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DZ3055A1 - Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant. - Google Patents

Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant.

Info

Publication number
DZ3055A1
DZ3055A1 DZ000113A DZ000113A DZ3055A1 DZ 3055 A1 DZ3055 A1 DZ 3055A1 DZ 000113 A DZ000113 A DZ 000113A DZ 000113 A DZ000113 A DZ 000113A DZ 3055 A1 DZ3055 A1 DZ 3055A1
Authority
DZ
Algeria
Prior art keywords
polymorphs
bicyclo
oct
pharmaceutical compositions
compositions containing
Prior art date
Application number
DZ000113A
Other languages
English (en)
Inventor
Douglas John Meldrum Allen
Troy Anthony Appleton
Michael John Gumkoswki
David Joseph Muehlbauer
Timothy Norris
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DZ3055A1 publication Critical patent/DZ3055A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D455/00Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/02Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DZ000113A 1999-06-22 2000-06-21 Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant. DZ3055A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14023399P 1999-06-22 1999-06-22

Publications (1)

Publication Number Publication Date
DZ3055A1 true DZ3055A1 (fr) 2004-03-27

Family

ID=22490317

Family Applications (1)

Application Number Title Priority Date Filing Date
DZ000113A DZ3055A1 (fr) 1999-06-22 2000-06-21 Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant.

Country Status (35)

Country Link
US (1) US6262067B1 (fr)
EP (1) EP1187834A1 (fr)
JP (1) JP2003502425A (fr)
KR (1) KR20020030280A (fr)
CN (1) CN1390216A (fr)
AP (1) AP2001002367A0 (fr)
AR (1) AR024411A1 (fr)
AU (1) AU767336B2 (fr)
BG (1) BG106205A (fr)
BR (1) BR0011835A (fr)
CA (1) CA2375265A1 (fr)
CO (1) CO5190663A1 (fr)
CZ (1) CZ20014458A3 (fr)
DZ (1) DZ3055A1 (fr)
EA (1) EA004264B1 (fr)
EC (1) ECSP003538A (fr)
EE (1) EE200100698A (fr)
HR (1) HRP20010920A2 (fr)
HU (1) HUP0201694A3 (fr)
IL (1) IL146410A0 (fr)
IS (1) IS6161A (fr)
MA (1) MA26744A1 (fr)
MX (1) MXPA02000033A (fr)
NO (1) NO20016187D0 (fr)
NZ (1) NZ515348A (fr)
OA (1) OA11952A (fr)
PA (1) PA8496701A1 (fr)
PE (1) PE20010322A1 (fr)
PL (1) PL352899A1 (fr)
SK (1) SK18672001A3 (fr)
TN (1) TNSN00137A1 (fr)
TR (1) TR200103688T2 (fr)
UY (1) UY26211A1 (fr)
WO (1) WO2000078759A1 (fr)
ZA (1) ZA200110387B (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6387925B1 (en) * 1999-06-01 2002-05-14 Pfizer Inc. Polymorphs of a crystalline azo-bicyclo (2.2.2) oct-3-yl amine citrate and their pharmaceutical compositions
US6939873B2 (en) 2000-07-26 2005-09-06 Taro Pharmaceuticals Industries Limited Non-sedating barbituric acid derivatives
US6756379B2 (en) * 2001-07-26 2004-06-29 Taro Pharmaceutical Industries Ltd. Non-sedating barbiturate compounds as neuroprotective agents
US7683071B2 (en) * 2000-07-26 2010-03-23 Taro Pharmaceuticals Industries Ltd. Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
JP2006503859A (ja) * 2002-10-04 2006-02-02 メルク シャープ エンド ドーム リミテッド 受容体拮抗薬としてのアザ二環式スピロエーテル誘導体
EP2156839A1 (fr) 2002-12-11 2010-02-24 Taro Pharmaceutical Industries Ltd. Methode de traitement de troubles moteurs a l' aide de derives de l' acide barbiturique.
WO2006003651A2 (fr) * 2004-07-02 2006-01-12 Taro Pharmaceutical Industries, Ltd Procede de preparation d'acide 1-methoxymethyl-5,5-diphenylbarbiturique
WO2008066704A2 (fr) * 2006-11-14 2008-06-05 Taro Pharmaceuticals North America, Inc. Procédé d'amélioration de la biodisponibilité pour les barbituriques non sédatifs
UA102128C2 (en) * 2008-12-05 2013-06-10 Х. Луннбек А/С Nalmefene hydrochloride dihydrate
TWI866977B (zh) * 2019-06-03 2024-12-21 以色列商以色列耶路撒冷希伯來大學伊索研究發展有限公司 吡唑化合物之非吸濕性結晶鹽及其醫藥組合物及用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990005525A1 (fr) * 1988-11-23 1990-05-31 Pfizer Inc. Derives de quinuclidine en tant qu'antagonsites de substance p
SK278788B6 (sk) * 1991-05-31 1998-02-04 Pfizer Inc. Chinuklidínové deriváty, spôsob ich prípravy a pou
KR950704311A (ko) * 1992-11-12 1995-11-17 알렌 제이. 스피겔 물질 p 길항체로서의 퀴누클리딘 유도체(quinuclidine derivative as substance p antagonist)
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis

Also Published As

Publication number Publication date
TNSN00137A1 (fr) 2002-05-30
EA004264B1 (ru) 2004-02-26
EA200101179A1 (ru) 2002-06-27
WO2000078759A1 (fr) 2000-12-28
HUP0201694A2 (en) 2002-09-28
AU4774500A (en) 2001-01-09
PL352899A1 (en) 2003-09-22
CZ20014458A3 (cs) 2002-03-13
NZ515348A (en) 2003-07-25
BG106205A (bg) 2002-07-31
UY26211A1 (es) 2001-01-31
HRP20010920A2 (en) 2003-02-28
IL146410A0 (en) 2002-07-25
SK18672001A3 (sk) 2002-08-06
US6262067B1 (en) 2001-07-17
JP2003502425A (ja) 2003-01-21
IS6161A (is) 2001-11-13
MXPA02000033A (es) 2002-07-02
OA11952A (en) 2006-04-13
CA2375265A1 (fr) 2000-12-28
EE200100698A (et) 2003-02-17
AR024411A1 (es) 2002-10-02
HUP0201694A3 (en) 2002-10-28
CO5190663A1 (es) 2002-08-29
PA8496701A1 (es) 2002-07-30
TR200103688T2 (tr) 2002-12-23
NO20016187L (no) 2001-12-18
CN1390216A (zh) 2003-01-08
AU767336B2 (en) 2003-11-06
ECSP003538A (es) 2002-01-25
EP1187834A1 (fr) 2002-03-20
BR0011835A (pt) 2002-03-05
KR20020030280A (ko) 2002-04-24
AP2001002367A0 (en) 2001-12-31
MA26744A1 (fr) 2004-12-20
PE20010322A1 (es) 2001-03-14
NO20016187D0 (no) 2001-12-18
ZA200110387B (en) 2002-12-19

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