DE602007006601D1 - Verfahren zur reinigung von tacrolimus - Google Patents
Verfahren zur reinigung von tacrolimusInfo
- Publication number
- DE602007006601D1 DE602007006601D1 DE602007006601T DE602007006601T DE602007006601D1 DE 602007006601 D1 DE602007006601 D1 DE 602007006601D1 DE 602007006601 T DE602007006601 T DE 602007006601T DE 602007006601 T DE602007006601 T DE 602007006601T DE 602007006601 D1 DE602007006601 D1 DE 602007006601D1
- Authority
- DE
- Germany
- Prior art keywords
- tacrolimus
- cleaning
- cleaning tacrolimus
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
- QJJXYPPXXYFBGM-LFZNUXCKSA-N Tacrolimus Chemical compound C1C[C@@H](O)[C@H](OC)C[C@@H]1\C=C(/C)[C@@H]1[C@H](C)[C@@H](O)CC(=O)[C@H](CC=C)/C=C(C)/C[C@H](C)C[C@H](OC)[C@H]([C@H](C[C@H]2C)OC)O[C@@]2(O)C(=O)C(=O)N2CCCC[C@H]2C(=O)O1 QJJXYPPXXYFBGM-LFZNUXCKSA-N 0.000 title 1
- 238000004140 cleaning Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 229960001967 tacrolimus Drugs 0.000 title 1
- QJJXYPPXXYFBGM-SHYZHZOCSA-N tacrolimus Natural products CO[C@H]1C[C@H](CC[C@@H]1O)C=C(C)[C@H]2OC(=O)[C@H]3CCCCN3C(=O)C(=O)[C@@]4(O)O[C@@H]([C@H](C[C@H]4C)OC)[C@@H](C[C@H](C)CC(=C[C@@H](CC=C)C(=O)C[C@H](O)[C@H]2C)C)OC QJJXYPPXXYFBGM-SHYZHZOCSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78275306P | 2006-03-15 | 2006-03-15 | |
| US84732306P | 2006-09-25 | 2006-09-25 | |
| US86035906P | 2006-11-20 | 2006-11-20 | |
| US87482306P | 2006-12-13 | 2006-12-13 | |
| US87986907P | 2007-01-10 | 2007-01-10 | |
| PCT/US2007/006642 WO2007106587A2 (en) | 2006-03-15 | 2007-03-15 | Process for purifying tacrolimus |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE602007006601D1 true DE602007006601D1 (de) | 2010-07-01 |
Family
ID=38510109
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE602007006601T Active DE602007006601D1 (de) | 2006-03-15 | 2007-03-15 | Verfahren zur reinigung von tacrolimus |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20080000834A1 (de) |
| JP (1) | JP4700022B2 (de) |
| DE (1) | DE602007006601D1 (de) |
| IL (1) | IL191920A0 (de) |
| TW (1) | TW200815458A (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1697383T1 (sl) * | 2003-12-05 | 2014-09-30 | Biocon Limited | Postopek za čiščenje takrolimusa |
| JP2010022888A (ja) * | 2008-07-15 | 2010-02-04 | Toshiba Corp | 水質浄化材料およびそれを用いた水質浄化方法 |
| KR100910165B1 (ko) * | 2008-09-18 | 2009-07-30 | (주) 제노텍 | 은 이온 용액 추출을 이용한 불포화 알킬기를 가진 락톤 화합물 정제방법 |
| KR101344012B1 (ko) | 2012-04-09 | 2013-12-23 | 인하대학교 산학협력단 | 모사이동층 크로마토그래피를 이용하여 타크로리무스와 아스코마이신의 혼합액으로부터 타크로리무스를 분리하는 방법 |
| KR101587321B1 (ko) | 2013-07-24 | 2016-01-20 | 주식회사 엘지화학 | 연성인쇄회로기판의 구조체 |
| RU2694354C1 (ru) * | 2018-09-25 | 2019-07-11 | Закрытое акционерное общество "БиоХимМак СТ" | Способ сорбционно-хроматографического выделения и очистки такролимуса |
| CN114428133B (zh) * | 2021-12-28 | 2023-06-09 | 江苏知原药业股份有限公司 | 一种用反相色谱法检测他克莫司软膏中杂质xv含量的方法 |
| CN114516884B (zh) * | 2022-01-05 | 2024-03-19 | 福建省微生物研究所 | 一种高纯度他克莫司的提纯方法 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4894366A (en) * | 1984-12-03 | 1990-01-16 | Fujisawa Pharmaceutical Company, Ltd. | Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same |
| US5194378A (en) * | 1991-01-28 | 1993-03-16 | Merck & Co., Inc. | Process for producing fk-506 |
| US5116756A (en) * | 1991-01-28 | 1992-05-26 | Merck & Co., Inc. | Process for producing FK-506 |
| WO1993018042A1 (en) * | 1992-03-02 | 1993-09-16 | Pfizer Inc. | Desosamino derivatives of macrolides as immunosuppressants and antifungal agents |
| JP2564765B2 (ja) * | 1992-03-02 | 1996-12-18 | ファイザー・インコーポレーテッド | マクロライド系抗生物質のフルオロ糖誘導体 |
| US5264355A (en) * | 1992-07-02 | 1993-11-23 | Merck & Co., Inc. | Methlating enzyme from streptomyces MA6858 |
| UA41884C2 (uk) * | 1993-11-05 | 2001-10-15 | Амерікан Хоум Продактс Корпорейшн | Спосіб відокремлення рапаміцину від кислотних, основних та неполярних нейтральних домішок, присутніх в концентраті екстрактів ферментаційного бульйону або маточних розчинів |
| US5622866A (en) * | 1994-06-23 | 1997-04-22 | Merck & Co., Inc. | Expression cassettes useful in construction of integrative and replicative expression vectors for Streptomyces |
| US5616595A (en) * | 1995-06-07 | 1997-04-01 | Abbott Laboratories | Process for recovering water insoluble compounds from a fermentation broth |
| AU773517B2 (en) * | 1998-10-02 | 2004-05-27 | Kosan Biosciences, Inc. | Polyketide synthase enzymes and recombinant DNA constructs therefor |
| DK1183261T3 (da) * | 1999-05-25 | 2005-01-17 | Fujisawa Pharmaceutical Co | Fremgangsmåde til separering af analoge organiske forbindelser |
| TW553946B (en) * | 1999-09-08 | 2003-09-21 | Fujisawa Pharmaceutical Co | Method for separating lactone-containing high-molecular weight compounds |
| CA2433840C (en) * | 2001-01-04 | 2010-05-04 | Albert Einstein College Of Medicine Of Yeshiva University | Inhibitors of adp-ribosyl transferases, cyclases, and hydrolases, and uses thereof |
-
2007
- 2007-03-15 TW TW096108955A patent/TW200815458A/zh unknown
- 2007-03-15 US US11/725,074 patent/US20080000834A1/en not_active Abandoned
- 2007-03-15 JP JP2007066494A patent/JP4700022B2/ja not_active Expired - Fee Related
- 2007-03-15 DE DE602007006601T patent/DE602007006601D1/de active Active
-
2008
- 2008-06-03 IL IL191920A patent/IL191920A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20080000834A1 (en) | 2008-01-03 |
| TW200815458A (en) | 2008-04-01 |
| JP2007262065A (ja) | 2007-10-11 |
| IL191920A0 (en) | 2009-08-03 |
| JP4700022B2 (ja) | 2011-06-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |