CL2018000525A1 - Derivados de espinosina y métodos de preparación. - Google Patents
Derivados de espinosina y métodos de preparación.Info
- Publication number
- CL2018000525A1 CL2018000525A1 CL2018000525A CL2018000525A CL2018000525A1 CL 2018000525 A1 CL2018000525 A1 CL 2018000525A1 CL 2018000525 A CL2018000525 A CL 2018000525A CL 2018000525 A CL2018000525 A CL 2018000525A CL 2018000525 A1 CL2018000525 A1 CL 2018000525A1
- Authority
- CL
- Chile
- Prior art keywords
- derivatives
- spinosin
- preparation methods
- spinosyne
- preparation
- Prior art date
Links
- 238000002360 preparation method Methods 0.000 title abstract 2
- VGGSULWDCMWZPO-ODEMIOGVSA-N spinosin Chemical class O([C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1C1=C(O)C=2C(=O)C=C(OC=2C=C1OC)C=1C=CC(O)=CC=1)[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O VGGSULWDCMWZPO-ODEMIOGVSA-N 0.000 title 1
- 241000239223 Arachnida Species 0.000 abstract 1
- 241000238631 Hexapoda Species 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 241000244206 Nematoda Species 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N45/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring
- A01N45/02—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring having three carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N2300/00—Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Agronomy & Crop Science (AREA)
- Environmental Sciences (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Saccharide Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicinal Preparation (AREA)
Abstract
<p>Se proveen composiciones y métodos de preparación de derivados de espinosinas. El método produce derivados de espinosina que exhiben actividad hacia insectos, arácnidos, y/o nemátodos y que resultan de utilidad en los mercados agrícola y de la salud animal.</p>
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562214083P | 2015-09-03 | 2015-09-03 | |
| US201662290676P | 2016-02-03 | 2016-02-03 | |
| US201662303015P | 2016-03-03 | 2016-03-03 | |
| US201662303078P | 2016-03-03 | 2016-03-03 | |
| US201662380664P | 2016-08-29 | 2016-08-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2018000525A1 true CL2018000525A1 (es) | 2018-07-13 |
Family
ID=56940400
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2018000527A CL2018000527A1 (es) | 2015-09-03 | 2018-02-27 | Derivados de espinosina y métodos de preparación. |
| CL2018000525A CL2018000525A1 (es) | 2015-09-03 | 2018-02-27 | Derivados de espinosina y métodos de preparación. |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2018000527A CL2018000527A1 (es) | 2015-09-03 | 2018-02-27 | Derivados de espinosina y métodos de preparación. |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US10570166B2 (es) |
| EP (3) | EP3344611B1 (es) |
| JP (3) | JP2018532708A (es) |
| KR (3) | KR20180048871A (es) |
| CN (3) | CN108137529A (es) |
| AU (3) | AU2016317854A1 (es) |
| BR (2) | BR112018004310A2 (es) |
| CA (3) | CA2997540A1 (es) |
| CL (2) | CL2018000527A1 (es) |
| IL (2) | IL257760A (es) |
| MX (3) | MX2018002540A (es) |
| WO (4) | WO2017040763A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10570166B2 (en) | 2015-09-03 | 2020-02-25 | Agrimetis, Llc | Spinosyn derivatives as insecticides |
| JP2020506891A (ja) | 2017-01-13 | 2020-03-05 | アグリメティス，エルエルシー | アジリジンスピノシン誘導体および製造方法 |
| CN119157876A (zh) * | 2017-12-15 | 2024-12-20 | 塔苏斯制药有限公司 | 用于治疗睑炎的异恶唑啉驱虫剂制剂和方法 |
| AR116524A1 (es) * | 2018-10-04 | 2021-05-19 | Elanco Tiergesundheit Ag | Potenciación de tratamiento de helmintos |
| US12502377B2 (en) | 2019-04-04 | 2025-12-23 | Tarsus Pharmaceuticals, Inc. | Method of eradicating ticks that attach to humans using lotilaner formulations |
| BR112023021924A2 (pt) | 2021-04-23 | 2024-01-16 | Acies Bio D O O | Composto, composição, uso de um composto, e, métodos para controlar uma praga e para proteger uma planta contra uma praga de plantas |
| EP4079744B1 (en) | 2021-04-23 | 2025-08-06 | Acies Bio d.o.o. | Novel spinosyn compounds and their use as a pesticide |
| EP4101858A1 (en) | 2021-06-08 | 2022-12-14 | Acies Bio d.o.o. | Novel spinosyn compounds |
Family Cites Families (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1049845B (de) | 1957-01-04 | 1959-02-05 | Consortium Elektrochem Ind | Verfahren zur Herstellung von Carbonylverbindungen |
| US5362634A (en) | 1989-10-30 | 1994-11-08 | Dowelanco | Process for producing A83543 compounds |
| US6030815A (en) | 1995-04-11 | 2000-02-29 | Neose Technologies, Inc. | Enzymatic synthesis of oligosaccharides |
| US5876980A (en) | 1995-04-11 | 1999-03-02 | Cytel Corporation | Enzymatic synthesis of oligosaccharides |
| US5728554A (en) | 1995-04-11 | 1998-03-17 | Cytel Corporation | Enzymatic synthesis of glycosidic linkages |
| US5922577A (en) | 1995-04-11 | 1999-07-13 | Cytel Corporation | Enzymatic synthesis of glycosidic linkages |
| CN1130369C (zh) * | 1995-06-14 | 2003-12-10 | 道农业科学公司 | 对刺糖多孢菌素化合物的合成修饰 |
| US6001981A (en) * | 1996-06-13 | 1999-12-14 | Dow Agrosciences Llc | Synthetic modification of Spinosyn compounds |
| US6143526A (en) | 1998-03-09 | 2000-11-07 | Baltz; Richard H. | Biosynthetic genes for spinosyn insecticide production |
| CZ296136B6 (cs) | 1998-07-02 | 2006-01-11 | Eli Lilly And Company | Prostredek pro péci o vlasy |
| EP1207757B1 (en) | 1999-08-12 | 2005-02-23 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
| US6927210B1 (en) | 1999-08-12 | 2005-08-09 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
| US6919464B1 (en) | 2001-03-21 | 2005-07-19 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
| TWI275592B (en) * | 2001-03-21 | 2007-03-11 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
| EP1492404B1 (en) | 2002-02-19 | 2011-12-28 | Dow AgroSciences LLC | Novel spinosyn-producing polyketide synthases |
| EP1615945B1 (en) | 2003-04-09 | 2011-09-28 | BioGeneriX AG | Glycopegylation methods and proteins/peptides produced by the methods |
| CA2563800C (en) | 2004-04-29 | 2011-06-28 | Eli Lilly And Company | Spinosyns for wound healing |
| WO2010032135A2 (en) | 2008-09-22 | 2010-03-25 | Kritikou, Christine | Spinosyn antifouling compositions, methods of use thereof and articles protected from attachment of biofouling organisms |
| EP2445506B1 (en) | 2009-06-24 | 2014-12-31 | Entarco SA | The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer |
| KR20120098930A (ko) | 2010-01-25 | 2012-09-05 | 일라이 릴리 앤드 캄파니 | 말과 말파리 유충을 내부적으로 억제 또는 처리하기 위한 방법 |
| JP2013542737A (ja) | 2010-11-05 | 2013-11-28 | イーライ リリー アンド カンパニー | 昆虫侵入を阻害するための方法 |
| EP2654757A1 (en) | 2010-12-22 | 2013-10-30 | Entarco SA | The use of spinosyns and spinosyn compositions as local anesthetics and as antiarrhythmic agents |
| KR101960110B1 (ko) | 2010-12-29 | 2019-03-19 | 다우 아그로사이언시즈 엘엘씨 | 곤충 방제 방법 |
