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CU20160119A7 - Formulaciones tópicas de heparina - Google Patents

Formulaciones tópicas de heparina

Info

Publication number
CU20160119A7
CU20160119A7 CUP2016000119A CU20160119A CU20160119A7 CU 20160119 A7 CU20160119 A7 CU 20160119A7 CU P2016000119 A CUP2016000119 A CU P2016000119A CU 20160119 A CU20160119 A CU 20160119A CU 20160119 A7 CU20160119 A7 CU 20160119A7
Authority
CU
Cuba
Prior art keywords
topical formulations
present
heparine
formulations
topical
Prior art date
Application number
CUP2016000119A
Other languages
English (en)
Other versions
CU24444B1 (es
Inventor
K R Patel
M R Patel
A K Patel
Prakash J Shah
Original Assignee
Troikaa Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52684592&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU20160119(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Troikaa Pharmaceuticals Ltd filed Critical Troikaa Pharmaceuticals Ltd
Publication of CU20160119A7 publication Critical patent/CU20160119A7/es
Publication of CU24444B1 publication Critical patent/CU24444B1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/726Glycosaminoglycans, i.e. mucopolysaccharides
    • A61K31/727Heparin; Heparan
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se relaciona con formulaciones tópicas avanzadas de sales farmacéuticamente aceptables de Heparina que proporcionan penetración transdérmica mejorada. La presente invención proporciona formulaciones líquidas, no pegajosas, claras en las que el fármaco está listo para la absorción y que son adecuadas para administración en la forma de una solución o una pulverización. Las formulaciones tópicas de la presente invención no forman película con escamas o similar al gel sobre la superficie de la piel luego de aplicación tópica.
CU2016000119A 2014-02-10 2015-02-10 Formulaciones tópicas de heparina CU24444B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN475MU2014 2014-02-10
PCT/IB2015/050986 WO2015118512A1 (en) 2014-02-10 2015-02-10 Topical formulations of heparin

Publications (2)

Publication Number Publication Date
CU20160119A7 true CU20160119A7 (es) 2016-10-28
CU24444B1 CU24444B1 (es) 2019-10-04

Family

ID=52684592

Family Applications (1)

Application Number Title Priority Date Filing Date
CU2016000119A CU24444B1 (es) 2014-02-10 2015-02-10 Formulaciones tópicas de heparina

Country Status (25)

Country Link
US (1) US9861655B2 (es)
EP (1) EP3104839B1 (es)
JP (1) JP6275877B2 (es)
KR (1) KR101822133B1 (es)
CN (1) CN106163498A (es)
AP (1) AP2016009350A0 (es)
AR (1) AR099333A1 (es)
AU (1) AU2015213569B2 (es)
CA (1) CA2938388C (es)
CL (1) CL2016001952A1 (es)
CU (1) CU24444B1 (es)
DK (1) DK3104839T3 (es)
DO (1) DOP2016000198A (es)
EA (1) EA032200B1 (es)
EC (1) ECSP16069947A (es)
IL (1) IL246974B (es)
MA (1) MA39304B1 (es)
MX (1) MX357765B (es)
MY (1) MY182620A (es)
NZ (1) NZ722830A (es)
PE (1) PE20161173A1 (es)
PH (1) PH12016501500B1 (es)
TW (1) TWI538697B (es)
UA (1) UA118279C2 (es)
WO (1) WO2015118512A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107115326B (zh) * 2010-04-13 2021-01-22 雷尔玛达治疗股份有限公司 1-甲基-n-(2,6-二甲苯基)-2-哌啶甲酰胺的皮肤用药物组合物及其使用方法
CN112546061B (zh) * 2021-02-25 2021-06-11 中南大学湘雅医院 一种肝素类药物组合物、喷鼻剂及其制备方法及应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3323389A1 (de) * 1983-06-29 1985-01-10 B. Braun Melsungen Ag, 3508 Melsungen Auf schleimhaeute des mundes, der nase und/oder des rachens wirkende arzneimittel auf der basis von heparin und tensiden
JPH02207018A (ja) * 1989-02-07 1990-08-16 Kao Corp 皮膚外用剤
EP0704206B1 (de) 1994-09-30 2002-09-04 MIKA Pharma Gesellschaft für die Entwicklung und Vermarktung pharmazeutischer Produkte mbH Pharmazeutische Zusammensetzung
IT1275955B1 (it) 1995-03-22 1997-10-24 Dompe Spa Formulazioni farmaceutiche in forma di gel tissotropico
JPH10279466A (ja) * 1997-04-07 1998-10-20 Kose Corp 外用剤
US6761903B2 (en) 1999-06-30 2004-07-13 Lipocine, Inc. Clear oil-containing pharmaceutical compositions containing a therapeutic agent
BRPI0101486B1 (pt) 2001-04-17 2017-09-19 Cristália Produtos Químicos Farmacêuticos Ltda. Pharmaceutical composition for topic use containing heparin for the treatment of skin or mucosal injuries caused by burns
CN101583369B (zh) * 2006-11-15 2015-03-11 关节炎缓痛补充剂有限公司 局部制剂及其用途
IT1400232B1 (it) * 2010-05-07 2013-05-24 Advance Holdings Ltd Composizione farmaceutica topica comprendente eparina
RU2013147883A (ru) * 2011-04-01 2015-05-10 Юниверсити Оф Флорида Рисеч Фаундэйшн, Инк. Термочувствительные, мукоадгезивные или кожно-адгезивные и усиливающие проникновение композиции для местной доставки терапевтических средств

Also Published As

Publication number Publication date
MY182620A (en) 2021-01-27
CA2938388C (en) 2018-07-17
MA39304B1 (fr) 2018-12-31
JP6275877B2 (ja) 2018-02-07
EP3104839B1 (en) 2019-11-13
CA2938388A1 (en) 2015-08-13
PE20161173A1 (es) 2016-10-27
US20170165291A1 (en) 2017-06-15
KR101822133B1 (ko) 2018-01-25
EP3104839A1 (en) 2016-12-21
KR20160117529A (ko) 2016-10-10
DOP2016000198A (es) 2016-10-31
CN106163498A (zh) 2016-11-23
US9861655B2 (en) 2018-01-09
MA39304A1 (fr) 2018-01-31
EA032200B1 (ru) 2019-04-30
AR099333A1 (es) 2016-07-13
WO2015118512A1 (en) 2015-08-13
AU2015213569B2 (en) 2018-01-04
PH12016501500A1 (en) 2017-02-06
UA118279C2 (uk) 2018-12-26
CL2016001952A1 (es) 2017-03-10
TW201532631A (zh) 2015-09-01
ECSP16069947A (es) 2018-06-30
IL246974B (en) 2018-07-31
TWI538697B (zh) 2016-06-21
AP2016009350A0 (en) 2016-07-31
DK3104839T3 (da) 2020-01-20
PH12016501500B1 (en) 2017-02-06
NZ722830A (en) 2018-01-26
MX2016010399A (es) 2017-02-23
CU24444B1 (es) 2019-10-04
EA201691596A1 (ru) 2017-01-30
MX357765B (es) 2018-07-23
AU2015213569A1 (en) 2016-08-18
JP2017505344A (ja) 2017-02-16

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