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DE29511484U1 - Light protection agents containing p-methoxycinnamate - Google Patents

Light protection agents containing p-methoxycinnamate

Info

Publication number
DE29511484U1
DE29511484U1 DE29511484U DE29511484U DE29511484U1 DE 29511484 U1 DE29511484 U1 DE 29511484U1 DE 29511484 U DE29511484 U DE 29511484U DE 29511484 U DE29511484 U DE 29511484U DE 29511484 U1 DE29511484 U1 DE 29511484U1
Authority
DE
Germany
Prior art keywords
tocopherol
light protection
acetate
methoxycinnamate
methoxycinnamic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE29511484U
Other languages
German (de)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Priority to DE29511484U priority Critical patent/DE29511484U1/en
Publication of DE29511484U1 publication Critical patent/DE29511484U1/en
Priority to JP8179425A priority patent/JPH09104856A/en
Priority to DE29611889U priority patent/DE29611889U1/en
Priority to IT96MI000497U priority patent/ITMI960497U3/en
Priority to IT96MI001443A priority patent/IT1283144B1/en
Priority to ES09601577A priority patent/ES2120892B1/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/678Tocopherol, i.e. vitamin E
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q17/00Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
    • A61Q17/04Topical preparations for affording protection against sunlight or other radiation; Topical sun tanning preparations

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Cosmetics (AREA)
  • Anti-Oxidant Or Stabilizer Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Light Receiving Elements (AREA)
  • Investigating Materials By The Use Of Optical Means Adapted For Particular Applications (AREA)
  • Photoreceptors In Electrophotography (AREA)

Description

BASF Aktiengesellschaft.: :"'959%*^4"" ;**q«I/ 0050/46019 BASF Aktiengesellschaft.: :"'959%*^4"" ;**q«I/ 0050/46019

p-Methoxyzimtsäureester enthaltende LichtschutzagentienSunscreen agents containing p-methoxycinnamate

Beschreibung
5
Description
5

Die Erfindung betrifft als Schutz gegen UV-Licht wirksame p-Methoxyzimt säureester, die mit Tocopherol bzw. dessen Acetat gegen Oxidation stabilisiert sind.The invention relates to p-methoxycinnamic acid esters which are effective as protection against UV light and which are stabilized against oxidation with tocopherol or its acetate.

p-Methoxyzimtsäureester wie p-Methoxyzimtsäure-2-ethylhexylester oder p-Methoxyzimtsäure-isoamylester sind bekannte Marktprodukte, die als UV-B-Filter in HautSchutzmitteln Verwendung finden. Diese Lichtschutzagentien sind üblicherweise mit BHT (butyliertes Hydroxytoluol, 2,6-Di-t-butyl-p-kresol) in Mengen bis zu 1 Gew.-% stabilisiert.p-Methoxycinnamic acid esters such as p-methoxycinnamic acid 2-ethylhexyl ester or p-methoxycinnamic acid isoamyl ester are well-known market products that are used as UV-B filters in skin protection products. These light protection agents are usually stabilized with BHT (butylated hydroxytoluene, 2,6-di-t-butyl-p-cresol) in amounts of up to 1% by weight.

Obgleich BHT sehr gute stabilisierende Eigenschaften hat, ist es erwünscht, in Präparationen, die mit dem menschlichen Körper in Kontakt kommen, BHT durch natürliche Antioxidantien zu ersetzen.Although BHT has very good stabilizing properties, it is desirable to replace BHT with natural antioxidants in preparations that come into contact with the human body.

Als in der Natur in verschiedenen Ölen vorkommendes Antioxidans ist Tocopherol wohlbekannt und wird bereits auf vielen Gebieten der Nahrungsmittel- und kosmetischen Industrie verwendet, wobei sowohl die Vitamin-E-Wirkung als auch die Antioxidans-Wirkung nebeneinander zur Geltung kommen. Im Vergleich zu BHT ist Tocopherol jedoch teurer und galt im allgemeinen als weniger wirksam bezogen auf die zu verwendende Menge.As an antioxidant that occurs naturally in various oils, tocopherol is well known and is already used in many areas of the food and cosmetic industries, where both the vitamin E and antioxidant effects come into play alongside one another. However, compared to BHT, tocopherol is more expensive and is generally considered less effective in relation to the amount used.

