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DE69620327D1 - Wässrige, haltbare Suspension von Mesalazin zum topischen Gebrauch - Google Patents

Wässrige, haltbare Suspension von Mesalazin zum topischen Gebrauch

Info

Publication number
DE69620327D1
DE69620327D1 DE69620327T DE69620327T DE69620327D1 DE 69620327 D1 DE69620327 D1 DE 69620327D1 DE 69620327 T DE69620327 T DE 69620327T DE 69620327 T DE69620327 T DE 69620327T DE 69620327 D1 DE69620327 D1 DE 69620327D1
Authority
DE
Germany
Prior art keywords
mesalazine
aqueous
topical use
durable suspension
durable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69620327T
Other languages
English (en)
Other versions
DE69620327T2 (de
Inventor
Giancarlo Farolfi
Franco Lattuada
Laura Ferro
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gentium SRL
Original Assignee
CRINOS INDUSTRIA FARMACOBIOLOGICA SpA VILLA GUARDIA
Crinos Industria Farmacobiologica SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by CRINOS INDUSTRIA FARMACOBIOLOGICA SpA VILLA GUARDIA, Crinos Industria Farmacobiologica SpA filed Critical CRINOS INDUSTRIA FARMACOBIOLOGICA SpA VILLA GUARDIA
Application granted granted Critical
Publication of DE69620327D1 publication Critical patent/DE69620327D1/de
Publication of DE69620327T2 publication Critical patent/DE69620327T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • A61K31/606Salicylic acid; Derivatives thereof having amino groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0031Rectum, anus
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicinal Preparation (AREA)
  • Color Printing (AREA)
  • Electrically Operated Instructional Devices (AREA)
  • Colloid Chemistry (AREA)
  • Lubricants (AREA)
DE69620327T 1995-09-28 1996-06-26 Wässrige, haltbare Suspension von Mesalazin zum topischen Gebrauch Expired - Lifetime DE69620327T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT95MI001987A IT1277663B1 (it) 1995-09-28 1995-09-28 Sospensioni acquose stabili di mesalazina per uso topico

Publications (2)

Publication Number Publication Date
DE69620327D1 true DE69620327D1 (de) 2002-05-08
DE69620327T2 DE69620327T2 (de) 2002-11-21

Family

ID=11372286

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69620327T Expired - Lifetime DE69620327T2 (de) 1995-09-28 1996-06-26 Wässrige, haltbare Suspension von Mesalazin zum topischen Gebrauch

Country Status (9)

Country Link
US (1) US5731302A (de)
EP (1) EP0765664B1 (de)
JP (1) JP4251671B2 (de)
AT (1) ATE215374T1 (de)
DE (1) DE69620327T2 (de)
DK (1) DK0765664T3 (de)
ES (1) ES2172611T3 (de)
IT (1) IT1277663B1 (de)
PT (1) PT765664E (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6326364B1 (en) 1999-02-08 2001-12-04 Cedars-Sinai Medical Center Use of 5-aminosalicylates as antimicrobial agents
GB9930058D0 (en) * 1999-12-20 2000-02-09 Novartis Ag Organic compounds
ES2333337T3 (es) 2000-08-29 2010-02-19 Biocon Limited Uso de una composicion farmaceutica que contiene un derivado de acido para-aminofenilacetico para tratar afecciones inflamatorias del tracto gastrointestinal.
CA2359812C (en) 2000-11-20 2004-02-10 The Procter & Gamble Company Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures
PT1997478E (pt) 2001-02-15 2013-12-10 Access Pharma Inc Formulações líquidas para a prevenção e para o tratamento de doenças e distúrbios das mucosas
US7544348B2 (en) 2001-02-15 2009-06-09 Access Pharmaceuticals, Inc. Liquid formulations for the prevention and treatment of mucosal diseases and disorders
US6585997B2 (en) 2001-08-16 2003-07-01 Access Pharmaceuticals, Inc. Mucoadhesive erodible drug delivery device for controlled administration of pharmaceuticals and other active compounds
US8048924B2 (en) * 2001-08-29 2011-11-01 Biocon Limited Methods and compositions employing 4-aminophenylacetic acid compounds
CA2520197A1 (en) * 2003-04-23 2004-11-04 Ferring B.V. Sachet for a pharmaceutical composition
EP1773767B1 (de) 2004-07-07 2016-03-09 Biocon Limited Synthese von azogebundenen, das immunsystem regulierenden verbindungen
US7645801B2 (en) 2007-01-29 2010-01-12 Alaven Pharmaceutical Llc Reduced irritant enema for treatment of inflammatory bowel disease (IBD)
KR20080076667A (ko) * 2007-02-15 2008-08-20 주식회사 중외제약 요변성 약학 조성물
WO2010077911A1 (en) * 2008-12-17 2010-07-08 Altheus Therapeutics, Inc. Enema formulations

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4664256A (en) * 1983-09-06 1987-05-12 Farmaceutisk Laboratorium Ferring A/S Packaged stable enema solution or suspension containing 5-aminosalicyclic acid
US4657900A (en) * 1983-09-27 1987-04-14 Rowell Laboratories Pharmaceutical article of manufacture comprising a bisulfite stabilized aqueous solution of 5-aminosalicylic acid and method
US5010069A (en) * 1989-05-15 1991-04-23 Marion Laboratories, Inc. Stable liquid form of 5-aminosalicylic acid
DE3924570A1 (de) * 1989-07-25 1991-01-31 Henning Berlin Gmbh Pharmazeutische zubereitung zur rektalen verabreichung
US5378470A (en) * 1989-07-25 1995-01-03 Henning Berlin Gmbh Rectally administered pharmaceutical preparation
IT1243379B (it) * 1990-07-27 1994-06-10 Giuliani Spa Composizione farmaceutica adatta alla somministrazione rettale di principi attivi che esplicano un'azione di medicazione a livello del colon prevalentemente di tipo topico
GB9101621D0 (en) * 1991-01-25 1991-03-06 Bioglan Lab Ltd A packaged pharmaceutical product

Also Published As

Publication number Publication date
EP0765664B1 (de) 2002-04-03
ATE215374T1 (de) 2002-04-15
US5731302A (en) 1998-03-24
DE69620327T2 (de) 2002-11-21
JP4251671B2 (ja) 2009-04-08
ITMI951987A0 (de) 1995-09-28
ES2172611T3 (es) 2002-10-01
JPH09110697A (ja) 1997-04-28
IT1277663B1 (it) 1997-11-11
DK0765664T3 (da) 2002-05-21
PT765664E (pt) 2002-07-31
ITMI951987A1 (it) 1997-03-28
EP0765664A1 (de) 1997-04-02

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8327 Change in the person/name/address of the patent owner

Owner name: GENTIUM S.P.A., VILLA GUARDIA, COMO, IT