DK400984D0 - Pyrimido(4-5-g)quinolin-derivater, fremgangsmaade til fremstilling hraf og mellemprodukt til brug ved fremgangsmaaden - Google Patents

Pyrimido(4-5-g)quinolin-derivater, fremgangsmaade til fremstilling hraf og mellemprodukt til brug ved fremgangsmaaden

Info

Publication number: DK400984D0
Authority: DK; Denmark
Prior art keywords: procedure; pyrimido; preparation; quinoline derivatives; quinoline
Prior art date: 1983-09-26

Application number

DK400984A

Other languages

English (en)

Other versions

DK164867B (da

DK164867C (da

DK400984A (da

Inventor

Cynthia Lynn Nichols

Edmund Carl Kornfeld

Mark Mortensen Foreman

John Mehnert Schaus

Diane Lynn Huser

Richard Nolan Booher

David Taiwai Wong

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-09-26

Filing date

1984-08-22

Publication date

1984-08-22

1983-09-26 Priority claimed from US06/535,474 external-priority patent/US4521421A/en

1983-09-26 Priority claimed from US06/535,503 external-priority patent/US4501890A/en

1984-01-30 Priority claimed from US06/575,126 external-priority patent/US4528290A/en

1984-08-22 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1984-08-22 Publication of DK400984D0 publication Critical patent/DK400984D0/da

1985-03-27 Publication of DK400984A publication Critical patent/DK400984A/da

1992-08-31 Publication of DK164867B publication Critical patent/DK164867B/da

1993-11-08 Application granted granted Critical

1993-11-08 Publication of DK164867C publication Critical patent/DK164867C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/10—Spiro-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK400984A 1983-09-26 1984-08-22 Pyrimidooe4,5-gaaquinolin-derivater eller salte deraf og farmaceutiske formuleringer indeholdende disse DK164867C (da)

Applications Claiming Priority (10)

Application Number	Priority Date	Filing Date	Title
US53551983A	1983-09-26	1983-09-26
US53547483		1983-09-26
US06/535,474 US4521421A (en)	1983-09-26	1983-09-26	Treatment of sexual dysfunction
US53551983		1983-09-26
US53550383		1983-09-26
US06/535,503 US4501890A (en)	1983-09-26	1983-09-26	Trans-(±)-2,4,6-substituted-5,5a,6,7,8,9,9a,10-octahydro-pyrimido[4,5-g]quinolines
US06/575,126 US4528290A (en)	1984-01-30	1984-01-30	Stimulating dopamine D-1 receptors
US57512684		1984-01-30
US60609184A	1984-05-02	1984-05-02
US60609184		1984-05-02

Publications (4)

Publication Number	Publication Date
DK400984D0 true DK400984D0 (da)	1984-08-22
DK400984A DK400984A (da)	1985-03-27
DK164867B DK164867B (da)	1992-08-31
DK164867C DK164867C (da)	1993-11-08

Family

ID=27541855

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
DK400984A DK164867C (da)	1983-09-26	1984-08-22	Pyrimidooe4,5-gaaquinolin-derivater eller salte deraf og farmaceutiske formuleringer indeholdende disse
DK296390A DK169948B1 (da)	1983-09-26	1990-12-13	Mellemprodukter til brug ved fremstilling af pyrimido[4,5-g]quinolin-derivater eller salte deraf
DK296290A DK169970B1 (da)	1983-09-26	1990-12-13	Mellemprodukter til brug ved fremstilling af pyrimido[4,5-g]quinolin-derivater eller salte deraf
DK296190A DK169622B1 (da)	1983-09-26	1990-12-13	Trans-(+)-stereoisomere af pyrimido[4,5-g]quinolin-derivater eller farmaceutisk acceptable syreadditionssalte deraf samt farmaceutiske formuleringer indeholdende sådanne forbindelser

Family Applications After (3)

Application Number	Title	Priority Date	Filing Date
DK296390A DK169948B1 (da)	1983-09-26	1990-12-13	Mellemprodukter til brug ved fremstilling af pyrimido[4,5-g]quinolin-derivater eller salte deraf
DK296290A DK169970B1 (da)	1983-09-26	1990-12-13	Mellemprodukter til brug ved fremstilling af pyrimido[4,5-g]quinolin-derivater eller salte deraf
DK296190A DK169622B1 (da)	1983-09-26	1990-12-13	Trans-(+)-stereoisomere af pyrimido[4,5-g]quinolin-derivater eller farmaceutisk acceptable syreadditionssalte deraf samt farmaceutiske formuleringer indeholdende sådanne forbindelser

Country Status (16)

Country	Link
EP (1)	EP0139393B1 (da)
JP (1)	JPH01151581A (da)
AU (2)	AU569539B2 (da)
CY (1)	CY1495A (da)
DE (1)	DE3484583D1 (da)
DK (4)	DK164867C (da)
FI (1)	FI78091C (da)
GB (1)	GB2146985B (da)
GR (1)	GR80201B (da)
HK (1)	HK98789A (da)
IE (1)	IE57848B1 (da)
IL (1)	IL72730A (da)
NZ (1)	NZ209295A (da)
PT (1)	PT79112B (da)
RO (1)	RO89126A (da)
SG (1)	SG46389G (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT80898B (pt) *	1984-08-03	1987-12-30	Lilly Co Eli	Processo para a preparacao de derivados triciclicos de quinolina
US4764609A (en) *	1986-03-31	1988-08-16	Eli Lilly And Company	Synthesis of 2-aminopyrimido[4,5-g]quinolines
US4826986A (en) *	1986-06-16	1989-05-02	Eli Lilly And Company	6-Oxo-trans-octa- and decahydroquinolines
US4762843A (en) *	1986-09-15	1988-08-09	Warner-Lambert Company	Hetero [f] fused carbocyclic pyridines as dopaminergic agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4198415A (en) *	1979-01-22	1980-04-15	Eli Lilly And Company	Prolactin inhibiting octahydro pyrazolo[3,4-g]quinolines
JPS59202892A (ja) *	1983-05-04	1984-11-16	Ricoh Co Ltd	光学的情報記録媒体
US4507478A (en) *	1983-09-26	1985-03-26	Eli Lilly And Company	2-Mercaptopyrimidohexahydroquinolines and related compounds
PT80898B (pt) *	1984-08-03	1987-12-30	Lilly Co Eli	Processo para a preparacao de derivados triciclicos de quinolina

1984
- 1984-08-20 RO RO84115536A patent/RO89126A/ro unknown
- 1984-08-20 IL IL72730A patent/IL72730A/xx not_active IP Right Cessation
- 1984-08-20 FI FI843282A patent/FI78091C/fi not_active IP Right Cessation
- 1984-08-21 EP EP84305684A patent/EP0139393B1/en not_active Expired - Lifetime
- 1984-08-21 NZ NZ209295A patent/NZ209295A/en unknown
- 1984-08-21 GB GB08421160A patent/GB2146985B/en not_active Expired
- 1984-08-21 CY CY1495A patent/CY1495A/en unknown
- 1984-08-21 DE DE8484305684T patent/DE3484583D1/de not_active Expired - Lifetime
- 1984-08-22 PT PT79112A patent/PT79112B/pt not_active IP Right Cessation
- 1984-08-22 AU AU32280/84A patent/AU569539B2/en not_active Ceased
- 1984-08-22 IE IE2154/84A patent/IE57848B1/en not_active IP Right Cessation
- 1984-08-22 DK DK400984A patent/DK164867C/da not_active IP Right Cessation
- 1984-08-23 GR GR80201A patent/GR80201B/el unknown
1987
- 1987-12-07 AU AU82168/87A patent/AU585473B2/en not_active Ceased
1988
- 1988-11-15 JP JP63289902A patent/JPH01151581A/ja active Granted
1989
- 1989-07-28 SG SG46389A patent/SG46389G/en unknown
- 1989-12-14 HK HK987/89A patent/HK98789A/xx not_active IP Right Cessation
1990
- 1990-12-13 DK DK296390A patent/DK169948B1/da not_active IP Right Cessation
- 1990-12-13 DK DK296290A patent/DK169970B1/da not_active IP Right Cessation
- 1990-12-13 DK DK296190A patent/DK169622B1/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
RO89126A (ro)	1986-04-30
IE842154L (en)	1985-03-26
DK296390A (da)	1990-12-13
DK169948B1 (da)	1995-04-10
NZ209295A (en)	1987-05-29
PT79112A (en)	1984-09-01
EP0139393A2 (en)	1985-05-02
GR80201B (en)	1985-01-02
IL72730A0 (en)	1984-11-30
GB2146985A (en)	1985-05-01
GB8421160D0 (en)	1984-09-26
DK296190D0 (da)	1990-12-13
AU8216887A (en)	1988-03-31
FI843282A7 (fi)	1985-03-27
IL72730A (en)	1987-10-30
AU3228084A (en)	1985-04-04
DK296290D0 (da)	1990-12-13
HK98789A (en)	1989-12-22
DK164867B (da)	1992-08-31
DK296190A (da)	1990-12-13
EP0139393A3 (en)	1988-01-13
DK296390D0 (da)	1990-12-13
DK296290A (da)	1990-12-13
DE3484583D1 (de)	1991-06-20
DK164867C (da)	1993-11-08
IE57848B1 (en)	1993-04-21
FI78091C (fi)	1989-06-12
GB2146985B (en)	1987-05-28
FI78091B (fi)	1989-02-28
CY1495A (en)	1990-02-16
EP0139393B1 (en)	1991-05-15
DK169622B1 (da)	1994-12-27
FI843282A0 (fi)	1984-08-20
AU569539B2 (en)	1988-02-04
SG46389G (en)	1989-12-22
DK169970B1 (da)	1995-04-18
JPH01151581A (ja)	1989-06-14
AU585473B2 (en)	1989-06-15
PT79112B (en)	1986-11-14
JPH0529398B2 (da)	1993-04-30
DK400984A (da)	1985-03-27

Publication	Publication Date	Title
IL73159A (en)	1990-08-31	Carboxyalkenamido-cephalosporins,processes for the preparation thereof and methods for the use thereof
NO864681D0 (no)	1986-11-21	Fremgangsmaate ved direkte genoverfoering i plastider og mitokondrier.
DK441184A (da)	1985-03-18	Pyrethroid-holdige formlegemer, deres fremstilling og anvendelse
DK457581A (da)	1982-04-18	4,5-polymethylen-4-isothiazolin-3-oner fremgangsmaade til deres fremstilling og deres anvendelse
FI842459A7 (fi)	1984-12-21	Tetrahydropyridatsinonijohdannaisia, menetelmiä niiden valmistamiseksi sekä niiden käyttö.
NO853120L (no)	1986-02-10	Isfjell og fremgangsmaate for fremstilling av samme.
NO843514L (no)	1985-04-18	Plasmastraale-renseapparat og fremgangsmaate ved anvendelse av samme
DK227884A (da)	1984-11-10	1-pyrimidinyloxy-3-hetarylalkylamino-2-propanoler, deres fremstilling og anvendelse
EP0146866A3 (en)	1987-05-13	Phenylsulfonephthaleinyl-beta-d-galactosides, methods for their preparation and their use in the determination of beta-d-galactosidase
DK594884A (da)	1985-06-14	Tvaerbundne polymerisater, deres fremstilling og anvendelse
DK527784A (da)	1985-05-08	Cyanopyrazol-forbindelser, deres fremstilling og anvendelse i herbicider
ZA849958B (en)	1985-08-28	Ortho-condensed pyrrole derivatives and their use
DK85084D0 (da)	1984-02-21	Immunglobulin-producerende hybridcellelinier, deres anvendelse og fremgangsmade til deres fremstilling
DE3477642D1 (en)	1989-05-18	Pulmonary surfactant, process for its preparation and its pharmaceutical use
NO822796L (no)	1983-03-04	Aminoorganoaminosilaner, fremgangsmaate til deres fremstilling og deres anvendelse
ZA83592B (en)	1983-11-30	Corynantheine derivatives,processes for their preparation,and their use
DK306184D0 (da)	1984-06-22	Guaninforbindelse, fremgangsmaade til fremstilling deraf og mellemprodukt til brug ved udoevelse af fremgangsmaaden
NO159346C (no)	1988-12-21	Ski og fremgangsmaate ved deres fremstilling.
NO165421C (no)	1991-02-13	Fremgangsmaate og anordning for avskinning.
DK586383D0 (da)	1983-12-20	Substituerede imidazo (1,5-a)pyridiner samt deres fremstilling og anvendelse
DK400984D0 (da)	1984-08-22	Pyrimido(4-5-g)quinolin-derivater, fremgangsmaade til fremstilling hraf og mellemprodukt til brug ved fremgangsmaaden
DK136784A (da)	1984-09-15	Pyrazolo(1,5-a)pyridinderivater samt fremgangsmaade til fremstilling deraf
NO874580L (no)	1988-08-10	Sveiste skjoeter og fremgangsmaate for deres fremstilling.
NO166726C (no)	1991-08-28	Fremgangsmaate for fremstilling av arylglycidyletere og 3-substituerte 1-alkylamino-2-propanoler.
DK136684D0 (da)	1984-02-29	Pyrazolo(1,5-a)pyridinderivater samt fremgangsmaade til fremstilling deraf

Legal Events

Date	Code	Title	Description
2002-03-25	PBP	Patent lapsed