Es wurde nun überraschenderweise gefunden, daß als Lichtschutzmittel wirkende p-Methoxyzimtsäureester statt mit BHT verbessert mit Tocopherol bzw. dessen Estern in Mengen von 0,01 bis 1 Gew.-% stabilisiert werden können, wobei bei Tocopherolzusatz die Lichtschutzagentien besonders bei längerer Lagerung besser stabilisiert werden und bei leicht erhöhter Tempratur keine Geruchsveränderungen aufweisen, während die herkömmlichen BHT-stabilisierten Agentien einen unerwünschten apfelartigen Geruch entwickeln.It has now surprisingly been found that p-methoxycinnamic acid esters acting as light stabilizers can be better stabilized with tocopherol or its esters in amounts of 0.01 to 1% by weight instead of BHT, whereby the light stabilizers are better stabilized with the addition of tocopherol, particularly during longer storage, and do not show any changes in odor at slightly higher temperatures, whereas the conventional BHT-stabilized agents develop an undesirable apple-like odor.

Gegenstand der Erfindung sind somit neue Stoffmischungen, bestehend ausschließlich aus (a) p-Methoxyzimtsäureestern und (b) untergeordneten Mengen Tocopherol bzw. dessen Acetat.The invention therefore relates to new mixtures of substances consisting exclusively of (a) p-methoxycinnamic acid esters and (b) minor amounts of tocopherol or its acetate.

Als Methoxyzimtsäureester kommen bevorzugt p-Methoxyzimtsäure-2-ethylhexylester oder -isoamylester in Betracht. Tocopherol ist vor allem cc-Tocopherol und dessen Acetat. Es kann entweder aus natürlichen Quellen, wie z.B. aus Sojadämpferöl, oder bevorzugt synthetisch hergestellt sein.The preferred methoxycinnamic acid esters are p-methoxycinnamic acid 2-ethylhexyl ester or -isoamyl ester. Tocopherol is mainly cc-tocopherol and its acetate. It can either be produced from natural sources, such as soy steamer oil, or preferably synthetically.

BASF Aktiengesellschaft·BASF Aktiengesellschaft·

0050/460190050/46019

Die Zusatzmengen des Tocopherols betragen in der Regel 0,01, bevorzugt 0,1 bis 1 Gew.-%, doch sind au größere Mengen möglich, die aber keine weitere Verbesserung der Stabilität bewirken. Demgemäß bestehen die neuen Stoffmischungen aus 99 bis 99,99, bevorzugt 99,9 Gew.-% Methoxyzimtsäureester und 0,01, bevorzugt 0,1 bis 1 Gew.-% Tocopherol.The amount of tocopherol added is generally 0.01, preferably 0.1 to 1% by weight, but larger amounts are also possible, although these do not result in any further improvement in stability. Accordingly, the new mixtures consist of 99 to 99.99, preferably 99.9% by weight of methoxycinnamate and 0.01, preferably 0.1 to 1% by weight of tocopherol.

Die Einmischung des Tocopherols erfolgt durch direktes Vermischen bzw. Einrühren des Tocopherols oder durch Einrühren einer konzentrierteren Lösung z.B. 10 % Vorlösung in dem entsprechenden Zimtsäureester. The tocopherol is mixed in by directly mixing or stirring in the tocopherol or by stirring in a more concentrated solution, e.g. 10% pre-solution in the corresponding cinnamic acid ester.

Für die Weiterverarbeitung der stabilisierten Zimt säureester in der kosmetischen Industrie zu Lichtschutzpräparationen stört der Tocopherolgehalt, insbesondere ein über die Wirksamkeitserfordernis erhöhter Gehalt an Tocopherol, nicht, da diese Präparationen in zunehmendem Maße natürliche Öle, wie Sonnenblumenöle, Weizenkeimöl oder Maiskaimöl enthalten, die ohnehin einen {geringen Gehalt an Tocopherol aufweisen.For the further processing of the stabilized cinnamic acid esters in the cosmetic industry to produce sunscreen preparations, the tocopherol content, especially a tocopherol content that exceeds the effectiveness requirement, is not a problem, since these preparations increasingly contain natural oils, such as sunflower oil, wheat germ oil or corn caim oil, which already have a low tocopherol content.

