DK3260455T3 - Selektive pi3k delta-hæmmere - Google Patents
Selektive pi3k delta-hæmmere Download PDFInfo
- Publication number
- DK3260455T3 DK3260455T3 DK17181585.5T DK17181585T DK3260455T3 DK 3260455 T3 DK3260455 T3 DK 3260455T3 DK 17181585 T DK17181585 T DK 17181585T DK 3260455 T3 DK3260455 T3 DK 3260455T3
- Authority
- DK
- Denmark
- Prior art keywords
- pi3k delta
- selective pi3k
- requests
- delta requests
- selective
- Prior art date
Links
- 102000010400 1-phosphatidylinositol-3-kinase activity proteins Human genes 0.000 title 1
- 108091007960 PI3Ks Proteins 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
- C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
- C12N9/10—Transferases (2.)
- C12N9/12—Transferases (2.) transferring phosphorus containing groups, e.g. kinases (2.7)
- C12N9/1205—Phosphotransferases with an alcohol group as acceptor (2.7.1), e.g. protein kinases
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12Y—ENZYMES
- C12Y207/00—Transferases transferring phosphorus-containing groups (2.7)
- C12Y207/01—Phosphotransferases with an alcohol group as acceptor (2.7.1)
- C12Y207/01137—Phosphatidylinositol 3-kinase (2.7.1.137)
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Physical Education & Sports Medicine (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Genetics & Genomics (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- General Engineering & Computer Science (AREA)
- Urology & Nephrology (AREA)
- Reproductive Health (AREA)
- Oncology (AREA)
- Obesity (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Dermatology (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN2692CH2012 | 2012-07-04 | ||
| IN2693CH2012 | 2012-07-04 | ||
| US201261691561P | 2012-08-21 | 2012-08-21 | |
| US201261691586P | 2012-08-21 | 2012-08-21 | |
| EP13744836.1A EP2870157B1 (en) | 2012-07-04 | 2013-07-02 | Selective pi3k delta inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3260455T3 true DK3260455T3 (da) | 2019-06-11 |
Family
ID=54193752
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK17181585.5T DK3260455T3 (da) | 2012-07-04 | 2013-07-02 | Selektive pi3k delta-hæmmere |
| DK13744836.1T DK2870157T3 (da) | 2012-07-04 | 2013-07-02 | Selektive pi3k delta-hæmmere |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK13744836.1T DK2870157T3 (da) | 2012-07-04 | 2013-07-02 | Selektive pi3k delta-hæmmere |
Country Status (32)
| Country | Link |
|---|---|
| US (7) | US9150579B2 (da) |
| EP (2) | EP2870157B1 (da) |
| JP (2) | JP6181173B2 (da) |
| KR (2) | KR102216606B1 (da) |
| CN (2) | CN104470923B (da) |
| AP (1) | AP2015008207A0 (da) |
| AR (1) | AR091677A1 (da) |
| AU (1) | AU2013285081B2 (da) |
| BR (1) | BR112014033055B1 (da) |
| CA (1) | CA2876995C (da) |
| CL (1) | CL2014003511A1 (da) |
| CO (1) | CO7170166A2 (da) |
| CY (2) | CY1119588T1 (da) |
| DK (2) | DK3260455T3 (da) |
| EA (1) | EA028750B1 (da) |
| ES (1) | ES2647416T3 (da) |
| HR (1) | HRP20171610T1 (da) |
| HU (1) | HUE034591T2 (da) |
| IL (1) | IL236351B (da) |
| LT (2) | LT2870157T (da) |
| MX (1) | MX357043B (da) |
| MY (1) | MY169987A (da) |
| PH (2) | PH12014502865B1 (da) |
| PL (2) | PL2870157T3 (da) |
| PT (1) | PT2870157T (da) |
| RS (2) | RS58793B1 (da) |
| SG (2) | SG11201408821SA (da) |
| SI (2) | SI2870157T1 (da) |
| SM (2) | SMT201900334T1 (da) |
| TW (1) | TWI598100B (da) |
| WO (1) | WO2014006572A1 (da) |
| ZA (2) | ZA201409329B (da) |
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| BR302012005615S1 (pt) | Configuração aplicada em arandela | |
| BR302012005617S1 (pt) | Configuração aplicada em arandela | |
| BR302012005616S1 (pt) | Configuração aplicada em arandela | |
| BR302012005100S1 (pt) | Configuracao aplicada em chinelo | |
| BR302012005102S1 (pt) | Configuracao aplicada em chinelo |