CU20160119A7 - Formulaciones tópicas de heparina - Google Patents
Formulaciones tópicas de heparinaInfo
- Publication number
- CU20160119A7 CU20160119A7 CUP2016000119A CU20160119A CU20160119A7 CU 20160119 A7 CU20160119 A7 CU 20160119A7 CU P2016000119 A CUP2016000119 A CU P2016000119A CU 20160119 A CU20160119 A CU 20160119A CU 20160119 A7 CU20160119 A7 CU 20160119A7
- Authority
- CU
- Cuba
- Prior art keywords
- topical formulations
- present
- heparine
- formulations
- topical
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
- A61K31/726—Glycosaminoglycans, i.e. mucopolysaccharides
- A61K31/727—Heparin; Heparan
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/12—Aerosols; Foams
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Molecular Biology (AREA)
- Inorganic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se relaciona con formulaciones tópicas avanzadas de sales farmacéuticamente aceptables de Heparina que proporcionan penetración transdérmica mejorada. La presente invención proporciona formulaciones líquidas, no pegajosas, claras en las que el fármaco está listo para la absorción y que son adecuadas para administración en la forma de una solución o una pulverización. Las formulaciones tópicas de la presente invención no forman película con escamas o similar al gel sobre la superficie de la piel luego de aplicación tópica.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN475MU2014 | 2014-02-10 | ||
| PCT/IB2015/050986 WO2015118512A1 (en) | 2014-02-10 | 2015-02-10 | Topical formulations of heparin |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CU20160119A7 true CU20160119A7 (es) | 2016-10-28 |
| CU24444B1 CU24444B1 (es) | 2019-10-04 |
Family
ID=52684592
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU2016000119A CU24444B1 (es) | 2014-02-10 | 2015-02-10 | Formulaciones tópicas de heparina |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US9861655B2 (es) |
| EP (1) | EP3104839B1 (es) |
| JP (1) | JP6275877B2 (es) |
| KR (1) | KR101822133B1 (es) |
| CN (1) | CN106163498A (es) |
| AP (1) | AP2016009350A0 (es) |
| AR (1) | AR099333A1 (es) |
| AU (1) | AU2015213569B2 (es) |
| CA (1) | CA2938388C (es) |
| CL (1) | CL2016001952A1 (es) |
| CU (1) | CU24444B1 (es) |
| DK (1) | DK3104839T3 (es) |
| DO (1) | DOP2016000198A (es) |
| EA (1) | EA032200B1 (es) |
| EC (1) | ECSP16069947A (es) |
| IL (1) | IL246974B (es) |
| MA (1) | MA39304B1 (es) |
| MX (1) | MX357765B (es) |
| MY (1) | MY182620A (es) |
| NZ (1) | NZ722830A (es) |
| PE (1) | PE20161173A1 (es) |
| PH (1) | PH12016501500B1 (es) |
| TW (1) | TWI538697B (es) |
| UA (1) | UA118279C2 (es) |
| WO (1) | WO2015118512A1 (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107115326B (zh) * | 2010-04-13 | 2021-01-22 | 雷尔玛达治疗股份有限公司 | 1-甲基-n-(2,6-二甲苯基)-2-哌啶甲酰胺的皮肤用药物组合物及其使用方法 |
| CN112546061B (zh) * | 2021-02-25 | 2021-06-11 | 中南大学湘雅医院 | 一种肝素类药物组合物、喷鼻剂及其制备方法及应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3323389A1 (de) * | 1983-06-29 | 1985-01-10 | B. Braun Melsungen Ag, 3508 Melsungen | Auf schleimhaeute des mundes, der nase und/oder des rachens wirkende arzneimittel auf der basis von heparin und tensiden |
| JPH02207018A (ja) * | 1989-02-07 | 1990-08-16 | Kao Corp | 皮膚外用剤 |
| EP0704206B1 (de) | 1994-09-30 | 2002-09-04 | MIKA Pharma Gesellschaft für die Entwicklung und Vermarktung pharmazeutischer Produkte mbH | Pharmazeutische Zusammensetzung |
| IT1275955B1 (it) | 1995-03-22 | 1997-10-24 | Dompe Spa | Formulazioni farmaceutiche in forma di gel tissotropico |
| JPH10279466A (ja) * | 1997-04-07 | 1998-10-20 | Kose Corp | 外用剤 |
| US6761903B2 (en) | 1999-06-30 | 2004-07-13 | Lipocine, Inc. | Clear oil-containing pharmaceutical compositions containing a therapeutic agent |
| BRPI0101486B1 (pt) | 2001-04-17 | 2017-09-19 | Cristália Produtos Químicos Farmacêuticos Ltda. | Pharmaceutical composition for topic use containing heparin for the treatment of skin or mucosal injuries caused by burns |
| CN101583369B (zh) * | 2006-11-15 | 2015-03-11 | 关节炎缓痛补充剂有限公司 | 局部制剂及其用途 |
| IT1400232B1 (it) * | 2010-05-07 | 2013-05-24 | Advance Holdings Ltd | Composizione farmaceutica topica comprendente eparina |
| RU2013147883A (ru) * | 2011-04-01 | 2015-05-10 | Юниверсити Оф Флорида Рисеч Фаундэйшн, Инк. | Термочувствительные, мукоадгезивные или кожно-адгезивные и усиливающие проникновение композиции для местной доставки терапевтических средств |
-
2015
- 2015-02-10 CN CN201580007796.6A patent/CN106163498A/zh active Pending
- 2015-02-10 WO PCT/IB2015/050986 patent/WO2015118512A1/en not_active Ceased
- 2015-02-10 MY MYPI2016702732A patent/MY182620A/en unknown
- 2015-02-10 UA UAA201608842A patent/UA118279C2/uk unknown
- 2015-02-10 KR KR1020167023895A patent/KR101822133B1/ko not_active Expired - Fee Related
- 2015-02-10 MX MX2016010399A patent/MX357765B/es active IP Right Grant
- 2015-02-10 US US15/116,060 patent/US9861655B2/en not_active Expired - Fee Related
- 2015-02-10 AP AP2016009350A patent/AP2016009350A0/en unknown
- 2015-02-10 DK DK15710252.6T patent/DK3104839T3/da active
- 2015-02-10 EA EA201691596A patent/EA032200B1/ru unknown
- 2015-02-10 TW TW104104460A patent/TWI538697B/zh not_active IP Right Cessation
- 2015-02-10 AR ARP150100384A patent/AR099333A1/es unknown
- 2015-02-10 CA CA2938388A patent/CA2938388C/en active Active
- 2015-02-10 MA MA39304A patent/MA39304B1/fr unknown
- 2015-02-10 CU CU2016000119A patent/CU24444B1/es unknown
- 2015-02-10 NZ NZ722830A patent/NZ722830A/en not_active IP Right Cessation
- 2015-02-10 EP EP15710252.6A patent/EP3104839B1/en active Active
- 2015-02-10 JP JP2016568157A patent/JP6275877B2/ja not_active Expired - Fee Related
- 2015-02-10 PE PE2016001445A patent/PE20161173A1/es unknown
- 2015-02-10 AU AU2015213569A patent/AU2015213569B2/en not_active Ceased
-
2016
- 2016-07-27 IL IL246974A patent/IL246974B/en active IP Right Grant
- 2016-07-28 PH PH12016501500A patent/PH12016501500B1/en unknown
- 2016-08-02 CL CL2016001952A patent/CL2016001952A1/es unknown
- 2016-08-03 DO DO2016000198A patent/DOP2016000198A/es unknown
- 2016-08-26 EC ECIEPI201669947A patent/ECSP16069947A/es unknown
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