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DE60118521D1 - Purin derivate, ihre herstellung und verwendung - Google Patents

Purin derivate, ihre herstellung und verwendung

Info

Publication number
DE60118521D1
DE60118521D1 DE60118521T DE60118521T DE60118521D1 DE 60118521 D1 DE60118521 D1 DE 60118521D1 DE 60118521 T DE60118521 T DE 60118521T DE 60118521 T DE60118521 T DE 60118521T DE 60118521 D1 DE60118521 D1 DE 60118521D1
Authority
DE
Germany
Prior art keywords
purine derivatives
preparation
derivatives
relates
methods
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60118521T
Other languages
English (en)
Other versions
DE60118521T2 (de
Inventor
Libor Havlicek
Vladimir Krystof
Vera Siglerov
Rene Lenobel
Onckelen Henri Van
Nisan Berneman
Herman Slegers
Edgard Esmans
Miroslav Strnad
Katrien Vermeulen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
UNIVERSITAIRE INSTELLING ANTWE
Institute of Experimental Botany Academy CAS
Original Assignee
UNIVERSITAIRE INSTELLING ANTWE
Institute of Experimental Botany Academy CAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by UNIVERSITAIRE INSTELLING ANTWE, Institute of Experimental Botany Academy CAS filed Critical UNIVERSITAIRE INSTELLING ANTWE
Publication of DE60118521D1 publication Critical patent/DE60118521D1/de
Application granted granted Critical
Publication of DE60118521T2 publication Critical patent/DE60118521T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DE60118521T 2000-01-07 2001-01-08 Purin derivate, ihre herstellung und verwendung Expired - Lifetime DE60118521T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP00200070 2000-01-07
EP00200070 2000-01-07
PCT/EP2001/000150 WO2001049688A1 (en) 2000-01-07 2001-01-08 Purine derivatives, process for their preparation and use thereof

Publications (2)

Publication Number Publication Date
DE60118521D1 true DE60118521D1 (de) 2006-05-18
DE60118521T2 DE60118521T2 (de) 2006-10-12

Family

ID=8170897

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60118521T Expired - Lifetime DE60118521T2 (de) 2000-01-07 2001-01-08 Purin derivate, ihre herstellung und verwendung

Country Status (11)

Country Link
US (1) US20030187261A1 (de)
EP (1) EP1244668B1 (de)
JP (1) JP2003519232A (de)
AT (1) ATE322494T1 (de)
AU (1) AU3540101A (de)
CA (1) CA2396276A1 (de)
CZ (1) CZ20022353A3 (de)
DE (1) DE60118521T2 (de)
IL (1) IL150594A0 (de)
NO (1) NO20023247L (de)
WO (1) WO2001049688A1 (de)

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US20030187261A1 (en) 2003-10-02
JP2003519232A (ja) 2003-06-17
ATE322494T1 (de) 2006-04-15
WO2001049688A8 (en) 2001-10-04
IL150594A0 (en) 2003-02-12
EP1244668B1 (de) 2006-04-05
CA2396276A1 (en) 2001-07-12
CZ20022353A3 (cs) 2003-02-12
NO20023247D0 (no) 2002-07-04
NO20023247L (no) 2002-09-09
WO2001049688A1 (en) 2001-07-12
DE60118521T2 (de) 2006-10-12
AU3540101A (en) 2001-07-16

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