NO20021253D0 - Quinolyl propyl piperidine derivatives and their use as antibacterial agents - Google Patents

Quinolyl propyl piperidine derivatives and their use as antibacterial agents

Info

Publication number: NO20021253D0
Authority: NO; Norway
Prior art keywords: antibacterial agents; piperidine derivatives; propyl piperidine; quinolyl propyl; quinolyl
Prior art date: 1999-09-17

Application number

NO20021253A

Other languages

Norwegian (no)

Other versions

NO20021253L (en

Inventor

Jean-Luc Malleron

Michel Tabart

Jean-Christophe Carry

Michel Evers

Youssef El Ahmad

Serge Mignani

Fabrice Viviani

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-09-17

Filing date

2002-03-13

Publication date

2002-03-13

2002-03-13 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2002-03-13 Publication of NO20021253D0 publication Critical patent/NO20021253D0/en

2002-04-24 Publication of NO20021253L publication Critical patent/NO20021253L/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

NO20021253A 1999-09-17 2002-03-13 Quinolylpropylpiperidine derivatives and their use as antibacterial agents NO20021253L (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9911679A FR2798656B1 (en)	1999-09-17	1999-09-17	DERIVATIVES OF QUINOLYL PROPYL PIPERIDINE, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM
PCT/FR2000/002541 WO2001025227A2 (en)	1999-09-17	2000-09-14	Quinolyl propyl piperidine derivatives and their use as antibacterial agents

Publications (2)

Publication Number	Publication Date
NO20021253D0 true NO20021253D0 (en)	2002-03-13
NO20021253L NO20021253L (en)	2002-04-24

Family

ID=9549990

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20021253A NO20021253L (en)	1999-09-17	2002-03-13	Quinolylpropylpiperidine derivatives and their use as antibacterial agents

Country Status (30)

Country	Link
EP (2)	EP1218370B1 (en)
JP (1)	JP2004527448A (en)
KR (1)	KR20020038757A (en)
CN (1)	CN1374959A (en)
AP (1)	AP2002002459A0 (en)
AT (1)	ATE284399T1 (en)
AU (1)	AU7429500A (en)
BG (1)	BG106524A (en)
BR (1)	BR0014060A (en)
CA (1)	CA2383836A1 (en)
CZ (1)	CZ2002940A3 (en)
DE (2)	DE60016611T2 (en)
DZ (1)	DZ3195A1 (en)
EA (1)	EA005183B1 (en)
EE (1)	EE200200138A (en)
FR (1)	FR2798656B1 (en)
GE (1)	GEP20043223B (en)
HR (1)	HRP20020214A2 (en)
HU (1)	HUP0204283A3 (en)
IL (1)	IL148720A0 (en)
MA (1)	MA26820A1 (en)
MX (1)	MXPA02001979A (en)
NO (1)	NO20021253L (en)
OA (1)	OA12022A (en)
PL (1)	PL354809A1 (en)
SK (1)	SK3632002A3 (en)
TN (1)	TNSN00184A1 (en)
WO (1)	WO2001025227A2 (en)
YU (1)	YU19002A (en)
ZA (1)	ZA200202073B (en)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9822440D0 (en)	1998-10-14	1998-12-09	Smithkline Beecham Plc	Medicaments
GB9917408D0 (en)	1999-07-23	1999-09-22	Smithkline Beecham Plc	Compounds
GB9917406D0 (en)	1999-07-23	1999-09-22	Smithkline Beecham Plc	Compounds
NZ523749A (en)	2000-07-26	2005-03-24	Smithkline Beecham P	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0031086D0 (en) *	2000-12-20	2001-01-31	Smithkline Beecham Plc	Medicaments
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
EP1470125A1 (en)	2002-01-29	2004-10-27	Glaxo Group Limited	Aminopiperidine derivatives
JP4508650B2 (en)	2002-01-29	2010-07-21	グラクソグループリミテッド	Aminopiperidine compound, process for producing the compound and pharmaceutical composition containing the compound
TW200406413A (en)	2002-06-26	2004-05-01	Glaxo Group Ltd	Compounds
TW200409637A (en)	2002-06-26	2004-06-16	Glaxo Group Ltd	Compounds
FR2842807A1 (en)	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
FR2844268B1 (en)	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
FR2844270B1 (en) *	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
BR0315221A (en) *	2002-10-10	2005-08-23	Morphochem Ag Komb Chemie	Compounds with antibacterial activity
EP1560488B1 (en)	2002-11-05	2010-09-01	Glaxo Group Limited	Antibacterial agents
ATE461928T1 (en)	2002-11-05	2010-04-15	Glaxosmithkline Llc	ANTIBACTERIAL ACTIVE INGREDIENTS
ATE411312T1 (en)	2002-12-04	2008-10-15	Glaxo Group Ltd	QUINOLINES AND NITROGEN-CONTAINING DERIVATIVES THEREOF AND THEIR USE AS ANTIBACTERIAL AGENTS
ES2343127T3 (en) *	2004-10-05	2010-07-23	Actelion Pharmaceuticals Ltd.	NEW ANTIBIOTICS OF PIPERIDINA.
EP1799674B1 (en) *	2004-10-05	2010-05-05	Actelion Pharmaceuticals Ltd.	New piperidine antibiotics
US7592334B2 (en)	2005-01-25	2009-09-22	Glaxo Group Limited	Antibacterial agents
US7648980B2 (en)	2005-01-25	2010-01-19	Glaxo Group Limited	Antibacterial agents
JP2008528598A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
US7709472B2 (en)	2005-01-25	2010-05-04	Glaxo Group Limited	Antibacterial agents
JP2009524643A (en)	2006-01-26	2009-07-02	アクテリオンファーマシューティカルズリミテッド	Tetrahydropyran antibiotics
JP2009532423A (en)	2006-04-06	2009-09-10	グラクソグループリミテッド	Pyrrolo-quinoxalinone derivatives as antibacterial agents
GB0613208D0 (en)	2006-07-03	2006-08-09	Glaxo Group Ltd	Compounds
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
KR20120011093A (en) *	2007-05-09	2012-02-06	화이자 인코포레이티드	Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterial agents
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
EP2352734A1 (en)	2008-10-17	2011-08-10	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
EP2379554B1 (en)	2009-01-15	2015-11-11	Glaxo Group Limited	Naphthyridin-2(1h)-one compounds useful as antibacterials
KR102365952B1 (en) *	2013-10-14	2022-02-22	에자이 알앤드디 매니지먼트 가부시키가이샤	Selectively substituted quinoline compounds
US10702521B2 (en)	2014-08-22	2020-07-07	Glaxosmithkline Intellectual Property Development Limited	Methods for treating neisseria gonorrhoeae infection with substituted 1,2-dihydro-2A,5,8A-triazaacenaphthylene-3,8-diones
TW201722965A (en)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	Compounds for use in antibacterial applications
SI3889145T1 (en)	2015-12-17	2024-05-31	Merck Patent Gmbh	8-cyano-5-piperidino-quinolines as tlr7/8 antagonists and their uses for treating immune disorders
SG11201900947RA (en)	2016-08-08	2019-02-27	Merck Patent Gmbh	Tlr7/8 antagonists and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2717899A (en) *	1998-01-26	1999-08-09	Smithkline Beecham Plc	Quinoline derivatives as antibacterials
WO2000043383A1 (en) *	1999-01-20	2000-07-27	Smithkline Beecham P.L.C.	Piperidinylquinolines as protein tyrosine kinase inhibitors

1999
- 1999-09-17 FR FR9911679A patent/FR2798656B1/en not_active Expired - Fee Related
2000
- 2000-09-14 EE EEP200200138A patent/EE200200138A/en unknown
- 2000-09-14 CZ CZ2002940A patent/CZ2002940A3/en unknown
- 2000-09-14 HR HR20020214A patent/HRP20020214A2/en not_active Application Discontinuation
- 2000-09-14 IL IL14872000A patent/IL148720A0/en unknown
- 2000-09-14 PL PL00354809A patent/PL354809A1/en not_active Application Discontinuation
- 2000-09-14 BR BR0014060-0A patent/BR0014060A/en not_active IP Right Cessation
- 2000-09-14 DE DE60016611T patent/DE60016611T2/en not_active Expired - Fee Related
- 2000-09-14 CA CA002383836A patent/CA2383836A1/en not_active Abandoned
- 2000-09-14 EP EP00962637A patent/EP1218370B1/en not_active Expired - Lifetime
- 2000-09-14 KR KR1020027003547A patent/KR20020038757A/en not_active Ceased
- 2000-09-14 OA OA1200200074A patent/OA12022A/en unknown
- 2000-09-14 DE DE60034713T patent/DE60034713T2/en not_active Expired - Fee Related
- 2000-09-14 EP EP04019136A patent/EP1484328B1/en not_active Expired - Lifetime
- 2000-09-14 CN CN00813020A patent/CN1374959A/en active Pending
- 2000-09-14 MX MXPA02001979A patent/MXPA02001979A/en unknown
- 2000-09-14 SK SK363-2002A patent/SK3632002A3/en unknown
- 2000-09-14 EA EA200200374A patent/EA005183B1/en not_active IP Right Cessation
- 2000-09-14 YU YU19002A patent/YU19002A/en unknown
- 2000-09-14 AU AU74295/00A patent/AU7429500A/en not_active Abandoned
- 2000-09-14 GE GEAP20006413A patent/GEP20043223B/en unknown
- 2000-09-14 AP APAP/P/2002/002459A patent/AP2002002459A0/en unknown
- 2000-09-14 AT AT00962637T patent/ATE284399T1/en not_active IP Right Cessation
- 2000-09-14 DZ DZ003195A patent/DZ3195A1/en active
- 2000-09-14 WO PCT/FR2000/002541 patent/WO2001025227A2/en not_active Ceased
- 2000-09-14 JP JP2001528171A patent/JP2004527448A/en active Pending
- 2000-09-14 HU HU0204283A patent/HUP0204283A3/en unknown
- 2000-09-15 TN TNTNSN00184A patent/TNSN00184A1/en unknown
2002
- 2002-03-13 ZA ZA200202073A patent/ZA200202073B/en unknown
- 2002-03-13 NO NO20021253A patent/NO20021253L/en not_active Application Discontinuation
- 2002-03-14 MA MA26554A patent/MA26820A1/en unknown
- 2002-03-15 BG BG106524A patent/BG106524A/en unknown

Also Published As

Publication number	Publication date
JP2004527448A (en)	2004-09-09
SK3632002A3 (en)	2003-04-01
EP1484328B1 (en)	2007-05-02
WO2001025227A3 (en)	2001-11-22
MXPA02001979A (en)	2002-08-20
FR2798656B1 (en)	2004-12-17
HRP20020214A2 (en)	2005-04-30
EP1484328A1 (en)	2004-12-08
DE60016611T2 (en)	2005-12-22
EP1218370A2 (en)	2002-07-03
ZA200202073B (en)	2003-08-27
ATE284399T1 (en)	2004-12-15
HUP0204283A2 (en)	2003-04-28
DE60034713D1 (en)	2007-06-14
AP2002002459A0 (en)	2002-06-30
EA200200374A1 (en)	2002-10-31
NO20021253L (en)	2002-04-24
YU19002A (en)	2005-06-10
HUP0204283A3 (en)	2004-07-28
MA26820A1 (en)	2004-12-20
AU7429500A (en)	2001-05-10
FR2798656A1 (en)	2001-03-23
BG106524A (en)	2003-01-31
KR20020038757A (en)	2002-05-23
EA005183B1 (en)	2004-12-30
EP1218370B1 (en)	2004-12-08
TNSN00184A1 (en)	2005-11-10
CA2383836A1 (en)	2001-04-12
IL148720A0 (en)	2002-09-12
EE200200138A (en)	2003-06-16
OA12022A (en)	2006-04-19
CZ2002940A3 (en)	2002-07-17
DZ3195A1 (en)	2001-04-12
GEP20043223B (en)	2004-04-26
DE60016611D1 (en)	2005-01-13
WO2001025227A2 (en)	2001-04-12
BR0014060A (en)	2002-05-21
DE60034713T2 (en)	2008-01-17
CN1374959A (en)	2002-10-16
PL354809A1 (en)	2004-02-23

Publication	Publication Date	Title
NO20021253D0 (en)	2002-03-13	Quinolyl propyl piperidine derivatives and their use as antibacterial agents
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NO20014135D0 (en)	2001-08-24	New sulfonamide compounds and their use
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NO20024742L (en)	2002-11-25	Heterocyclic compounds, their preparation and use
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NO20024107L (en)	2002-09-27	Tienopyridine derivatives, their preparation and use
FI112705B (en)	2003-12-31	hinges
DK1330453T3 (en)	2006-08-07	Indolylpiperidine derivatives as antihistamine and anti-allergy agents
DK1200409T3 (en)	2004-06-28	Substituted isoquinoline derivatives and their use as anticonvulsants
NO20001782L (en)	2000-10-09	3-Amino-3-arylpropan-1-ol derivatives, their preparation and use

Legal Events

Date	Code	Title	Description
2006-03-13	FC2A	Withdrawal, rejection or dismissal of laid open patent application