Die neuen stabilisierten p-Methoxy&zgr;imtSäurezubereitungen zeichnen sich durch eine ausgezeichnete Lagerstabilität aus.The new stabilized p-methoxyζimt acid preparations are characterized by excellent storage stability.

Beispiel 1example 1

p-Methoxyzimtsäure-2-ethylhexylester wird mit 0,1 Gew.-%, bezogen auf die Gesamtmischung an a-Tocopherol versetzt und durch Rühren gleichmäßig verteilt. Solcherart stabilisierte Proben werden bei 6°C, bei Raumtemperatur und bei 45°C in Polyethylenflaschen unter Luftabschluß gelagert. Die spezifische Absorption einer 1 %igen Lösung in Ethanol, gemessen in einer Schichtdicke von einem cm, der sogenannten E -j- -Wert in Ethanol, beträgt nach neunmonatiger Lagerung bei 6°C 869, bei Raumtemperatur 866 und bei 450C 858. Parallel unter gleichen Bedingungen gelagert Proben, die mit entsprechenden Mengen BHT stabilisiert waren, wiesen mit E !j· = 854 bei 6°C-Lagerung, 864 bei Raumtemperatur und 856 bei 45°C etwas geringere Werte für die spezifische Absorption auf, die ein empfindliches Maß für den Wirkstoffgehalt darstellt. In Bezug auf die Farbzahl unterschieden sich die verschieden stabilisierten Proben nicht.0.1% by weight of a-tocopherol, based on the total mixture, is added to p-methoxycinnamic acid-2-ethylhexyl ester and evenly distributed by stirring. Samples stabilized in this way are stored in polyethylene bottles at 6°C, at room temperature and at 45°C under exclusion of air. The specific absorption of a 1% solution in ethanol, measured in a layer thickness of one cm, the so-called E -j- value in ethanol, is 869 after nine months of storage at 6°C, 866 at room temperature and 858 at 45 0 C. Samples stored in parallel under the same conditions which were stabilized with corresponding amounts of BHT showed slightly lower values for the specific absorption, which is a sensitive measure of the active ingredient content, with E !j· = 854 when stored at 6°C, 864 at room temperature and 856 at 45°C. With regard to the color number, the differently stabilized samples did not differ.

Ferner wiesen die mit Tocopherol stabilisierten Proben keine Geruchsveränderungen auf, während die mit BHT stabilisierte und bei 450C gelagerte Proben einen unerwünschten apfelartigen Geruch entwickelte. Furthermore, the samples stabilized with tocopherol showed no odor changes, while the samples stabilized with BHT and stored at 45 ° C developed an undesirable apple-like odor.

Claims (6)

BASF Aktiengesellschaft ·· &Igr;'.' SchutzansprücheBASF Aktiengesellschaft ·· &Igr;'.' Protection claims 1. Gegen Oxidation stabilisierte Lichtschutzagentien, bestehend ausschließlich aus1. Antioxidant stabilized photoprotective agents consisting exclusively of {a) als UV-Filter wirksamen p-Methoxyzimtsäurestern und{a) p-methoxycinnamic acid esters effective as UV filters and (b) untergeordneten Mengen Tocopherol bzw. dessen Acetat als(b) minor amounts of tocopherol or its acetate as Antioxidans. 10Antioxidant. 10 2. Lichtschutzagentien gemäß Schutzanspruch 1, bestehend aus2. Light protection agents according to claim 1, consisting of (a) p-Methoxyzimtsäure-2-ethylhexylester und(a) p-methoxycinnamic acid 2-ethylhexyl ester and (b) a-Tocopherol. 15(b) a-tocopherol. 15 3. Lichtschutzagentien gemäß Schutzanspurch 1, bestehend aus3. Light protection agents according to protection claim 1, consisting of (a) p-Methoxyzimtsäure-isoamylester und(a) p-methoxycinnamic acid isoamyl ester and (b) a-Tocopherol. 20(b) a-tocopherol. 20 4. Lichtschutzagentien gemäß Schutzanspruch 1, bestehend aus4. Light protection agents according to claim 1, consisting of (a) p-Methoxyzimtsäure-2-ethylhexylester oder -isoamylester und (b) a-Tocopherolacetat.(a) 2-ethylhexyl or isoamyl p-methoxycinnamate and (b) a-tocopherol acetate. 5. Lichtschutzagentien gemäß Schutzanspruch 1, enthaltend mindestens 0,01 Gew.-% Tocopherol bzw. dessen Acetat.5. Sunscreen agents according to claim 1, containing at least 0.01% by weight of tocopherol or its acetate. 6. Lichtschutzagentien gemäß Schutzanspruch 1, enthaltend 0,01 bis 1 Gew.-% Tocopherol bzw. dessen Acetat.6. Sunscreen agents according to claim 1, containing 0.01 to 1 wt.% tocopherol or its acetate. 338/95 Hp/Br 14.07.1995 45338/95 Hp/Br 14.07.1995 45
DE29511484U 1995-07-15 1995-07-15 Light protection agents containing p-methoxycinnamate Expired - Lifetime DE29511484U1 (en)

