DE60029517D1 - VERFAHREN ZUR HERSTELLUNG VON threo-1,2-EPOXY-3-AMINO-4-PHENYLBUTAN-DERIVATEN - Google Patents

VERFAHREN ZUR HERSTELLUNG VON threo-1,2-EPOXY-3-AMINO-4-PHENYLBUTAN-DERIVATEN

Info

Publication number: DE60029517D1
Authority: DE; Germany
Prior art keywords: threo; amino; epoxy; phenylbutane; preparation
Prior art date: 1999-01-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Lifetime

Application number

DE60029517T

Other languages

English (en)

Other versions

DE60029517T2 (de

Inventor

Katsuji Maehara

Yukinori Tokuda

Hiroshi Murao

Yasuyoshi Ueda

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Kaneka Corp

Original Assignee

Kaneka Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-29

Filing date

2000-01-31

Publication date

2006-09-07

2000-01-31 Application filed by Kaneka Corp filed Critical Kaneka Corp

2006-09-07 Application granted granted Critical

2006-09-07 Publication of DE60029517D1 publication Critical patent/DE60029517D1/de

2006-11-23 Publication of DE60029517T2 publication Critical patent/DE60029517T2/de

2020-02-01 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D301/00—Preparation of oxiranes
- C07D301/02—Synthesis of the oxirane ring
- C07D301/24—Synthesis of the oxirane ring by splitting off HAL—Y from compounds containing the radical HAL—C—C—OY
- C07D301/26—Y being hydrogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/36—Compounds containing oxirane rings with hydrocarbon radicals, substituted by nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Epoxy Compounds (AREA)

DE60029517T 1999-01-29 2000-01-31 VERFAHREN ZUR HERSTELLUNG VON threo-1,2-EPOXY-3-AMINO-4-PHENYLBUTAN-DERIVATEN Expired - Lifetime DE60029517T2 (de)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
JP2164099		1999-01-29
JP2164099		1999-01-29
JP23972099		1999-08-26
JP23972099		1999-08-26
PCT/JP2000/000495 WO2000044736A1 (en)	1999-01-29	2000-01-31	PROCESSES FOR THE PREPARATION OF threo-1,2-EPOXY-3-AMINO-4-PHENYLBUTANE DERIVATIVES

Publications (2)

Publication Number	Publication Date
DE60029517D1 true DE60029517D1 (de)	2006-09-07
DE60029517T2 DE60029517T2 (de)	2006-11-23

Family

ID=26358729

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE60029517T Expired - Lifetime DE60029517T2 (de)	1999-01-29	2000-01-31	VERFAHREN ZUR HERSTELLUNG VON threo-1,2-EPOXY-3-AMINO-4-PHENYLBUTAN-DERIVATEN

Country Status (8)

Country	Link
US (1)	US6344572B1 (de)
EP (2)	EP1067125B1 (de)
AT (1)	ATE334121T1 (de)
AU (1)	AU2322600A (de)
CA (1)	CA2325919C (de)
DE (1)	DE60029517T2 (de)
ES (1)	ES2267494T3 (de)
WO (1)	WO2000044736A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR100708221B1 (ko)	1999-08-31	2007-04-17	아지노모토 가부시키가이샤	에폭사이드 결정의 제조방법
GB2369356B (en) *	2000-09-18	2004-02-04	Phoenix Chemicals Ltd	Process
JP4651178B2 (ja) *	2000-10-23	2011-03-16	三菱レイヨン株式会社	２−グリシジルオキシエチル（メタ）アクリレートの製造方法
JPWO2002044136A1 (ja)	2000-11-30	2004-04-02	味の素株式会社	Ｎ保護−β−アミノアルコールの製造法およびＮ保護−β−アミノエポキシドの製造法
KR20020046948A (ko)	2000-12-12	2002-06-21	에가시라 구니오	에폭사이드 결정의 제조방법
EP1456239B1 (de) *	2001-07-31	2009-04-01	Wayne State University	Auf heparansulfat-proteoglycane gerichtete hybridproteine mit neuregulin-heparin-bindungsdomäne
ME01059B (me)	2003-12-23	2012-10-20	Janssen Sciences Ireland Uc	Proces za pripremanje (3r,3as,6ar)-heksahidrofuro [2,3-b] furan-3-il (1s,2r)-3-[[(4-aminofenil) sulfonil] (izobutil) amino]-1-benzil-2- hidroksipropilkarbamata
BRPI0417272B8 (pt)	2003-12-23	2021-05-25	Janssen R&D Ireland	processo para a preparação de (3r, 3as, 6ar)-hexahidrofuro [2,3-b] furan-3-il (1s, 2r)-3-[[(4-aminofenil) sulfonil] (isobutil) amino]-1-benzil-2-hidroxipropilcarbamato
US7582468B2 (en) *	2005-05-25	2009-09-01	Bristol-Myers Squibb Company	Process for preparing (2R,3S)-1,2-epoxy-3-(protected)amino-4-substituted butane and intermediates thereof
RU2464266C2 (ru)	2006-11-09	2012-10-20	Тиботек Фармасьютикалз Лтд.	СПОСОБЫ ПОЛУЧЕНИЯ ГЕКСАГИДРОФУРО[2,3-b] ФУРАН-3-ОЛА
ES2360654T3 (es)	2007-04-27	2011-06-08	Tibotec Pharmaceuticals	Métodos para la preparación de derivados de n-isobutil-n-(2-hidroxi-3-amino-4-fenilbutil)-p-nitrobencenosulfonilamida.
ATE500820T1 (de) *	2007-06-22	2011-03-15	Bristol Myers Squibb Co	Tablettierte atazanavirhaltige zusammensetzungen
ES2360336T3 (es) *	2007-06-22	2011-06-03	Bristol-Myers Squibb Company	Composiciones en comprimidos que contienen atazanavir.
ATE503467T1 (de) *	2007-06-22	2011-04-15	Bristol Myers Squibb Co	Tablettierte atazanavirhaltige zusammensetzungen
DK2170292T3 (da) *	2007-06-22	2014-04-07	Bristol Myers Squibb Holdings Ireland	Atazanavirholdige sammensætninger i tabletform
US20110178305A1 (en) *	2008-05-08	2011-07-21	Ranbaxy Laboratories Limited	Process for the preparation of 3,4-epoxy-2-amino-1-substituted butane derivatives and intermediate compounds thereof
TWI482775B (zh)	2008-09-01	2015-05-01	Tibotec Pharm Ltd	用於製備（３ｒ，３ａｓ，６ａｒ）－六氫呋喃并〔２，３－ｂ〕呋喃－３－基（１ｓ，２ｒ）－３－〔〔（４－胺基苯基）磺醯基〕（異丁基）胺基〕－１－苯甲基－２－羥基丙基胺基甲酸酯之方法
US8921415B2 (en)	2009-01-29	2014-12-30	Mapi Pharma Ltd.	Polymorphs of darunavir
BR112012018862A2 (pt)	2010-01-28	2015-10-13	Mapi Pharma Ltd	processo para a preparação de darunavir e intermediários de darunavir

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BR9306058A (pt) *	1992-03-11	1997-11-18	Narhex Ltd	Derivados de amina de hidrocarbonetos oxo- e hidroxi- substituidos
US5559256A (en) *	1992-07-20	1996-09-24	E. R. Squibb & Sons, Inc.	Aminediol protease inhibitors
US5481011A (en) *	1994-12-13	1996-01-02	Bristol-Myers Squibb Company	Process for preparing N-protected amino acid α-halomethyl ketones and alcohols from N-protected amino acid esters
CN1091088C (zh) *	1995-02-03	2002-09-18	钟渊化学工业株式会社	α－卤代酮、α－卤代醇和环氧化物的制备方法
EP1097919A3 (de) *	1995-11-17	2003-08-06	Ajinomoto Co., Inc.	Verfahren zur Herstellung eines 4-Amino-3-oxo-butansäureesters
JPH09323960A (ja) *	1996-06-05	1997-12-16	Ajinomoto Co Inc	３−アミノ−１，２−オキシランの製造方法

2000
- 2000-01-31 AT AT00901998T patent/ATE334121T1/de not_active IP Right Cessation
- 2000-01-31 WO PCT/JP2000/000495 patent/WO2000044736A1/ja not_active Ceased
- 2000-01-31 ES ES00901998T patent/ES2267494T3/es not_active Expired - Lifetime
- 2000-01-31 AU AU23226/00A patent/AU2322600A/en not_active Abandoned
- 2000-01-31 CA CA002325919A patent/CA2325919C/en not_active Expired - Fee Related
- 2000-01-31 US US09/647,340 patent/US6344572B1/en not_active Expired - Lifetime
- 2000-01-31 EP EP00901998A patent/EP1067125B1/de not_active Expired - Lifetime
- 2000-01-31 DE DE60029517T patent/DE60029517T2/de not_active Expired - Lifetime
- 2000-01-31 EP EP06110625A patent/EP1661893A3/de not_active Withdrawn

Also Published As

Publication number	Publication date
EP1067125A4 (de)	2004-06-16
CA2325919C (en)	2009-07-21
EP1661893A3 (de)	2006-06-07
DE60029517T2 (de)	2006-11-23
ATE334121T1 (de)	2006-08-15
WO2000044736A1 (en)	2000-08-03
EP1067125B1 (de)	2006-07-26
EP1067125A1 (de)	2001-01-10
AU2322600A (en)	2000-08-18
EP1661893A2 (de)	2006-05-31
ES2267494T3 (es)	2007-03-16
US6344572B1 (en)	2002-02-05
CA2325919A1 (en)	2000-08-03

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Legal Events

Date	Code	Title	Description
2007-08-16	8364	No opposition during term of opposition