CZ105598A3 - Deriváty 5-O-desoaminyl 6-O-methyl erytronolidu A, způsob jejich přípravy a použití při přípravě biologicky aktivních produktů - Google Patents

Deriváty 5-O-desoaminyl 6-O-methyl erytronolidu A, způsob jejich přípravy a použití při přípravě biologicky aktivních produktů

Info

Publication number: CZ105598A3
Authority: CZ; Czechia
Prior art keywords: desoaminyl; derivatives; preparation; biologically active; active products
Prior art date: 1995-10-09

Application number

CZ981055A

Other languages

English (en)

Other versions

CZ293430B6 (cs

Inventor

Alain Bonnet

Bernadette Chappert

Jaques Lagouardat

Original Assignee

Hoechst Marion Roussel

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-10-09

Filing date

1996-10-08

Publication date

1998-07-15

1996-10-08 Application filed by Hoechst Marion Roussel filed Critical Hoechst Marion Roussel

1998-07-15 Publication of CZ105598A3 publication Critical patent/CZ105598A3/cs

2004-04-14 Publication of CZ293430B6 publication Critical patent/CZ293430B6/cs

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)

CZ19981055A 1995-10-09 1996-10-08 Sloučeniny 5-O-desoaminyl 6-O-methylerytronolidu A a způsob jejich přípravy CZ293430B6 (cs)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9511861A FR2739620B1 (fr)	1995-10-09	1995-10-09	Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (2)

Publication Number	Publication Date
CZ105598A3 true CZ105598A3 (cs)	1998-07-15
CZ293430B6 CZ293430B6 (cs)	2004-04-14

Family

ID=9483377

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CZ19981055A CZ293430B6 (cs)	1995-10-09	1996-10-08	Sloučeniny 5-O-desoaminyl 6-O-methylerytronolidu A a způsob jejich přípravy

Country Status (33)

Country	Link
US (1)	US6011142A (cs)
EP (1)	EP0854879B1 (cs)
JP (1)	JP4327248B2 (cs)
KR (1)	KR100451063B1 (cs)
CN (1)	CN1067401C (cs)
AP (1)	AP888A (cs)
AR (1)	AR004688A1 (cs)
AT (1)	ATE212034T1 (cs)
AU (1)	AU708351B2 (cs)
BG (1)	BG63752B1 (cs)
BR (1)	BR9610959A (cs)
CA (1)	CA2231562C (cs)
CZ (1)	CZ293430B6 (cs)
DE (1)	DE69618607T2 (cs)
DK (1)	DK0854879T3 (cs)
EA (1)	EA000765B1 (cs)
EE (1)	EE03878B1 (cs)
ES (1)	ES2171722T3 (cs)
FR (1)	FR2739620B1 (cs)
GE (1)	GEP20032899B (cs)
HU (1)	HUP9900136A3 (cs)
IL (1)	IL123613A0 (cs)
MX (1)	MX9802655A (cs)
NO (1)	NO312592B1 (cs)
PL (1)	PL183645B1 (cs)
PT (1)	PT854879E (cs)
RO (1)	RO118874B1 (cs)
SI (1)	SI0854879T1 (cs)
SK (1)	SK283619B6 (cs)
TR (1)	TR199800624T1 (cs)
UA (1)	UA52621C2 (cs)
WO (1)	WO1997013774A2 (cs)
ZA (1)	ZA966666B (cs)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2777282B1 (fr) *	1998-04-08	2001-04-20	Hoechst Marion Roussel Inc	Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
MXPA01010521A (es)	1999-04-16	2003-08-19	Johnson & Johnson	Antibacteriales de cetolidos.
US6590083B1 (en)	1999-04-16	2003-07-08	Ortho-Mcneil Pharmaceutical, Inc.	Ketolide antibacterials
WO2000063224A2 (en) *	1999-04-16	2000-10-26	Kosan Biosciences, Inc.	Macrolide antiinfective agents
GB0031312D0 (en) *	2000-12-21	2001-02-07	Glaxo Group Ltd	Macrolides
EP3738591A3 (en)	2003-03-10	2021-03-24	Merck Sharp & Dohme Corp.	Novel antibacterial agents
WO2009055557A1 (en) *	2007-10-25	2009-04-30	Cempra Pharmaceuticals, Inc.	Process for the preparation of macrolide antibacterial agents
HRP20160222T1 (hr) *	2008-10-24	2016-04-08	Cempra Pharmaceuticals, Inc.	Biozaštite uporabom makrolida koji sadrže triazol
US9937194B1 (en)	2009-06-12	2018-04-10	Cempra Pharmaceuticals, Inc.	Compounds and methods for treating inflammatory diseases
AU2010292010B2 (en)	2009-09-10	2016-01-07	Cempra Pharmaceuticals, Inc.	Methods for treating malaria, tuberculosis and MAC diseases
NZ602544A (en)	2010-03-22	2014-11-28	Cempra Pharmaceuticals Inc	Crystalline forms of a macrolide, and uses therefor
RU2608390C2 (ru)	2010-05-20	2017-01-18	Семпра Фармасьютикалз, Инк.	Способы получения макролидов и кетолидов, и промежуточных соединений для их получения
JP6042334B2 (ja)	2010-09-10	2016-12-14	センプラファーマシューティカルズ，インコーポレイテッド	疾患治療のための水素結合形成フルオロケトライド
HK1205939A1 (en)	2012-03-27	2015-12-31	Cempra Pharmaceuticals, Inc.	Parenteral formulations for administering macrolide antibiotics
HK1217665A1 (zh)	2013-03-14	2017-01-20	森普拉制药公司	用於治療呼吸道疾病的方法及其製劑
AU2014233240B2 (en)	2013-03-15	2018-08-09	Cempra Pharmaceuticals, Inc.	Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3923784A (en) *	1973-09-10	1975-12-02	Hoffmann La Roche	Erythromycin a derivatives
US4518590A (en) *	1984-04-13	1985-05-21	Pfizer Inc.	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) *	1986-06-04	1988-05-03	Abbott Laboratories	Semisynthetic erythromycin antibiotics
US4921839A (en) *	1987-02-24	1990-05-01	Beecham Group P.L.C.	Erythromycin a 11,12-carbonate 9-oxime derivatives
US5523399A (en) *	1991-12-27	1996-06-04	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives
ES2096915T3 (es) *	1992-04-22	1997-03-16	Taisho Pharmaceutical Co Ltd	Derivado de 5-o-desosaminileritronolida a.
FR2692579B1 (fr) *	1992-06-19	1995-06-02	Roussel Uclaf	Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
EP0682038A4 (en) *	1993-01-26	1996-12-27	Taisho Pharmaceutical Co Ltd	5-0-DESOSAMINYLERYTHRONOLIDE DERIVATIVE.

