IL148720A0/en unknown
- 2000-09-14 EP EP00962637A patent/EP1218370B1/en not_active Expired - Lifetime
- 2000-09-14 CZ CZ2002940A patent/CZ2002940A3/en unknown
- 2000-09-14 AP APAP/P/2002/002459A patent/AP2002002459A0/en unknown
- 2000-09-14 YU YU19002A patent/YU19002A/en unknown
- 2000-09-14 AU AU74295/00A patent/AU7429500A/en not_active Abandoned
- 2000-09-14 PL PL00354809A patent/PL354809A1/en not_active Application Discontinuation
- 2000-09-14 OA OA1200200074A patent/OA12022A/en unknown
- 2000-09-14 HU HU0204283A patent/HUP0204283A3/en unknown
- 2000-09-14 MX MXPA02001979A patent/MXPA02001979A/en unknown
- 2000-09-14 SK SK363-2002A patent/SK3632002A3/en unknown
- 2000-09-14 DZ DZ003195A patent/DZ3195A1/en active
- 2000-09-14 CN CN00813020A patent/CN1374959A/en active Pending
- 2000-09-14 EE EEP200200138A patent/EE200200138A/en unknown
- 2000-09-14 JP JP2001528171A patent/JP2004527448A/en active Pending
- 2000-09-14 EP EP04019136A patent/EP1484328B1/en not_active Expired - Lifetime
- 2000-09-14 DE DE60016611T patent/DE60016611T2/en not_active Expired - Fee Related
- 2000-09-14 BR BR0014060-0A patent/BR0014060A/en not_active IP Right Cessation
- 2000-09-14 AT AT00962637T patent/ATE284399T1/en not_active IP Right Cessation
- 2000-09-14 WO PCT/FR2000/002541 patent/WO2001025227A2/en not_active Ceased
- 2000-09-14 HR HR20020214A patent/HRP20020214A2/en not_active Application Discontinuation
- 2000-09-14 DE DE60034713T patent/DE60034713T2/en not_active Expired - Fee Related
- 2000-09-15 TN TNTNSN00184A patent/TNSN00184A1/en unknown
2002
- 2002-03-13 ZA ZA200202073A patent/ZA200202073B/en unknown
- 2002-03-13 NO NO20021253A patent/NO20021253L/en not_active Application Discontinuation
- 2002-03-14 MA MA26554A patent/MA26820A1/en unknown
- 2002-03-15 BG BG106524A patent/BG106524A/en unknown

Also Published As

Publication number	Publication date
EP1218370B1 (en)	2004-12-08
GEP20043223B (en)	2004-04-26
FR2798656A1 (en)	2001-03-23
MA26820A1 (en)	2004-12-20
OA12022A (en)	2006-04-19
EE200200138A (en)	2003-06-16
HUP0204283A2 (en)	2003-04-28
HRP20020214A2 (en)	2005-04-30
ATE284399T1 (en)	2004-12-15
MXPA02001979A (en)	2002-08-20
EA005183B1 (en)	2004-12-30
DE60034713T2 (en)	2008-01-17
PL354809A1 (en)	2004-02-23
EP1484328A1 (en)	2004-12-08
WO2001025227A2 (en)	2001-04-12
DE60034713D1 (en)	2007-06-14
SK3632002A3 (en)	2003-04-01
IL148720A0 (en)	2002-09-12
NO20021253L (en)	2002-04-24
KR20020038757A (en)	2002-05-23
DE60016611D1 (en)	2005-01-13
CN1374959A (en)	2002-10-16
NO20021253D0 (en)	2002-03-13
DE60016611T2 (en)	2005-12-22
ZA200202073B (en)	2003-08-27
AU7429500A (en)	2001-05-10
EP1484328B1 (en)	2007-05-02
BG106524A (en)	2003-01-31
EP1218370A2 (en)	2002-07-03
AP2002002459A0 (en)	2002-06-30
CZ2002940A3 (en)	2002-07-17
WO2001025227A3 (en)	2001-11-22
CA2383836A1 (en)	2001-04-12
JP2004527448A (en)	2004-09-09
EA200200374A1 (en)	2002-10-31
BR0014060A (en)	2002-05-21
FR2798656B1 (en)	2004-12-17
HUP0204283A3 (en)	2004-07-28
TNSN00184A1 (en)	2005-11-10
YU19002A (en)	2005-06-10

Publication	Publication Date	Title
DZ3195A1 (en)	2001-04-12	Quinolyl propyl piperidine derivatives and their use as antibacterials.
PT1140935E (en)	2003-10-31	1,2-CYCLISED QUINOLINE DERIVATIVES
DE60019577D1 (en)	2005-05-25	4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUM-AGENT
ATE248812T1 (en)	2003-09-15	ARYLSULFONYLHYDROXAMIC ACID DERIVATIVES
DK1003720T3 (en)	2004-05-10	Aryloxyarylsulfonylaminohydroxamic acid derivatives
DE69930518D1 (en)	2006-05-11	ALKINYL-SUBSTITUTED CHINOLIN-2-ON DERIVATIVES USED AS ANTICROGEN AGENTS
TR200000520A3 (en)	2001-06-21	4-Phenyl-pyridine derivatives.
PT1244641E (en)	2005-08-31	TIAZOLYLAMIDE DERIVATIVES
TR199802289A3 (en)	1999-06-21	Phosphonacid-substituted benzazepinone-n-acetic acid derivatives.
TR199901077A3 (en)	1999-12-21	Pharmaceutical formulations.
PT1097139E (en)	2003-04-30	QUINOLINE DERIVATIVES
PT1187814E (en)	2004-10-29	5-PHENYL-PYRIMIDINE DERIVATIVES
ATE298760T1 (en)	2005-07-15	2-HALO-6-0-SUBSTITUTED KETOLIDE DERIVATIVES
NO20020565D0 (en)	2002-02-05	Interleukin-5-inhibiting 6-azauracil derivatives
IS5730A (en)	2000-11-24	Substituted thiazolo-pyridazine derivatives, pharmaceutical formulations thereof
DE60003072D1 (en)	2003-07-03	THIAZOLIDINDEIDE DERIVATIVES AS ANTIDIBIA
NO307708B1 (en)	2000-05-15	ferrocene derivatives
NO994386D0 (en)	1999-09-10	2-substituted benzoylcycloalkyl-1-carboxylic acid derivatives
DE60012038D1 (en)	2004-08-12	NON-Greasy make-up remover
DE50009678D1 (en)	2005-04-07	PESTICIDENT / PF 1022-221
FI974001L (en)	1999-04-21	New methylenebisphosphonic acid derivatives
DE50005694D1 (en)	2004-04-22	CENTRIFUGE
SE9903645D0 (en)	1999-10-08	safety
SE9903723D0 (en)	1999-10-13	safety
ES1036216Y (en)	1997-12-16	PERFECTED FOLDING STAND.