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GB1022749A - Tocopheryl 3,4-disubstituted cinnamates and their preparation - Google Patents

Tocopheryl 3,4-disubstituted cinnamates and their preparation

Info

Publication number
GB1022749A
GB1022749A GB49997/64A GB4999764A GB1022749A GB 1022749 A GB1022749 A GB 1022749A GB 49997/64 A GB49997/64 A GB 49997/64A GB 4999764 A GB4999764 A GB 4999764A GB 1022749 A GB1022749 A GB 1022749A
Authority
GB
United Kingdom
Prior art keywords
methoxy
hydroxy
cinnamates
disubstituted
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB49997/64A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Publication of GB1022749A publication Critical patent/GB1022749A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • C07D311/70Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with two hydrocarbon radicals attached in position 2 and elements other than carbon and hydrogen in position 6
    • C07D311/723,4-Dihydro derivatives having in position 2 at least one methyl radical and in position 6 one oxygen atom, e.g. tocopherols

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention comprises compounds of formula <FORM:1022749/C2/1> wherein R1 and R2 are H or methyl and R3 and R4 are H, C1-6-alkyl, C1-6-alkoxy-carbonyl or monocarboxylic acyl. Specified are alphatocopheryl cinnamates substituted as follows: 3,4 - dihydroxy; 3,4 - dimethoxycarbonyloxy; 3,4 - diethoxycarbonyloxy; 3,4 - diacetoxy; 3 - methoxy - 4 - methoxycarbonyloxy; 3-methoxy - 4 - ethoxycarbonyloxy; 3 - methoxy-4 - hydroxy. The compounds are prepared by reacting together the corresponding tocopherol and 3,4-disubstituted cinnamic acid or a reactive derivative of the latter; alternatively, where one or both of R3 and R4 are hydroxy, the corresponding alkoxycarbonyloxy or acyloxy compounds are first prepared and the groups referred to are hydrolysed to hydroxy.
GB49997/64A 1963-12-21 1964-12-08 Tocopheryl 3,4-disubstituted cinnamates and their preparation Expired GB1022749A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP6909963 1963-12-21

Publications (1)

Publication Number Publication Date
GB1022749A true GB1022749A (en) 1966-03-16

Family

ID=13392819

Family Applications (1)

Application Number Title Priority Date Filing Date
GB49997/64A Expired GB1022749A (en) 1963-12-21 1964-12-08 Tocopheryl 3,4-disubstituted cinnamates and their preparation

Country Status (3)

Country Link
FR (1) FR4130M (en)
GB (1) GB1022749A (en)
NL (1) NL6414867A (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2120892A1 (en) * 1995-07-15 1998-11-01 Basf Ag Light-intercepting agent stabilized against oxidation
CN121248561A (en) * 2025-12-04 2026-01-02 广州同隽医药科技有限公司 Highly stable pyranol derivatives with photoprotective and whitening activities, their preparation methods and applications

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2120892A1 (en) * 1995-07-15 1998-11-01 Basf Ag Light-intercepting agent stabilized against oxidation
CN121248561A (en) * 2025-12-04 2026-01-02 广州同隽医药科技有限公司 Highly stable pyranol derivatives with photoprotective and whitening activities, their preparation methods and applications

Also Published As

Publication number Publication date
NL6414867A (en) 1965-06-22
FR4130M (en) 1966-05-02

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