DD284027A5 - Verfahren zur herstellung von renininhibitoren - Google Patents

Verfahren zur herstellung von renininhibitoren Download PDF

Info

Publication number: DD284027A5
Authority: DD; German Democratic Republic
Prior art keywords: cha; ala; carbon atoms; lead; compound
Prior art date: 1988-06-28

Application number

DD89330012A

Other languages

German (de)

English (en)

Inventor

Jan O Karlsson

Erik M H Sohtell

Rolf Ch Westerlund

Original Assignee

��@��k��

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-06-28

Filing date

1989-06-27

Publication date

1990-10-31

1989-06-27 Application filed by ��@��k�� filed Critical ��@��k��

1990-10-31 Publication of DD284027A5 publication Critical patent/DD284027A5/de

Links

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- C07K—PEPTIDES
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- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/14—Angiotensins: Related peptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C317/28—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Cardiology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Heart & Thoracic Surgery (AREA)
Vascular Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DD89330012A 1988-06-28 1989-06-27 Verfahren zur herstellung von renininhibitoren DD284027A5 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
SE8802428A SE8802428D0 (sv)	1988-06-28	1988-06-28	New compounds

Publications (1)

Publication Number	Publication Date
DD284027A5 true DD284027A5 (de)	1990-10-31

Family

ID=20372758

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DD89330012A DD284027A5 (de)	1988-06-28	1989-06-27	Verfahren zur herstellung von renininhibitoren

Country Status (14)

Country	Link
EP (1)	EP0353211A1 (no)
JP (1)	JPH0285245A (no)
KR (1)	KR900000383A (no)
CN (1)	CN1039028A (no)
AU (1)	AU3671189A (no)
DD (1)	DD284027A5 (no)
DK (1)	DK300989A (no)
FI (1)	FI893118A7 (no)
HU (1)	HUT51291A (no)
NO (1)	NO892564L (no)
PT (1)	PT90992A (no)
SE (1)	SE8802428D0 (no)
YU (1)	YU132789A (no)
ZA (1)	ZA894544B (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1991009838A1 (en) *	1989-12-22	1991-07-11	Aktiebolaget Astra	New amides
US5314920A (en) *	1992-07-20	1994-05-24	G. D. Searle & Co.	Ethynyl-alanine aryl/alkylsulfonyl-terminated amino-diol compounds for treatment of hypertension
US5317039A (en) *	1992-07-20	1994-05-31	G. D. Searle & Co.	Cyclopropyl-alanine aryl/alkylsulfide/sulfonyl-terminated amino-diol compounds for treatment of hypertension
US8168616B1 (en) *	2000-11-17	2012-05-01	Novartis Ag	Combination comprising a renin inhibitor and an angiotensin receptor inhibitor for hypertension
KR20010088472A (ko) *	2001-07-19	2001-09-28	이강섭	석재, 철, 콘크리트, 목재, 플라스틱 등 기존의 모든물건의 바탕에 자연적으로 대리석 무늬를 형성하는 공법

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4645759A (en) *	1984-06-22	1987-02-24	Abbott Laboratories	Renin inhibiting compounds
JPS63503380A (ja) *	1986-01-16	1988-12-08	アボット・ラボラトリーズ	ペプチド類似体
WO1988002374A2 (en) *	1986-09-30	1988-04-07	The Upjohn Company	Renin inhibitory peptides having novel c-terminal moieties
SE8605573D0 (sv) *	1986-12-29	1986-12-29	Haessle Ab	Novel compounds

1988
- 1988-06-28 SE SE8802428A patent/SE8802428D0/xx unknown
1989
- 1989-06-14 ZA ZA894544A patent/ZA894544B/xx unknown
- 1989-06-19 DK DK300989A patent/DK300989A/da unknown
- 1989-06-20 EP EP89850205A patent/EP0353211A1/en not_active Withdrawn
- 1989-06-21 NO NO89892564A patent/NO892564L/no unknown
- 1989-06-22 AU AU36711/89A patent/AU3671189A/en not_active Abandoned
- 1989-06-27 HU HU893239A patent/HUT51291A/hu unknown
- 1989-06-27 DD DD89330012A patent/DD284027A5/de not_active IP Right Cessation
- 1989-06-27 JP JP1162851A patent/JPH0285245A/ja active Pending
- 1989-06-27 PT PT90992A patent/PT90992A/pt not_active Application Discontinuation
- 1989-06-27 KR KR1019890008878A patent/KR900000383A/ko not_active Withdrawn
- 1989-06-27 FI FI893118A patent/FI893118A7/fi not_active Application Discontinuation
- 1989-06-28 YU YU132789A patent/YU132789A/sh unknown
- 1989-06-28 CN CN89104514A patent/CN1039028A/zh active Pending

Also Published As

Publication number	Publication date
ZA894544B (en)	1990-07-25
YU132789A (sh)	1992-09-07
DK300989A (da)	1989-12-29
SE8802428D0 (sv)	1988-06-28
AU3671189A (en)	1990-01-04
DK300989D0 (da)	1989-06-19
CN1039028A (zh)	1990-01-24
JPH0285245A (ja)	1990-03-26
FI893118A7 (fi)	1989-12-29
EP0353211A1 (en)	1990-01-31
PT90992A (pt)	1989-12-29
NO892564D0 (no)	1989-06-21
HUT51291A (en)	1990-04-28
NO892564L (no)	1989-12-29
FI893118A0 (fi)	1989-06-27
KR900000383A (ko)	1990-01-30

Publication	Publication Date	Title
EP0184550B1 (de)	1992-03-18	5-Amino-4-hydroxyvalerylamid-Derivate
DE3789371T2 (de)	1994-09-08	Aryloxy- und Arylacyloxymethyl-Ketone als Thiolprotease-Hemmungsstoffe.
EP0090341B1 (de)	1987-07-29	Spiro(4.(3+n))-2-aza-alkan-3-carbonsäure-Derivate, Verfahren zu ihrer Herstellung, diese enthaltende Mittel und ihre Verwendung
DE69404324T2 (de)	1998-01-08	Matrix metallprotease inhibitoren
DE4004820A1 (de)	1991-04-25	Renininhibitoren, verfahren zur herstellung und ihre verwendung in arzneimitteln
DE3643977A1 (de)	1987-07-02	Harnstoff-derivate mit renin inhibierender wirkung
DD243932A5 (de)	1987-03-18	Verfahren zur herstellung von n,n'-dialkylguanidino-dipeptiden
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DE69405572T2 (de)	1998-02-12	Matrix-metalloprotease inhibitoren
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