| US9631195B2 (en) | 2011-12-28 | 2017-04-25 | Dow Agrosciences Llc | Identification and characterization of the spinactin biosysnthesis gene cluster from spinosyn producing saccharopolyspora spinosa |
| US9895388B1 (en) * | 2012-07-27 | 2018-02-20 | ParaPRO | Methods and compositions useful for controlling cutaneous mites |
| CN102977166B (zh) * | 2012-12-05 | 2015-07-29 | 湖南化工研究院 | 13-硫醚取代多杀菌素衍生物及其制备方法 |
| ES2616114T3 (es) * | 2013-01-22 | 2017-06-09 | Actelion Pharmaceuticals Ltd. | Derivados de amida heterocíclica como antagonistas del receptor P2X7 |
| MX2016005308A (es) | 2013-10-22 | 2016-08-08 | Dow Agrosciences Llc | Composiciones pesticidas sinergicas y metodos relacionados. |
| US9873639B1 (en) | 2015-07-17 | 2018-01-23 | Joe Doccola | Agricultural biomass as a matrix for release of plant active compounds |
| US10570166B2 (en) | 2015-09-03 | 2020-02-25 | Agrimetis, Llc | Spinosyn derivatives as insecticides |
-
2016
- 2016-09-01 US US15/757,204 patent/US10570166B2/en active Active
- 2016-09-01 WO PCT/US2016/049870 patent/WO2017040763A1/en not_active Ceased
- 2016-09-01 BR BR112018004310A patent/BR112018004310A2/pt not_active Application Discontinuation
- 2016-09-01 CN CN201680061132.2A patent/CN108137529A/zh active Pending
- 2016-09-01 MX MX2018002540A patent/MX2018002540A/es unknown
- 2016-09-01 CA CA2997540A patent/CA2997540A1/en not_active Abandoned
- 2016-09-01 EP EP16767084.3A patent/EP3344611B1/en active Active
- 2016-09-01 EP EP16767424.1A patent/EP3344612B1/en active Active
- 2016-09-01 MX MX2018002538A patent/MX2018002538A/es unknown
- 2016-09-01 KR KR1020187008942A patent/KR20180048871A/ko not_active Withdrawn
- 2016-09-01 WO PCT/US2016/049879 patent/WO2017040769A1/en not_active Ceased
- 2016-09-01 AU AU2016317854A patent/AU2016317854A1/en not_active Abandoned
- 2016-09-01 JP JP2018512331A patent/JP2018532708A/ja not_active Withdrawn
- 2016-09-01 BR BR112018004313A patent/BR112018004313A2/pt not_active Application Discontinuation
- 2016-09-01 CA CA2997499A patent/CA2997499A1/en not_active Abandoned
- 2016-09-01 CN CN201680056085.2A patent/CN108026063A/zh active Pending
- 2016-09-01 KR KR1020187008943A patent/KR20180050340A/ko not_active Withdrawn
- 2016-09-01 AU AU2016317848A patent/AU2016317848A1/en not_active Abandoned
- 2016-09-01 US US15/757,317 patent/US10717756B2/en active Active
- 2016-09-01 JP JP2018512332A patent/JP2018531912A/ja not_active Withdrawn
- 2016-09-02 AU AU2016315860A patent/AU2016315860A1/en not_active Abandoned
- 2016-09-02 JP JP2018512326A patent/JP2018532707A/ja not_active Withdrawn
- 2016-09-02 WO PCT/US2016/050034 patent/WO2017040882A1/en not_active Ceased
- 2016-09-02 EP EP16766747.6A patent/EP3344610B1/en active Active
- 2016-09-02 KR KR1020187008941A patent/KR20180041755A/ko not_active Withdrawn
- 2016-09-02 WO PCT/US2016/050028 patent/WO2017040878A1/en not_active Ceased
- 2016-09-02 CN CN201680057361.7A patent/CN108137528A/zh active Pending
- 2016-09-02 US US15/757,307 patent/US10711026B2/en active Active
- 2016-09-02 CA CA2997639A patent/CA2997639A1/en not_active Abandoned
- 2016-09-02 MX MX2018002539A patent/MX2018002539A/es unknown
-
2018
- 2018-02-27 IL IL257760A patent/IL257760A/en unknown
- 2018-02-27 CL CL2018000527A patent/CL2018000527A1/es unknown
- 2018-02-27 IL IL257759A patent/IL257759A/en unknown
- 2018-02-27 CL CL2018000525A patent/CL2018000525A1/es unknown
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