Priority Applications (6)

Application Number Priority Date Filing Date Title
DE29511484U DE29511484U1 (en) 1995-07-15 1995-07-15 Light protection agents containing p-methoxycinnamate
JP8179425A JPH09104856A (en) 1995-07-15 1996-07-09 Light-intercepting agent stabilized against oxidation
DE29611889U DE29611889U1 (en) 1995-07-15 1996-07-09 Light protection agents containing p-methoxycinnamate
IT96MI000497U ITMI960497U3 (en) 1995-07-15 1996-07-12 LIGHT PROTECTIVE AGENTS CONTAINING P-METHOXICINNAMIC ACID ESTERS
IT96MI001443A IT1283144B1 (en) 1995-07-15 1996-07-12 PHOTOPROTECTOR AGENTS CONTAINING FOREIGN P-METHOXYNYNAMIC ACID
ES09601577A ES2120892B1 (en) 1995-07-15 1996-07-15 PROTECTIVE AGENTS AGAINST LIGHT CONTAINING ESTERS OF P-METOXYCINAMIC ACID.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE29511484U DE29511484U1 (en) 1995-07-15 1995-07-15 Light protection agents containing p-methoxycinnamate

Publications (1)

Publication Number Publication Date
DE29511484U1 true DE29511484U1 (en) 1995-10-05

Family

ID=8010589

Family Applications (2)

Application Number Title Priority Date Filing Date
DE29511484U Expired - Lifetime DE29511484U1 (en) 1995-07-15 1995-07-15 Light protection agents containing p-methoxycinnamate
DE29611889U Expired - Lifetime DE29611889U1 (en) 1995-07-15 1996-07-09 Light protection agents containing p-methoxycinnamate

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE29611889U Expired - Lifetime DE29611889U1 (en) 1995-07-15 1996-07-09 Light protection agents containing p-methoxycinnamate

Country Status (4)

Country Link
JP (1) JPH09104856A (en)
DE (2) DE29511484U1 (en)
ES (1) ES2120892B1 (en)
IT (2) IT1283144B1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4091746B2 (en) 2001-02-06 2008-05-28 日清オイリオグループ株式会社 Use for improving the stability of UV-absorbing substances, UV absorbers and cosmetics
US6869598B2 (en) * 2002-03-22 2005-03-22 Unilever Home & Personal Care Usa Division Of Conopco, Inc. Stabilization of sunscreens in cosmetic compositions

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1022749A (en) * 1963-12-21 1966-03-16 Fujisawa Pharmaceutical Co Tocopheryl 3,4-disubstituted cinnamates and their preparation
JPH0625053B2 (en) * 1986-05-15 1994-04-06 株式会社資生堂 External skin preparation
US4833259A (en) * 1986-09-15 1989-05-23 Hoffmann-La Roche Inc. Light screening agents
US4847072A (en) * 1987-10-22 1989-07-11 The Procter & Gamble Company Photoprotection compositions comprising tocopherol sorbate

Also Published As

Publication number Publication date
ITMI960497U3 (en) 1998-01-12
DE29611889U1 (en) 1996-09-12
ES2120892A1 (en) 1998-11-01
ITMI961443A1 (en) 1998-01-12
JPH09104856A (en) 1997-04-22
ITMI961443A0 (en) 1996-07-12
IT1283144B1 (en) 1998-04-07
ITMI961443A3 (en) 1998-01-12
ITMI960497V0 (en) 1996-07-12
ES2120892B1 (en) 1999-07-01

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Legal Events

Date Code Title Description
R207 Utility model specification

Effective date: 19951116

R156 Lapse of ip right after 3 years

Effective date: 19980829