DE60223227T8 - Benzo[b]thiophenderivate und Verfahren zu deren Herstellung - Google Patents
Benzo[b]thiophenderivate und Verfahren zu deren Herstellung Download PDFInfo
- Publication number
- DE60223227T8 DE60223227T8 DE60223227T DE60223227T DE60223227T8 DE 60223227 T8 DE60223227 T8 DE 60223227T8 DE 60223227 T DE60223227 T DE 60223227T DE 60223227 T DE60223227 T DE 60223227T DE 60223227 T8 DE60223227 T8 DE 60223227T8
- Authority
- DE
- Germany
- Prior art keywords
- thiophene
- bromomethyl
- benzo
- preparation
- thiophene derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/64—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001046275 | 2001-02-22 | ||
| JP2001046275 | 2001-02-22 | ||
| JP2001135927 | 2001-05-07 | ||
| JP2001135927 | 2001-05-07 | ||
| PCT/JP2002/001611 WO2002066457A1 (en) | 2001-02-22 | 2002-02-22 | BENZO[b]THIOPHENE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DE60223227D1 DE60223227D1 (de) | 2007-12-13 |
| DE60223227T2 DE60223227T2 (de) | 2008-08-14 |
| DE60223227T8 true DE60223227T8 (de) | 2008-11-27 |
Family
ID=26609879
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60223227T Active DE60223227T8 (de) | 2001-02-22 | 2002-02-22 | Benzo[b]thiophenderivate und Verfahren zu deren Herstellung |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US6884896B2 (de) |
| EP (2) | EP1362854B1 (de) |
| JP (1) | JP3999128B2 (de) |
| KR (1) | KR100922485B1 (de) |
| CN (1) | CN100457750C (de) |
| AT (1) | ATE376830T1 (de) |
| AU (1) | AU2002233698B2 (de) |
| CA (1) | CA2406913C (de) |
| DE (1) | DE60223227T8 (de) |
| ES (1) | ES2292712T3 (de) |
| NO (1) | NO328158B1 (de) |
| NZ (1) | NZ522150A (de) |
| PL (1) | PL358494A1 (de) |
| PT (1) | PT1362854E (de) |
| WO (1) | WO2002066457A1 (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1944415B (zh) * | 2001-02-22 | 2011-04-13 | 帝人株式会社 | 苯并[b]噻吩衍生物及其制备方法 |
| CL2004001034A1 (es) * | 2003-05-14 | 2005-03-28 | Teijin Pharma Ltd | Formas cristalinas de acido 4-(1-((,etilbenzotiofen-3-il)me til)benzimidazol-2-iltio)butanoico; procedimiento de preparacion de las formas cristalinas; composicion farmaceutica; y su uso para el tratamiento de enfermedades inflamatorias, alergicas, r |
| AU2004266536A1 (en) * | 2003-08-22 | 2005-03-03 | Teijin Pharma Limited | Drug containing chymase inhibitor as the active ingredient |
| US7169807B2 (en) * | 2004-04-09 | 2007-01-30 | Allergan, Inc. | 10-Hydroxy-11-dihydroprostaglandin analogs as selective EP4 agonists |
| DE102004021637A1 (de) * | 2004-05-03 | 2005-12-01 | Merck Patent Gmbh | Dihydrobenzothiophene |
| JPWO2006052026A1 (ja) * | 2004-11-12 | 2008-05-29 | 帝人ファーマ株式会社 | ベンズイミダゾール誘導体の酸性塩及びその結晶 |
| CA2627325A1 (en) | 2005-10-27 | 2007-05-03 | Teijin Pharma Limited | 3-hydroxymethylbenzo[b]thiophene derivative and method for producing same |
| WO2007049813A1 (ja) | 2005-10-27 | 2007-05-03 | Teijin Pharma Limited | ベンゾ［ｂ］チオフェン誘導体およびその製造方法 |
| UA95788C2 (en) | 2005-12-15 | 2011-09-12 | Ф. Хоффманн-Ля Рош Аг | Fused pyrrole derivatives |
| TWI666205B (zh) | 2012-11-14 | 2019-07-21 | 日商帝人製藥股份有限公司 | 吡啶衍生物 |
| AU2017239816B9 (en) * | 2016-03-31 | 2020-09-24 | Fujifilm Corporation | Method for producing 5-(bromomethyl)-1-benzothiophene |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1174411A (en) * | 1966-03-02 | 1969-12-17 | Aspro Nicholas Ltd | Novel Benzothiophen Compounds, Compositions containing them and processes for their manufacture |