1995
- 1995-10-09 FR FR9511861A patent/FR2739620B1/fr not_active Expired - Fee Related
1996
- 1996-08-06 ZA ZA9606666A patent/ZA966666B/xx unknown
- 1996-08-10 UA UA98041836A patent/UA52621C2/uk unknown
- 1996-10-07 AR ARP960104634A patent/AR004688A1/es not_active Application Discontinuation
- 1996-10-08 BR BR9610959A patent/BR9610959A/pt not_active Application Discontinuation
- 1996-10-08 EP EP96933501A patent/EP0854879B1/fr not_active Expired - Lifetime
- 1996-10-08 SK SK431-98A patent/SK283619B6/sk unknown
- 1996-10-08 CZ CZ19981055A patent/CZ293430B6/cs not_active IP Right Cessation
- 1996-10-08 DK DK96933501T patent/DK0854879T3/da active
- 1996-10-08 HU HU9900136A patent/HUP9900136A3/hu unknown
- 1996-10-08 ES ES96933501T patent/ES2171722T3/es not_active Expired - Lifetime
- 1996-10-08 PL PL96326001A patent/PL183645B1/pl not_active IP Right Cessation
- 1996-10-08 EA EA199800280A patent/EA000765B1/ru not_active IP Right Cessation
- 1996-10-08 SI SI9630452T patent/SI0854879T1/xx unknown
- 1996-10-08 EE EE9800109A patent/EE03878B1/xx not_active IP Right Cessation
- 1996-10-08 KR KR10-1998-0702581A patent/KR100451063B1/ko not_active Expired - Lifetime
- 1996-10-08 AT AT96933501T patent/ATE212034T1/de active
- 1996-10-08 GE GEAP19964227A patent/GEP20032899B/en unknown
- 1996-10-08 PT PT96933501T patent/PT854879E/pt unknown
- 1996-10-08 US US09/051,378 patent/US6011142A/en not_active Ceased
- 1996-10-08 CA CA002231562A patent/CA2231562C/fr not_active Expired - Lifetime
- 1996-10-08 JP JP51476697A patent/JP4327248B2/ja not_active Expired - Lifetime
- 1996-10-08 TR TR1998/00624T patent/TR199800624T1/xx unknown
- 1996-10-08 RO RO98-00826A patent/RO118874B1/ro unknown
- 1996-10-08 WO PCT/FR1996/001567 patent/WO1997013774A2/fr not_active Ceased
- 1996-10-08 CN CN96197514A patent/CN1067401C/zh not_active Expired - Lifetime
- 1996-10-08 IL IL12361396A patent/IL123613A0/xx not_active IP Right Cessation
- 1996-10-08 DE DE69618607T patent/DE69618607T2/de not_active Expired - Lifetime
- 1996-10-08 AP APAP/P/1998/001216A patent/AP888A/en active
- 1996-10-08 AU AU72208/96A patent/AU708351B2/en not_active Expired
1998
- 1998-03-25 BG BG102350A patent/BG63752B1/bg unknown
- 1998-04-03 MX MX9802655A patent/MX9802655A/es unknown
- 1998-04-08 NO NO19981630A patent/NO312592B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
ATE212034T1 (de)	2002-02-15
EE9800109A (et)	1998-10-15
MX9802655A (es)	1998-11-30
PL326001A1 (en)	1998-08-17
KR100451063B1 (ko)	2004-12-17
PT854879E (pt)	2002-07-31
DE69618607D1 (de)	2002-02-21
AU7220896A (en)	1997-04-30
PL183645B1 (pl)	2002-06-28
UA52621C2 (uk)	2003-01-15
JP4327248B2 (ja)	2009-09-09
US6011142A (en)	2000-01-04
WO1997013774A2 (fr)	1997-04-17
TR199800624T1 (xx)	1998-06-22
BG102350A (en)	1999-03-31
CA2231562C (fr)	2006-11-28
DE69618607T2 (de)	2002-08-14
DK0854879T3 (da)	2002-05-06
CA2231562A1 (fr)	1997-04-17
EA000765B1 (ru)	2000-04-24
EA199800280A1 (ru)	1998-10-29
EP0854879B1 (fr)	2002-01-16
FR2739620A1 (fr)	1997-04-11
CZ293430B6 (cs)	2004-04-14
NO312592B1 (no)	2002-06-03
NO981630L (no)	1998-04-08
EE03878B1 (et)	2002-10-15
RO118874B1 (ro)	2003-12-30
CN1199403A (zh)	1998-11-18
HUP9900136A3 (en)	2000-04-28
IL123613A0 (en)	1998-10-30
SI0854879T1 (en)	2002-08-31
WO1997013774A3 (fr)	1997-05-29
BR9610959A (pt)	1999-03-02
KR19990064100A (ko)	1999-07-26
NO981630D0 (no)	1998-04-08
SK43198A3 (en)	1998-11-04
AU708351B2 (en)	1999-08-05
GEP20032899B (en)	2003-02-25
FR2739620B1 (fr)	1997-12-19
HUP9900136A1 (hu)	1999-05-28
EP0854879A2 (fr)	1998-07-29
BG63752B1 (bg)	2002-11-29
ES2171722T3 (es)	2002-09-16
SK283619B6 (sk)	2003-10-07
ZA966666B (en)	1997-08-06
JPH11513401A (ja)	1999-11-16
AP888A (en)	2000-11-10
AR004688A1 (es)	1999-03-10
CN1067401C (zh)	2001-06-20

Publication	Publication Date	Title
HUP9802930A3 (en)	1999-12-28	Novel 5-o-deoaminyl 6-o-methyl erythronolide a derivatives, method for preparing same and application thereof for preparing biologically active products
SI0680967T1 (en)	1999-02-28	Erythromycin derivatives, their process of preparation and their use as medicaments
ZA952059B (en)	1996-03-13	Erythromycin derivatives their preparation process and their use as medicaments
CZ105598A3 (cs)	1998-07-15	Deriváty 5-O-desoaminyl 6-O-methyl erytronolidu A, způsob jejich přípravy a použití při přípravě biologicky aktivních produktů
HUT70411A (en)	1995-10-30	Antiparasitic avermectin derivatives, process for preparing them and pharmaceutical compositions containing them
AU5625696A (en)	1997-01-09	Stable vaccine compositions for parenteral administration, a method for their use, and a process for their preparation
HUP0002252A3 (en)	2002-01-28	9-oxime erythromycin derivatives, process for preparing them and pharmaceutical compositions containing them
ZA955992B (en)	1996-02-22	Organometallic derivatives of group IIIA and process for their preparation
CZ20011622A3 (cs)	2001-09-12	Nové deriváty erythromycinu, způsob jejich přípravy a jejich použití jako léčiv
HUP9802320A3 (en)	1999-03-29	Macrolides, procedure of the preparation of macrolides, macrolides containing pharmaceutical products
ZA997176B (en)	2000-11-20	Derivatives of erythromycin, their preparation process and their use as medicaments.
IL132761A0 (en)	2001-03-19	Crystalline macrolides and process for their preparation
AU4946896A (en)	1996-09-18	Novel bi-tryptaminic derivatives, preparation process and utilization as drugs
AU3853597A (en)	1998-02-10	New derivatives of erythromycin, their preparation process and their use as medicaments
ZA9711101B (en)	1998-12-10	Derivatives of erythromycin their preparation process and their use as medicaments
HUP0001245A3 (en)	2003-05-28	Novel erythromycin derivatives, method of preparation and application as medicines
AU5667998A (en)	1998-07-17	New derivatives of erythromycin, a method for preparing them, and their use as medicines
ZA961986B (en)	1996-11-21	Phosponomonoester nucleic acids, process for their preparation, and their use
AU7297196A (en)	1997-05-22	Pyridylacetic acid derivatives, process and intermediate products for their preparation, and their use

Legal Events

Date	Code	Title	Description
2000-06-30	PD00	Pending as of 2000-06-30 in czech republic
2006-06-14	MM4A	Patent lapsed due to non-payment of fee	Effective date: 20051008