| US3910955A (en) * | 1970-12-21 | 1975-10-07 | Aspro Nicholas Ltd | Benzothiophene-ethylamines |
| US4255196A (en) * | 1979-02-23 | 1981-03-10 | Rohm And Haas Company | Lithographic ink of reduced volatile solvent content for reducing atmospheric pollution |
| EP0791589B1 (de) * | 1994-04-11 | 2002-03-06 | Chugai Seiyaku Kabushiki Kaisha | 4,6-DI-t-BUTYL-2,3-DIHYDROBENZOTHIOPHENE, DIE LDL OXIDATION HEMMEN |
| SK212001A3 (en) * | 1998-07-15 | 2001-11-06 | Teijin Ltd | Thiobenzimidazole derivatives |
| DE60026404T2 (de) * | 1999-08-02 | 2006-10-19 | F. Hoffmann-La Roche Ag | Verfahren zur Herstellung von Benzothiophen-Derivaten |
| DE60130865T2 (de) * | 2000-01-17 | 2008-07-17 | Teijin Pharma Ltd. | Benzimidazol-derivate als menschliche chymase - inhibitoren |
| JP2001199968A (ja) | 2000-01-18 | 2001-07-24 | Teijin Ltd | アミノベンズイミダゾール誘導体 |
| GB0001439D0 (en) * | 2000-01-21 | 2000-03-08 | R P Adam Limited | Method of controlling microbiological activity in water storage tanks and apparatus for use in such method |
| WO2002090345A1 (fr) * | 2001-05-07 | 2002-11-14 | Teijin Limited | Derives de 3-hydroxymethylbenzo[b]thiopene et procede de preparation |
-
2002
- 2002-02-22 AU AU2002233698A patent/AU2002233698B2/en not_active Ceased
- 2002-02-22 US US10/258,173 patent/US6884896B2/en not_active Expired - Fee Related
- 2002-02-22 PL PL02358494A patent/PL358494A1/xx not_active IP Right Cessation
- 2002-02-22 CN CNB028012909A patent/CN100457750C/zh not_active Expired - Fee Related
- 2002-02-22 AT AT02700711T patent/ATE376830T1/de not_active IP Right Cessation
- 2002-02-22 EP EP02700711A patent/EP1362854B1/de not_active Expired - Lifetime
- 2002-02-22 CA CA2406913A patent/CA2406913C/en not_active Expired - Fee Related
- 2002-02-22 ES ES02700711T patent/ES2292712T3/es not_active Expired - Lifetime
- 2002-02-22 WO PCT/JP2002/001611 patent/WO2002066457A1/ja not_active Ceased
- 2002-02-22 DE DE60223227T patent/DE60223227T8/de active Active
- 2002-02-22 KR KR1020027014185A patent/KR100922485B1/ko not_active Expired - Fee Related
- 2002-02-22 PT PT02700711T patent/PT1362854E/pt unknown
- 2002-02-22 EP EP06076752A patent/EP1792614A1/de not_active Withdrawn
- 2002-02-22 JP JP2002565972A patent/JP3999128B2/ja not_active Expired - Fee Related
- 2002-02-22 NZ NZ522150A patent/NZ522150A/xx unknown
- 2002-10-21 NO NO20025053A patent/NO328158B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CA2406913C (en) | 2011-04-19 |
| JPWO2002066457A1 (ja) | 2004-06-17 |
| KR100922485B1 (ko) | 2009-10-20 |
| ATE376830T1 (de) | 2007-11-15 |
| ES2292712T3 (es) | 2008-03-16 |
| DE60223227D1 (de) | 2007-12-13 |
| NO20025053D0 (no) | 2002-10-21 |
| WO2002066457A1 (en) | 2002-08-29 |
| US20030176490A1 (en) | 2003-09-18 |
| DE60223227T2 (de) | 2008-08-14 |
| NZ522150A (en) | 2006-03-31 |
| HK1057215A1 (en) | 2004-03-19 |
| CA2406913A1 (en) | 2002-08-29 |
| EP1362854A1 (de) | 2003-11-19 |
| EP1362854B1 (de) | 2007-10-31 |
| US6884896B2 (en) | 2005-04-26 |
| EP1362854A4 (de) | 2004-06-09 |
| JP3999128B2 (ja) | 2007-10-31 |
| AU2002233698B2 (en) | 2007-11-08 |
| NO328158B1 (no) | 2009-12-21 |
| EP1792614A1 (de) | 2007-06-06 |
| CN1461301A (zh) | 2003-12-10 |
| PL358494A1 (en) | 2004-08-09 |
| PT1362854E (pt) | 2008-01-21 |
| KR20030005293A (ko) | 2003-01-17 |
| NO20025053L (no) | 2002-11-29 |
| CN100457750C (zh) | 2009-02-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |